Discovery of Orally Bioavailable and Liver-Targeted Hypoxia-Inducible Factor Prolyl Hydroxylase (HIF-PHD) Inhibitors for the Treatment of Anemia
发现口服生物利用度高且靶向肝脏的缺氧诱导因子脯氨酰羟化酶 (HIF-PHD) 抑制剂用于治疗贫血
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.8b00274
Liu, Ping; Wang, Liping; DuBois, Byron G; Colandrea, Vincent J; Liu, Rongqiang; Cai, Jiaqiang; Du, Xiaoxing; Quan, Weiguo; Morris, William; Bai, Jianwu; Bishwokarma, Bimjhana; Cheng, Mangeng; Piesvaux, Jennifer; Ray, Kallol; Alpert, Carla; Chiu, Chi-Sung; Zielstorff, Mark; Metzger, Joseph M; Yang, Liming; Leung, Dennis; Alleyne, Candice; Vincent, Stella H; Pucci, Vincenzo; Li, Xiaofang; Crespo, Alejandro; Stickens, Dominique; Hale, Jeffrey J; Ujjainwalla, Feroze; Sinz, Christopher J