Identification of alkynyl nicotinamide HSN748 as a RET solvent-front mutant inhibitor with intracranial efficacy.
鉴定炔基烟酰胺 HSN748 为具有颅内疗效的 RET 溶剂前沿突变体抑制剂
期刊:RSC Medicinal Chemistry
影响因子:3.6
doi:10.1039/d5md00245a
Khatri Ujjwol, Dayal Neetu, Owusu Kofi B, Hunjan Mandeep Kaur, Pandey Shriya, Harper Haley Anne, McMahan Carli, Elzey Bennett D, Shen Tao, Hu Xueqing, Evans Kurt W, El-Sheikh Ahmed, Jo Seong Jun, Holtsberg Frederick W, Aman M Javad, Meric-Bernstam Funda, Woo Sukyung, Sintim Herman O, Wu Jie