日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, Synthesis, and Pharmacological Characterization of a Potent Soluble Epoxide Hydrolase Inhibitor for the Treatment of Acute Pancreatitis

用于治疗急性胰腺炎的强效可溶性环氧化物水解酶抑制剂的设计、合成和药理学表征

Simona Musella, Danilo D'Avino, Lukas Klaus Peltner, Veronica Di Sarno, Ida Cerqua, Fabrizio Merciai, Vincenzo Vestuto, Tania Ciaglia, Gerardina Smaldone, Francesca Di Matteo, Simone Di Micco, Valeria Napolitano, Giuseppe Bifulco, Giacomo Pepe, Eduardo Maria Sommella, Manuela Giovanna Basilicata, Gi

Discovery and Optimization of Indoline-Based Compounds as Dual 5-LOX/sEH Inhibitors: In Vitro and In Vivo Anti-Inflammatory Characterization

发现和优化吲哚啉基化合物作为双重 5-LOX/sEH 抑制剂:体外和体内抗炎特性

Ida Cerqua, Simona Musella, Lukas Klaus Peltner, Danilo D'Avino, Veronica Di Sarno, Elisabetta Granato, Vincenzo Vestuto, Rita Di Matteo, Simona Pace, Tania Ciaglia, Rossella Bilancia, Gerardina Smaldone, Francesca Di Matteo, Simone Di Micco, Giuseppe Bifulco, Giacomo Pepe, Manuela Giovanna Basilica

Rational design of the zonulin inhibitor AT1001 derivatives as potential anti SARS-CoV-2

zonulin 抑制剂 AT1001 衍生物作为潜在抗 SARS-CoV-2 药物的合理设计

Simone Di Micco, Rahila Rahimova, Marina Sala, Maria C Scala, Giovanni Vivenzio, Simona Musella, Graciela Andrei, Kim Remans, Léa Mammri, Robert Snoeck, Giuseppe Bifulco, Francesca Di Matteo, Vincenzo Vestuto, Pietro Campiglia, José A Márquez, Alessio Fasano

In Silico Identification and In Vitro Evaluation of New ABCG2 Transporter Inhibitors as Potential Anticancer Agents

通过计算机模拟鉴定和体外评估新型 ABCG2 转运蛋白抑制剂作为潜在抗癌剂的作用

Simone Di Micco, Veronica Di Sarno, Martina Rossi, Vincenzo Vestuto, Takumi Konno, Sara Novi, Mario Felice Tecce, Valeria Napolitano, Tania Ciaglia, Andrea Vitale, Isabel Maria Gomez-Monterrey, Giuseppe Bifulco, Alessia Bertamino, Carmine Ostacolo, Paolo Blasi, Alessio Fasano, Pietro Campiglia, Simo

Overcome Chemoresistance: Biophysical and Structural Analysis of Synthetic FHIT-Derived Peptides

克服化学耐药性:合成 FHIT 衍生肽的生物物理和结构分析

Maria Carmina Scala, Simone Di Micco, Delia Lanzillotta, Simona Musella, Veronica Di Sarno, Barbara Parrino, Stella Maria Casciofierro, Giuseppe Bifulco, Francesco Trapasso, Pietro Campiglia, Marina Sala

Peptide Derivatives of the Zonulin Inhibitor Larazotide (AT1001) as Potential Anti SARS-CoV-2: Molecular Modelling, Synthesis and Bioactivity Evaluation

连蛋白抑制剂拉唑肽 (AT1001) 的肽衍生物作为潜在抗 SARS-CoV-2 药物:分子建模、合成和生物活性评估

Simone Di Micco, Simona Musella, Marina Sala, Maria C Scala, Graciela Andrei, Robert Snoeck, Giuseppe Bifulco, Pietro Campiglia, Alessio Fasano

Identification by Inverse Virtual Screening of magnolol-based scaffold as new tankyrase-2 inhibitors

通过逆向虚拟筛选鉴定基于厚朴酚的支架作为新型 tankyrase-2 抑制剂

Simone Di Micco, Luana Pulvirenti, Ines Bruno, Stefania Terracciano, Alessandra Russo, Maria C Vaccaro, Dafne Ruggiero, Vera Muccilli, Nunzio Cardullo, Corrado Tringali, Raffaele Riccio, Giuseppe Bifulco

Lactoferrin-derived Peptides Active towards Influenza: Identification of Three Potent Tetrapeptide Inhibitors

乳铁蛋白衍生的抗流感肽:三种有效四肽抑制剂的鉴定

Maria Carmina Scala, Marina Sala, Agostina Pietrantoni, Antonia Spensiero, Simone Di Micco, Mariangela Agamennone, Alessia Bertamino, Ettore Novellino, Giuseppe Bifulco, Isabel M Gomez-Monterrey, Fabiana Superti, Pietro Campiglia