日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Lithocholic acid derivatives as potent modulators of the nuclear receptor RORγt

石胆酸衍生物作为核受体RORγt的有效调节剂

Somaya A Abdel-Rahman ,Simone Brogi ,Moustafa T Gabr

Synthesis, enzyme inhibition assay, and molecular modeling study of novel pyrazolines linked to 4-methylsulfonylphenyl scaffold: antitumor activity and cell cycle analysis

新型吡唑啉与 4-甲基磺酰基苯基支架的合成、酶抑制试验及分子建模研究:抗肿瘤活性和细胞周期分析

Alaa A-M Abdel-Aziz, Adel S El-Azab, Simone Brogi, Rezk R Ayyad, Hamad M Alkahtani, Hatem A Abuelizz, Ibrahim A Al-Suwaidan, Abdulrahman M Al-Obaid

Antitumor Activity and Multi-Target Mechanism of Phenolic Schiff Bases Bearing Methanesulfonamide Fragments: Cell Cycle Analysis and a Molecular Modeling Study

含甲磺酰胺片段的酚醛席夫碱的抗肿瘤活性和多靶点机制:细胞周期分析和分子建模研究

Alaa A-M Abdel-Aziz, Adel S El-Azab, Simone Brogi, Rezk R Ayyad, Ibrahim A Al-Suwaidan, Mohamed Hefnawy

Novel analgesic/anti-inflammatory agents: 1,5-Diarylpyrrole nitrooxyethyl sulfides and related compounds as Cyclooxygenase-2 inhibitors containing a nitric oxide donor moiety endowed with vasorelaxant properties

新型镇痛/抗炎剂:1,5-二芳基吡咯硝基氧乙基硫化物和相关化合物作为环氧合酶-2抑制剂,含有具有血管舒张特性的一氧化氮供体部分

Mario Saletti, Samuele Maramai, Annalisa Reale, Marco Paolino, Simone Brogi, Angela Di Capua, Andrea Cappelli, Gianluca Giorgi, Danilo D'Avino, Antonietta Rossi, Carla Ghelardini, Lorenzo Di Cesare Mannelli, Roccaldo Sardella, Andrea Carotti, Gerald Woelkart, Burkhard Klösch, Chiara Bigogno, Giulio

Design and synthesis of multifunctional microtubule targeting agents endowed with dual pro-apoptotic and anti-autophagic efficacy

具有双重促凋亡和抗自噬功效的多功能微管靶向药物的设计与合成

Giuseppe Campiani, Tuhina Khan, Cristina Ulivieri, Leopoldo Staiano, Chiara Papulino, Stefania Magnano, Seema Nathwani, Anna Ramunno, Daniel Lucena-Agell, Nicola Relitti, Stefano Federico, Luca Pozzetti, Gabriele Carullo, Alice Casagni, Simone Brogi, Francesca Vanni, Paola Galatello, Magda Ghanim, N

Pro-Apoptotic Activity of the Marine Sponge Dactylospongia elegans Metabolites Pelorol and 5- epi-Ilimaquinone on Human 501Mel Melanoma Cells

海洋海绵Dactylospongia elegans代谢物Pelorol和5-表-Ilimaquinone对人类501Mel黑色素瘤细胞的促凋亡活性

Sara Carpi, Egeria Scoditti, Beatrice Polini, Simone Brogi, Vincenzo Calderone, Peter Proksch, Sherif S Ebada, Paola Nieri

Crystal structures of Schistosoma mansoni histone deacetylase 8 reveal a novel binding site for allosteric inhibitors

曼氏血吸虫组蛋白去乙酰化酶 8 的晶体结构揭示了变构抑制剂的新型结合位点

Fulvio Saccoccia, Luca Pozzetti, Roberto Gimmelli, Stefania Butini, Alessandra Guidi, Giuliana Papoff, Marialaura Giannaccari, Simone Brogi, Viviana Scognamiglio, Sandra Gemma, Giovina Ruberti, Giuseppe Campiani

Design and Synthesis of Oligopeptidic Parvulin Inhibitors

寡肽类 Parvulin 抑制剂的设计和合成

Nicola Relitti, A Prasanth Saraswati, Gabriele Carullo, Alessandro Papa, Alessandra Monti, Rosaria Benedetti, Eugenia Passaro, Simone Brogi, Vincenzo Calderone, Stefania Butini, Sandra Gemma, Lucia Altucci, Giuseppe Campiani, Nunzianna Doti

Resveratrol-like Compounds as SIRT1 Activators

白藜芦醇类化合物作为 SIRT1 激活剂

Lidia Ciccone, Eugenia Piragine, Simone Brogi, Caterina Camodeca, Raffaele Fucci, Vincenzo Calderone, Susanna Nencetti, Alma Martelli, Elisabetta Orlandini

Harnessing the Role of HDAC6 in Idiopathic Pulmonary Fibrosis: Design, Synthesis, Structural Analysis, and Biological Evaluation of Potent Inhibitors

利用 HDAC6 在特发性肺纤维化中的作用:强效抑制剂的设计、合成、结构分析和生物学评估

Giuseppe Campiani, Caterina Cavella, Jeremy D Osko, Margherita Brindisi, Nicola Relitti, Simone Brogi, A Prasanth Saraswati, Stefano Federico, Giulia Chemi, Samuele Maramai, Gabriele Carullo, Benedikt Jaeger, Alfonso Carleo, Rosaria Benedetti, Federica Sarno, Stefania Lamponi, Paola Rottoli, Elena B