日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Reciprocal links between methionine metabolism, DNA repair and therapy resistance in glioblastoma

胶质母细胞瘤中蛋氨酸代谢、DNA修复和治疗耐药性之间的相互联系

Korimerla, Navyateja; Meghdadi, Baharan; Haq, Isra; Wilder-Romans, Kari; Xu, Jie; Becker, Nicole; Zhu, Ziqing; Kalev, Peter; Qi, Nathan; Evans, Charles; Kachman, Maureen; Zhao, Zitong; Lin, Angelica; Scott, Andrew J; O'Brien, Alexandra; Kothari, Ayesha; Sajjakulnukit, Peter; Zhang, Li; Palavalasa, Sravya; Peterson, Erik R; Hyer, Marc L; Marjon, Katya; Sleger, Taryn; Morgan, Meredith A; Lyssiotis, Costas A; Stone, Everett M; Ferris, Sean P; Lawrence, Theodore S; Nagrath, Deepak; Zhou, Weihua; Wahl, Daniel R

Discovery of M-1121 as an Orally Active Covalent Inhibitor of Menin-MLL Interaction Capable of Achieving Complete and Long-Lasting Tumor Regression

发现 M-1121 是一种口服的 Menin-MLL 相互作用共价抑制剂,能够实现完全且持久的肿瘤消退

Meng Zhang, Angelo Aguilar, Shilin Xu, Liyue Huang, Krishnapriya Chinnaswamy, Taryn Sleger, Bo Wang, Stefan Gross, Brandon N Nicolay, Sebastien Ronseaux, Kaitlin Harvey, Yu Wang, Donna McEachern, Paul D Kirchhoff, Zhaomin Liu, Jeanne Stuckey, Adriana E Tron, Tao Liu, Shaomeng Wang

A chemical biology screen identifies a vulnerability of neuroendocrine cancer cells to SQLE inhibition

化学生物学筛选确定神经内分泌癌细胞对 SQLE 抑制的脆弱性

Christopher E Mahoney, David Pirman, Victor Chubukov, Taryn Sleger, Sebastian Hayes, Zi Peng Fan, Eric L Allen, Ying Chen, Lingling Huang, Meina Liu, Yingjia Zhang, Gabrielle McDonald, Rohini Narayanaswamy, Sung Choe, Yue Chen, Stefan Gross, Giovanni Cianchetta, Anil K Padyana, Stuart Murray, Wei Li