日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

N‑Alkyl and N‑Aryl Aminopyrazole Spirocarbamates: A Two-Pronged Lead Optimization Strategy to Identify Orally Bioavailable Plasma Kallikrein Inhibitors

N-烷基和N-芳基氨基吡唑螺环氨基甲酸酯:一种用于筛选口服生物利用度高的血浆激肽释放酶抑制剂的双管齐下先导化合物优化策略

Merchant, Rohan R; Chernyak, Natalia; Lopez, Jovan A; Sharp, Phillip P; Mandal, Mihir; He, Jiafang; Hruza, Alan; Rearden, Paul; Tatosian, Daniel A; Esmay, Joel; Yang, Song; Cheng, Alan C; Ellsworth, Ken; Ogawa, Aimie; Piou, Tiffany; Fier, Patrick; Hicks, Jacqueline; Sinz, Christopher; Ogawa, Anthony K

HypoxyStat, a small-molecule form of hypoxia therapy that increases oxygen-hemoglobin affinity.

HypoxyStat 是一种小分子缺氧疗法,可提高氧合血红蛋白的亲和力

Blume Skyler Y, Garg Ankur, Martí-Mateos Yolanda, Midha Ayush D, Chew Brandon T L, Lin Baiwei, Yu Cecile, Dick Ryan, Lee Patrick S, Situ Eva, Sarwaikar Richa, Green Eric, Ramanan Vyas, Grotenbreg Gijsbert, Hoek Maarten, Sinz Christopher, Jain Isha H

Discovery of Orally Bioavailable and Liver-Targeted Hypoxia-Inducible Factor Prolyl Hydroxylase (HIF-PHD) Inhibitors for the Treatment of Anemia

发现口服生物利用度高且靶向肝脏的缺氧诱导因子脯氨酰羟化酶 (HIF-PHD) 抑制剂用于治疗贫血

Liu, Ping; Wang, Liping; DuBois, Byron G; Colandrea, Vincent J; Liu, Rongqiang; Cai, Jiaqiang; Du, Xiaoxing; Quan, Weiguo; Morris, William; Bai, Jianwu; Bishwokarma, Bimjhana; Cheng, Mangeng; Piesvaux, Jennifer; Ray, Kallol; Alpert, Carla; Chiu, Chi-Sung; Zielstorff, Mark; Metzger, Joseph M; Yang, Liming; Leung, Dennis; Alleyne, Candice; Vincent, Stella H; Pucci, Vincenzo; Li, Xiaofang; Crespo, Alejandro; Stickens, Dominique; Hale, Jeffrey J; Ujjainwalla, Feroze; Sinz, Christopher J

Total synthesis of diazonamide A

重氮酰胺A的全合成

Knowles, Robert R; Carpenter, Joseph; Blakey, Simon B; Kayano, Akio; Mangion, Ian K; Sinz, Christopher J; Macmillan, David W C

Enantioselective organocatalytic construction of pyrroloindolines by a cascade addition-cyclization strategy: synthesis of (-)-flustramine B

通过级联加成-环化策略对映选择性有机催化构建吡咯并吲哚啉:(-)-氟司他明B的合成

Austin, Joel F; Kim, Sung-Gon; Sinz, Christopher J; Xiao, Wen-Jing; MacMillan, David W C