日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

African Natural Products Database (ANPDB): A resource for exploring the therapeutic potential of natural compounds from Africa

非洲天然产物数据库(ANPDB):一个用于探索非洲天然化合物治疗潜力的资源库

Betow, Jude Y; Qaseem, Ammar; Bekono, Boris D; Feng, Yue; Moumbock, Aurélien F A; Simoben, Conrad V; Babiaka, Smith B; Tanyi, Solange A; Shu, Vanessa A; Ndi, Ariane T; Onguéné, Pascal Amoa; Metuge, Clovis S; Akame, Simeon; Eni, Donatus B; Namba-Nzanguim, Cyril T; Tjegbe, Mathieu J M; Dikande, Marianka N L; Akeh, Patience T; Balgah, Sounders Jr; Meh, Cyprian D; Ibezim, Akachukwu; Tabi, Idris F; Malange, Yvette I; Ndingkokhar, Bakoh; Njume, Leonel E; Telukunta, Kiran K; Amrani, Said; Ebob, Oyere T; Sippl, Wolfgang; Günther, Stefan; Ntie-Kang, Fidele

Insights into the Design of MYC-Targeting Proteolysis Targeting Chimeras (PROTACs)

MYC靶向蛋白水解靶向嵌合体(PROTACs)的设计见解

Alfayomy, Abdallah M; Hagemann, Sven; Schmidt, Matthias; Fouad, Ali; El-Zahabi, Mohamed Ayman; Hüttelmaier, Stefan; Sippl, Wolfgang

Stimulated Raman Spectroscopy for Intraoperative Glioblastoma Diagnosis-A Complementary Tool to Frozen Section?

受激拉曼光谱法在术中胶质母细胞瘤诊断中的应用——冰冻切片的补充工具?

Sippl, Christoph; Stark, Felix; Schneider, K Isabel; Reyes Medina, Bernardo; Schulz-Schaeffer, Walter; Brinkmann, Maximilian; Neumann, Felix; Droop, Ramon; Ullmann, Steffen; Würthwein, Thomas; Hellwig, Tim; Hoffmann, Lucas; Monfroy, Nathan; Khafaji, Fatemeh; Saffour, Safwan; Gaber, Karim; Linsler, Stefan

Capsaicin-Inspired Hydroxamate Hybrids as Selective HDAC6 Inhibitors with Antiproliferative Activity in Hematological Malignancies

辣椒素衍生的羟肟酸酯杂合物作为选择性 HDAC6 抑制剂,在血液恶性肿瘤中具有抗增殖活性

Gimenez Borges, Lara; Alves, Thais Nascimento de Oliveira; Vassiliades, Sandra Valeria; Carlos, Jorge Antonio Elias Godoy; Waitman, Karoline de Barros; Hilscher, Sebastian; Schutkowski, Mike; Sippl, Wolfgang; Tavares, Maurício Temotheo; Toledo, Monica Franco Zannini Junqueira; Costa-Lotufo, Letícia Veras; Kronenberger, Thales; Machado-Neto, João Agostinho; Parise-Filho, Roberto

Bisamidine Derivatives as Candidates for Tegumentary Leishmaniasis Therapy: Phenotypic Screening in Infection of Macrophages and Mechanistic Insights with Dual RNA-seq

双脒衍生物作为皮肤利什曼病治疗候选药物:巨噬细胞感染表型筛选及双重RNA测序机制研究

Agripino, Joice; Tahira, Ana C; de Souza, Luciana Ângelo; Silva E Bastos, Matheus; Sauer, Benjamin; Schmidt, Matthias; Bressan, Gustavo Costa; de Souza Vasconcellos, Raphael; Sippl, Wolfgang; Pierce, Raymond; Sena Amaral, Murilo; Verjovski-Almeida, Sergio; Rangel Fietto, Juliana Lopes

AI-Based Prediction of PROTAC- and Molecular Glue-Mediated Ternary Complexes: A Comparative Evaluation of AlphaFold 3 and Boltz-2

基于人工智能的PROTAC和分子胶介导的三元复合物预测:AlphaFold 3和Boltz-2的比较评估

Riepenhausen, Lino; Sarnow, Anne-Christin; Robaa, Dina; Sippl, Wolfgang

Accuracy of indocyanine green videoangiography in predicting visual outcomes for anterior skull base surgeries, compared to intraoperative visual evoked potential: a pilot explorative study

吲哚菁绿血管造影术预测前颅底手术视觉结果的准确性与术中视觉诱发电位的比较:一项初步探索性研究

Khafaji, Fatemeh; Reyes Medina, Bernardo; Sippl, Christoph; Linsler, Stefan

Accuracy and effectiveness of thoracolumbar pedicle screw placement with a mixed reality head mounted device: first clinical experience and results

使用混合现实头戴式设备进行胸腰椎椎弓根螺钉置入的准确性和有效性:初步临床经验和结果

Reyes Medina, Bernardo; Khafaji, Fatemeh; Saffour, Safwan; Sippl, Christoph; Linsler, Stefan

Inhibition of RNA-binding proteins enhances immunotherapy in ovarian cancer

抑制RNA结合蛋白可增强卵巢癌的免疫疗法

Bley, Nadine; Rausch, Alexander; Müller, Simon; Simon, Theresa; Glaß, Markus; Misiak, Danny; Schian, Laura; Peters, Lara Meret; Dipto, Mohammad; Hmedat, Ali; Busch, Bianca; Schott, Annekatrin; Lederer, Marcell; Wedler, Alice; Rolnik, Robin Benedikt; Elrewany, Hend; Ghazy, Ehab; Sippl, Wolfgang; Vetter, Martina; Wallwiener, Markus; Hüttelmaier, Stefan

Identification of a Proteolysis-Targeting-Chimera that Addresses Activated Checkpoint Kinase-1 Reveals its Non-Catalytic Functions in Tumor Cells

鉴定出一种靶向激活的检查点激酶-1的蛋白水解嵌合体,揭示了其在肿瘤细胞中的非催化功能

Ashry, Ramy; Abdelsalam, Mohamed; Hausen, Julia; Hieber, Christoph; Zeyn, Yanira; Sarnow, Anne-Christin; Schmidt, Matthias; Najafi, Sara; Oehme, Ina; Bros, Matthias; Chen, Jia-Xuan; Dejung, Mario; Sippl, Wolfgang; Krämer, Oliver H