日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cell membrane cholesterol affects serotonin transporter efflux due to altered transporter oligomerization

细胞膜胆固醇通过改变转运蛋白寡聚化影响血清素转运蛋白的外排。

Rudin, Deborah; Luethi, Dino; Niello, Marco; Yang, Jae-Won; Burger, Isabella; Sandtner, Walter; Birner-Gruenberger, Ruth; Schütz, Gerhard J; Sitte, Harald H

The psychedelic phenethylamine 25C-NBF, a selective 5-HT2A agonist, shows psychoplastogenic properties and rapid antidepressant effects in male rodents

迷幻苯乙胺类化合物 25C-NBF 是一种选择性 5-HT2A 激动剂,在雄性啮齿动物中表现出精神可塑性特性和快速抗抑郁作用。

Nadal-Gratacós, Núria; Puigseslloses, Pol; Guzmán, Laura; Weiss, Nicola; Pottie, Eline; Riera-Colomer, Clara; Lardeux, Virginie; Thiriet, Nathalie; Wang, Fu-Hua; Källsten, Liselott; Pérez-Esteban, Irene; Ketsela, Gabriel; Margall, Joel; Berzosa, Xavier; Pubill, David; Rodríguez-Arias, Marta; Ettcheto, Miren; Kehr, Jan; Stove, Christophe; Solinas, Marcello; Sitte, Harald H; Escubedo, Elena; López-Arnau, Raul

Correction to "Next-Generation MDMA Analogue SDMA: Pharmacological and Metabolic Insights"

对“下一代 MDMA 类似物 SDMA:药理学和代谢学见解”的更正

Kastner, Nina; Nadal-Gratacós, Núria; Hemmer, Selina; Alves da Silva, Leticia; McKee, John L; Hell, Tamara; Cicalese, Giulia; Holy, Marion; Kooti, Fatemeh; Jäntsch, Kathrin; Baron, Ricarda; Shacham, Naomi; Cuccurazzu, Bruna; Halberstadt, Adam L; McCorvy, John D; Stockner, Thomas; Meyer, Markus R; López-Arnau, Raúl; Grill, Matthias; Sitte, Harald H

Trials and tribulations of responsible people trying to uphold scientific standards

负责任的人们为维护科学标准而经历的考验和磨难

Sitte, Harald H; Hübner, Jutta; Aust, Norbert; Weisshäupl, Viktor; Ernst, Edzard

Revealing the location and dynamics of a concealed binding site in the dopamine transporter.

揭示多巴胺转运蛋白中隐藏结合位点的位置和动态

Zhu Rong, Sandtner Walter, Stockner Thomas, Heilinger Alexander, Holy Marion, Kudlacek Oliver, Wildling Linda, Saha Kusumika, Fröhlich Anna Sophie, Bindl Michael, Tziortzouda Paraskevi, Haider Anna, Gobl Julia, Suh Saanfor Hubert, Khan Jawad Akbar, Bicher Julia, Kastner Nina, Ebner Andreas, Gruber Hermann J, Freissmuth Michael, Newman Amy Hauck, Sitte Harald H, Hinterdorfer Peter

Fluorescent PyrAte-(S)-citalopram conjugates enable imaging of the serotonin transporter in living tissue

荧光标记的PyrAte-(S)-西酞普兰缀合物可用于活体组织中血清素转运蛋白的成像

Belleza, Oliver J V; Saridakis, Iakovos; Singer, Nadja K; Westergaard, Xavier; Armentia Matheu, Sergio; Lemmerer, Miran; Riomet, Margaux; Sánchez-Murcia, Pedro A; Kastner, Nina; Rukavina, Stefanie; Xiao, Yi; Jäntsch, Kathrin; Niello, Marco; Schicker, Klaus; Sulzer, David; González, Leticia; Maulide, Nuno; Sitte, Harald H

Health risks of cocaine adulteration: local anesthetics as modulators of monoamine and organic cation transporters

可卡因掺杂的健康风险:局部麻醉剂作为单胺和有机阳离子转运体的调节剂

Kudlacek, Oliver; Senning, Niklas; Karden, Alexandra; Ludwig, Iina; Bicher, Julia; Kooti, Fatemeh; Holy, Marion; Stockner, Thomas; Luf, Anton; Sitte, Harald H

Careful Examination of a Novel Azobenzene Paroxetine Derivative and Its Interactions With Biogenic Amine Transporters.

仔细研究一种新型偶氮苯帕罗西汀衍生物及其与生物胺转运体的相互作用

Dreier Dominik, Belleza Oliver John V, Schlögl Katharina, Kickinger Stefanie, Hellsberg Eva, Mayer Felix P, Sandtner Walter, Mikšovsky Philipp, Schittmayer Matthias, Hu Yuntao, Jäntsch Kathrin, Holy Marion, Ecker Gerhard F, Sitte Harald H, Mihovilovic Marko D

Next-Generation MDMA Analogue SDMA: Pharmacological and Metabolic Insights

下一代MDMA类似物SDMA:药理学和代谢学见解

Kastner, Nina; Nadal-Gratacós, Núria; Hemmer, Selina; Alves da Silva, Leticia; McKee, John L; Hell, Tamara; Cicalese, Giulia; Holy, Marion; Kooti, Fatemeh; Jäntsch, Kathrin; Baron, Ricarda; Shacham, Naomi; Cuccurazzu, Bruna; Halberstadt, Adam L; McCorvy, John D; Stockner, Thomas; Meyer, Markus R; López-Arnau, Raúl; Grill, Matthias; Sitte, Harald H

Prolintane analogs as hybrid monoamine transporter ligands: Structural determinants and species differences

脯氨酰胺类似物作为杂合单胺转运体配体:结构决定因素和物种差异

Kastner, Nina; Islam, Mohammad N; Dybek, Michael; Roth, Evelyn; Heisinger, Simon; Holy, Marion; Jäntsch, Kathrin; Walther, Donna; Stockner, Thomas; Baumann, Michael H; Brandt, Simon D; Wallach, Jason; Sitte, Harald H; Kudlacek, Oliver