日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Shaping Antimalarials: A Geometry-First Approach to PfCLK3 Covalent Inhibitors

抗疟药的调控:一种基于几何结构的PfCLK3共价抑制剂设计方法

Brettell, Skye B; Fuentes-Guerra Bustos, Carla; Sharma, Saumya; Cann, Gillian; Carruthers, Lauren V; Begen, Abbey; Milligan, Graeme; Clarke, David J; Tobin, Andrew B; Jamieson, Andrew G

Lysine targeting covalent inhibitors of malarial kinase PfCLK3

赖氨酸靶向共价抑制疟原虫激酶 PfCLK3 的抑制剂

Brettell, Skye B; Cann, Gillian; Begen, Abbey; Sharma, Saumya; Mahindra, Amit; Carruthers, Lauren V; Milligan, Graeme; Clarke, David J; Tobin, Andrew B; Jamieson, Andrew G

Targeting PfCLK3 with Covalent Inhibitors: A Novel Strategy for Malaria Treatment

利用共价抑制剂靶向 PfCLK3:一种治疗疟疾的新策略

Brettell, Skye B; Janha, Omar; Begen, Abbey; Cann, Gillian; Sharma, Saumya; Olaniyan, Niniola; Yelland, Tamas; Hole, Alison J; Alam, Benazir; Mayville, Emily; Gillespie, Ross; Capper, Michael; Fidock, David A; Milligan, Graeme; Clarke, David J; Tobin, Andrew B; Jamieson, Andrew G