日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A mild and atom-efficient four-component cascade strategy for the construction of biologically relevant 4-hydroxyquinolin-2(1H)-one derivatives

一种温和且原子经济的四组分级联策略,用于构建具有生物学意义的4-羟基喹啉-2(1H)-酮衍生物

Grishin, Dmitrii A; Sharkovskaia, Kseniia I; Kolmakov, Ilya G; Ipatova, Daria A; Petrov, Rostislav A; Dagaev, Nikolai D; Skvortsov, Dmitry A; Khrenova, Maria G; Andreychev, Valeriy V; Evteev, Sergei A; Ivanenkov, Yan A; Antipin, Roman L; Dontsova, Olga А; Beloglazkina, Elena K

Ancestral intronic splicing regulatory elements in the SCNα gene family

SCNα基因家族中的祖先内含子剪接调控元件

Chernyavskaya, Ekaterina; Vorobeva, Margarita; Spirin, Sergei A; Skvortsov, Dmitry A; Pervouchine, Dmitri D

Photoactivatable Cisplatin-Combretastatin-BODIPY Pt(IV) Prodrug for Dual-Action Light-Controlled Chemotherapy

用于双效光控化疗的光活化顺铂-康布瑞他汀-BODIPY Pt(IV)前药

Spector, Daniil V; Karetnikov, Georgy; Bubley, Anna; Akasov, Roman A; Isaeva, Yulia A; Egorova, Tatiana V; Martynov, Alexander G; Bunin, Dmitry; Skvortsov, Dmitry A; Ipatova, Daria; Erofeev, Alexander S; Gorelkin, Petr V; Mamed-Nabizade, Vugara; Kolmogorov, Vasilii S; Vaneev, Alexander N; Rodin, Igor A; Vokuev, Mikhail F; Grishin, Yuri K; Roznyatovsky, Vitaly A; Nikitina, Vita N; Beloglazkina, Elena K; Krasnovskaya, Olga O

3,4-Diarylisoxazoles-Analogues of Combretastatin A-4: Design, Synthesis, and Biological Evaluation In Vitro and In Vivo

3,4-二芳基异噁唑类化合物——康布瑞他汀A-4类似物:设计、合成及体外和体内生物学评价

Karetnikov, Georgy L; Vasilyeva, Lilya A; Babayeva, Gulalek; Pokrovsky, Vadim S; Skvortsov, Dmitry A; Bondarenko, Oksana B

[4+2]-Cycloaddition to 5-Methylidene-Hydantoins and 5-Methylidene-2-Thiohydantoins in the Synthesis of Spiro-2-Chalcogenimidazolones

[4+2]环加成反应与5-亚甲基乙内酰脲和5-亚甲基-2-硫代乙内酰脲反应合成螺-2-硫代咪唑酮

Shybanov, Dmitry E; Kukushkin, Maxim E; Hrytseniuk, Yanislav S; Grishin, Yuri K; Roznyatovsky, Vitaly A; Tafeenko, Viktor A; Skvortsov, Dmitry A; Zyk, Nikolai V; Beloglazkina, Elena K

Verubulin (Azixa) Analogues with Increased Saturation: Synthesis, SAR and Encapsulation in Biocompatible Nanocontainers Based on Ca(2+) or Mg(2+) Cross-Linked Alginate.

具有更高饱和度的维鲁布林(Azixa)类似物:基于 Ca(2+) 或 Mg(2+) 交联藻酸盐的生物相容性纳米容器中的合成、SAR 和封装

Sedenkova Kseniya N, Leschukov Denis N, Grishin Yuri K, Zefirov Nikolay A, Gracheva Yulia A, Skvortsov Dmitry A, Hrytseniuk Yanislav S, Vasilyeva Lilja A, Spirkova Elena A, Shevtsov Pavel N, Shevtsova Elena F, Lukmanova Alina R, Spiridonov Vasily V, Markova Alina A, Nguyen Minh T, Shtil Alexander A, Zefirova Olga N, Yaroslavov Alexander A, Milaeva Elena R, Averina Elena B

The Synthesis and Biological Evaluation of 2-(1H-Indol-3-yl)quinazolin-4(3H)-One Derivatives

2-(1H-吲哚-3-基)喹唑啉-4(3H)-酮衍生物的合成及生物学评价

Mendogralo, Elena Y; Nesterova, Larisa Y; Nasibullina, Ekaterina R; Shcherbakov, Roman O; Tkachenko, Alexander G; Sidorov, Roman Y; Sukonnikov, Maxim A; Skvortsov, Dmitry A; Uchuskin, Maxim G

Synthesis and Biological Evaluation of Novel Dispiro-Indolinones with Anticancer Activity

新型二螺吲哚啉酮的合成及抗癌活性生物学评价

Ivanenkov, Yan A; Kukushkin, Maxim E; Beloglazkina, Anastasia A; Shafikov, Radik R; Barashkin, Alexander A; Ayginin, Andrey A; Serebryakova, Marina S; Majouga, Alexander G; Skvortsov, Dmitry A; Tafeenko, Viktor A; Beloglazkina, Elena K

Panel of potential lncRNA biomarkers can distinguish various types of liver malignant and benign tumors

一组潜在的lncRNA生物标志物可以区分各种类型的肝脏恶性肿瘤和良性肿瘤。

Burenina, Olga Y; Lazarevich, Natalia L; Kustova, Inna F; Shavochkina, Daria A; Moroz, Ekaterina A; Kudashkin, Nikolay E; Patyutko, Yuriy I; Metelin, Alexey V; Kim, Eduard F; Skvortsov, Dmitry A; Zatsepin, Timofei S; Rubtsova, Maria P; Dontsova, Olga A

Identification of Novel Antibacterials Using Machine Learning Techniques

利用机器学习技术鉴定新型抗菌药物

Ivanenkov, Yan A; Zhavoronkov, Alex; Yamidanov, Renat S; Osterman, Ilya A; Sergiev, Petr V; Aladinskiy, Vladimir A; Aladinskaya, Anastasia V; Terentiev, Victor A; Veselov, Mark S; Ayginin, Andrey A; Kartsev, Victor G; Skvortsov, Dmitry A; Chemeris, Alexey V; Baimiev, Alexey Kh; Sofronova, Alina A; Malyshev, Alexander S; Filkov, Gleb I; Bezrukov, Dmitry S; Zagribelnyy, Bogdan A; Putin, Evgeny O; Puchinina, Maria M; Dontsova, Olga A