日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and biological activity of conformationally restricted indole-based inhibitors of neurotropic alphavirus replication: Generation of a three-dimensional pharmacophore

构象受限的吲哚类神经嗜性甲病毒复制抑制剂的合成及生物活性:三维药效团的构建

Barraza, Scott J; Sindac, Janice A; Dobry, Craig J; Delekta, Philip C; Lee, Pil H; Miller, David J; Larsen, Scott D

Discovery, Radiolabeling, and Evaluation of Subtype-Selective Inhibitors for Positron Emission Tomography Imaging of Brain Phosphodiesterase-4D

脑磷酸二酯酶-4D正电子发射断层扫描成像亚型选择性抑制剂的发现、放射性标记和评价

Wakabayashi, Yuichi; Telu, Sanjay; Dick, Rachel M; Fujita, Masahiro; Ooms, Maarten; Morse, Cheryl L; Liow, Jeih-San; Hong, Jinsoo S; Gladding, Robert L; Manly, Lester S; Zoghbi, Sami S; Mo, Xuesheng; D'Amato, Emily C; Sindac, Janice A; Nugent, Richard A; Marron, Brian E; Gurney, Mark E; Innis, Robert B; Pike, Victor W

Design and Synthesis of Selective Phosphodiesterase 4D (PDE4D) Allosteric Inhibitors for the Treatment of Fragile X Syndrome and Other Brain Disorders

选择性磷酸二酯酶4D (PDE4D) 变构抑制剂的设计与合成及其在脆性X综合征和其他脑部疾病治疗中的应用

Gurney, Mark E; Nugent, Richard A; Mo, Xuesheng; Sindac, Janice A; Hagen, Timothy J; Fox, David 3rd; O'Donnell, James M; Zhang, Chong; Xu, Ying; Zhang, Han-Ting; Groppi, Vincent E; Bailie, Marc; White, Ronald E; Romero, Donna L; Vellekoop, A Samuel; Walker, Joel R; Surman, Matthew D; Zhu, Lei; Campbell, Robert F

Optimization of novel indole-2-carboxamide inhibitors of neurotropic alphavirus replication

优化新型吲哚-2-甲酰胺类神经嗜性甲病毒复制抑制剂

Sindac, Janice A; Barraza, Scott J; Dobry, Craig J; Xiang, Jianming; Blakely, Pennelope K; Irani, David N; Keep, Richard F; Miller, David J; Larsen, Scott D

Novel inhibitors of neurotropic alphavirus replication that improve host survival in a mouse model of acute viral encephalitis

新型神经嗜性甲病毒复制抑制剂可提高急性病毒性脑炎小鼠模型中的宿主存活率

Sindac, Janice A; Yestrepsky, Bryan D; Barraza, Scott J; Bolduc, Kyle L; Blakely, Pennelope K; Keep, Richard F; Irani, David N; Miller, David J; Larsen, Scott D

Erratum: “Model for the fast estimation of basis set superposition error in biomolecular systems” [J. Chem. Phys. 135, 144110 (2011)]

勘误:“生物分子系统中基组叠加误差快速估计模型”[J. Chem. Phys. 135, 144110 (2011)]

Delekta, Phillip C; Dobry, Craig J; Sindac, Janice A; Barraza, Scott J; Blakely, Pennelope K; Xiang, Jianming; Kirchhoff, Paul D; Keep, Richard F; Irani, David N; Larsen, Scott D; Miller, David J; Kim, Jaegil; Straub, John E; Faver, John C; Zheng, Zheng; Merz, Kenneth M Jr