日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of benzyl carbamate inhibitors of coronavirus M(pro) enzymes from a legacy collection of cysteine protease inhibitors

从一系列已知的半胱氨酸蛋白酶抑制剂中发现冠状病毒M(pro)酶的苄基氨基甲酸酯抑制剂

Sá Magalhães Serafim, Mateus; Kronenberger, Thales; Francisco, Karol R; de Sousa Reis, Erik Vinicius; Gonçalves de Oliveira, Ellen; Marcelino E Oliveira, Fernanda Kelly; Serraglio Fortes, Isadora; Maciel Fernandes, Thaís Helena; Barbosa da Silva, Elany; Fajtova, Pavla; Skinner, Danielle E; Syed, Rafay O; Lage de Siqueira-Neto, Jair; Poso, Antti; Fernandes Mota, Bruno Eduardo; Alves Coelho-Dos-Reis, Jordana Grazziela; Santos Abrahão, Jônatas; Gonçalves Maltarollo, Vinícius; O'Donoghue, Anthony J; Caffrey, Conor R

Enhancing schistosomiasis drug discovery approaches with optimized proteasome substrates.

利用优化的蛋白酶体底物增强血吸虫病药物发现方法

Silva Elany B, Jiang Zhenze, Liu Chenxi, Fajtová Pavla, Teixeira Thaiz R, de Castro Fiorini Maia Giovana, Liu Lawrence J, El-Sakkary Nelly, Skinner Danielle E, Syed Ali, Wang Steven C, Caffrey Conor R, O'Donoghue Anthony J

Comprehensive Analysis of Clinically Discontinued Compounds Using an In Vitro Secondary Pharmacology Panel to Predict Potential Safety Risks during Drug Development

利用体外二级药理学指标对临床终止的化合物进行全面分析,以预测药物研发过程中的潜在安全风险

Albert, Verena; Skinner, Danielle E; Karnwal, Saloni; Guili, Lauren N; Vazquez, Miguel; Ledezma, Omar; Shaffer, Rebecca; Celniker, Aura; De La Cruz, Alexander; Caliendo, Matthew; Hanna, Andrew M; Galdieri, Luciano; King, Alastair J; Servant, Nicole B; Jahic, Mirza

How might flukes and tapeworms maintain genome integrity without a canonical piRNA pathway?

在没有典型的piRNA通路的情况下,吸虫和绦虫如何维持基因组的完整性?

Skinner, Danielle E; Rinaldi, Gabriel; Koziol, Uriel; Brehm, Klaus; Brindley, Paul J

An antibiotic selection marker for schistosome transgenesis

血吸虫转基因的抗生素选择标记

Rinaldi, Gabriel; Suttiprapa, Sutas; Tort, José F; Folley, Anne E; Skinner, Danielle E; Brindley, Paul J