日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Isoniazid-rhodanine molecular hybrids: design, synthesis, antimycobacterial activity and computational validation

异烟肼-罗丹宁分子杂合物:设计、合成、抗分枝杆菌活性及计算验证

Kumar, Gobind; Mishra, Sahil; Seboletswe, Pule; Manhas, Neha; Ghumran, Safiyah; Roquet-Banères, Françoise; Kremer, Laurent; Bhargava, Gaurav; Singh, Parvesh

Rational Design and Antimycobacterial Evaluation of Aryl Sulfonamide-Linked Isoniazid Hydrazones Against Mycobacterium Tuberculosis

合理设计并评价芳基磺酰胺连接的异烟肼腙类化合物对结核分枝杆菌的抗结核活性

Kadima, Mukanda Gedeon; Mishra, Sahil; Kumar, Gobind; Seboletswe, Pule; Kajee, Afsana; Ankit; Roquet-Banères, Françoise; Foubert, Maëlle; Kremer, Laurent; Karpoormath, Rajshekhar; Singh, Parvesh

A Systematic Review of Synthetic and Anticancer and Antimicrobial Activity of Quinazoline/Quinazolin-4-one Analogues

喹唑啉/喹唑啉-4-酮类似物的合成、抗癌和抗菌活性的系统综述

Manhas, Neha; Kumar, Gobind; Dhawan, Sanjeev; Makhanya, Talent; Singh, Parvesh

One-Pot Synthesis of Novel β-Carboline-{α-Acylaminoamide}-Bisindole Derivatives: Antibacterial Evaluation, Molecular Docking, and Density Functional Theory Studies

新型β-咔啉-{α-酰基氨基酰胺}-双吲哚衍生物的一锅法合成:抗菌活性评价、分子对接和密度泛函理论研究

Atri, Ankit Kumar; Khullar, Lavanya; Kumar, Gobind; Mishra, Sahil; Dua, Tamanna; Singh, Vinay; Harjai, Kusum; Singh, Parvesh; Singh, Vasundhara

Rapid and Environmentally-Friendly Synthesis of Thiazolidinone Analogues in Deep Eutectic Solvent Complemented with Computational Studies

利用计算研究,在低共熔溶剂中快速、环保地合成噻唑烷酮类似物

Kumar, Gobind; Seboletswe, Pule; Gcabashe, Nontobeko; Dhawan, Sanjeev; Manhas, Neha; Bhargava, Gaurav; Kumar, Rupesh; Singh, Parvesh

Benzylidenehydrazine Derivatives: Synthesis, Antidiabetic Evaluation, Antioxidation, Mode of Inhibition, DFT and Molecular Docking Studies

亚苄基肼衍生物:合成、抗糖尿病活性评价、抗氧化活性、抑制机制、DFT计算和分子对接研究

Seboletswe, Pule; Kumar, Gobind; Gcabashe, Nontobeko; Olofinsan, Kolawole; Islam, Shahidul; Idris, ALmahi; Singh, Parvesh

DES-Promoted Synthesis of 3,4-Dihydropyrimidinones and Their Antidiabetic and Antioxidant Evaluation Supported With Computational Studies

DES促进的3,4-二氢嘧啶酮的合成及其抗糖尿病和抗氧化活性评价(基于计算研究)

Kumar, Gobind; Mishra, Sahil; Seboletswe, Pule; Gcabashe, Nontobeko; Gummidi, Lalitha; Manhas, Neha; Makhanya, Talent; Bhargava, Gaurav; Idris, Almahi; Islam, Md Shahidul; Singh, Parvesh

Antidiabetic Evaluation of New Pyrimidine-Thiazoline Hybrids Endorsed With Enzyme Kinetic Studies and Computational Analysis

新型嘧啶-噻唑啉杂合物的抗糖尿病活性评价:酶动力学研究和计算分析的支持

Kumar, Gobind; Seboletswe, Pule; Manhas, Neha; Ghumran, Safiyah; Gcabashe, Nontobeko; Bhargava, Gaurav; Idris, Almahi; Islam, Md Shahidul; Singh, Parvesh

Rationally Designed InhA Inhibitors: A Comparative Anti-Tubercular Activity Study of Sulfonate Esters of Isoniazid Hydrazones and Their Structurally Flexible Benzyl Analogues

合理设计的InhA抑制剂:异烟肼腙磺酸酯及其结构灵活的苄基类似物的抗结核活性比较研究

Kadima, Mukanda Gedeon; Mishra, Sahil; Kumar, Gobind; Seboletswe, Pule; Roquet-Banères, Françoise; Foubert, Maëlle; Kremer, Laurent; Karpoormath, Rajshekhar; Singh, Parvesh

A density functional theory study of a series of symmetric dibenzylideneacetone analogues as potential chemical UV-filters

利用密度泛函理论研究一系列对称的二亚苄基丙酮类似物作为潜在的化学紫外线过滤剂

Magaji, Buhari; Singh, Parvesh; Skelton, Adam A; Martincigh, Bice S