日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Target Class Ligandability Evaluation of WD40 Repeat-Containing Proteins

WD40重复序列蛋白的靶向配体结合能力评价

Ackloo, Suzanne; Li, Fengling; Szewczyk, Magda; Seitova, Almagul; Loppnau, Peter; Zeng, Hong; Xu, Jin; Ahmad, Shabbir; Arnautova, Yelena A; Baghaie, A J; Beldar, Serap; Bolotokova, Albina; Centrella, Paolo A; Chau, Irene; Clark, Matthew A; Cuozzo, John W; Dehghani-Tafti, Saba; Disch, Jeremy S; Dong, Aiping; Dumas, Antoine; Feng, Jianwen A; Ghiabi, Pegah; Gibson, Elisa; Gilmer, Justin; Goldman, Brian; Green, Stuart R; Guié, Marie-Aude; Guilinger, John P; Harms, Nathan; Herasymenko, Oleksandra; Houliston, Scott; Hutchinson, Ashley; Kearnes, Steven; Keefe, Anthony D; Kimani, Serah W; Kramer, Trevor; Kutera, Maria; Kwak, Haejin A; Lento, Cristina; Li, Yanjun; Liu, Jenny; Loup, Joachim; Machado, Raquel A C; Mulhern, Christopher J; Perveen, Sumera; Righetto, Germanna L; Riley, Patrick; Shrestha, Suman; Sigel, Eric A; Silva, Madhushika; Sintchak, Michael D; Slakman, Belinda L; Taylor, Rhys D; Thompson, James; Torng, Wen; Underkoffler, Carl; von Rechenberg, Moritz; Walsh, Ryan T; Watson, Ian; Wilson, Derek J; Wolf, Esther; Yadav, Manisha; Yazdi, Aliakbar K; Zhang, Junyi; Zhang, Ying; Santhakumar, Vijayaratnam; Edwards, Aled M; Barsyte-Lovejoy, Dalia; Schapira, Matthieu; Brown, Peter J; Halabelian, Levon; Arrowsmith, Cheryl H

Mechanistic study of Uba5 enzyme and the Ufm1 conjugation pathway

Uba5 酶与 Ufm1 结合途径的机制研究

James M Gavin, Kara Hoar, Qing Xu, Jingya Ma, Yafang Lin, Jiejin Chen, Wei Chen, Frank J Bruzzese, Sean Harrison, William D Mallender, Nancy J Bump, Michael D Sintchak, Neil F Bence, Ping Li, Lawrence R Dick, Alexandra E Gould, Jesse J Chen

Sequence analysis of β-subunit genes of the 20S proteasome in patients with relapsed multiple myeloma treated with bortezomib or dexamethasone

对接受硼替佐米或地塞米松治疗的复发性多发性骨髓瘤患者的20S蛋白酶体β亚基基因进行序列分析

Lichter, David I; Danaee, Hadi; Pickard, Michael D; Tayber, Olga; Sintchak, Michael; Shi, Hongliang; Richardson, Paul G; Cavenagh, Jamie; Bladé, Joan; Façon, Thierry; Niesvizky, Ruben; Alsina, Melissa; Dalton, William; Sonneveld, Pieter; Lonial, Sagar; van de Velde, Helgi; Ricci, Deborah; Esseltine, Dixie-Lee; Trepicchio, William L; Mulligan, George; Anderson, Kenneth C

Mechanistic studies of substrate-assisted inhibition of ubiquitin-activating enzyme by adenosine sulfamate analogues

腺苷氨基磺酸盐类似物底物辅助抑制泛素活化酶的机制研究

Jesse J Chen, Christopher A Tsu, James M Gavin, Michael A Milhollen, Frank J Bruzzese, William D Mallender, Michael D Sintchak, Nancy J Bump, Xiaofeng Yang, Jingya Ma, Huay-Keng Loke, Qing Xu, Ping Li, Neil F Bence, James E Brownell, Lawrence R Dick

Characterization of a new series of non-covalent proteasome inhibitors with exquisite potency and selectivity for the 20S beta5-subunit

对一系列新型非共价蛋白酶体抑制剂进行表征,这些抑制剂对 20S β5 亚基具有极高的效力和选择性。

Blackburn, Christopher; Gigstad, Kenneth M; Hales, Paul; Garcia, Khristofer; Jones, Matthew; Bruzzese, Frank J; Barrett, Cynthia; Liu, Jane X; Soucy, Teresa A; Sappal, Darshan S; Bump, Nancy; Olhava, Edward J; Fleming, Paul; Dick, Lawrence R; Tsu, Christopher; Sintchak, Michael D; Blank, Jonathan L

Endogenous spartin (SPG20) is recruited to endosomes and lipid droplets and interacts with the ubiquitin E3 ligases AIP4 and AIP5

内源性斯巴汀(SPG20)被募集到内体和脂滴中,并与泛素E3连接酶AIP4和AIP5相互作用。

Bastea, Ligia I; Döppler, Heike; Pearce, Sarah E; Durand, Nisha; Spratley, Samantha J; Storz, Peter; Nordin, N; Guskov, A; Phua, T; Sahaf, N; Xia, Y; Lu, S; Eshaghi, H; Eshaghi, S; O'Leary, B; Rao, S K; Plaxton, W C; Blackburn, C; Gigstad, K M; Hales, P; Garcia, K; Jones, M; Bruzzese, F J; Barrett, C; Liu, J X; Soucy, T A; Sappal, D S; Bump, N; Olhava, E J; Fleming, P; Dick, L R; Tsu, C; Sintchak, M D; Blank, J L; Nomikos, M; Elgmati, K; Theodoridou, M; Calver, B L; Cumbes, B; Nounesis, G; Swann, K; Lai, F A; Brand, M D; Nicholls, D G; Edwards, T L; Clowes, V E; Tsang, H T H; Connell, J W; Sanderson, C M; Luzio, J P; Reid, E