日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Tetrahydroisoquinoline CXCR4 Antagonists Adopt a Hybrid Binding Mode within the Peptide Subpocket of the CXCR4 Receptor

四氢异喹啉类CXCR4拮抗剂在CXCR4受体的肽亚口袋内采用混合结合模式

Katzman, Brooke M; Cox, Bryan D; Prosser, Anthony R; Alcaraz, Ana A; Murat, Brigitte; Héroux, Madeleine; Tebben, Andrew; Zhang, Yong; Schroeder, Gretchen M; Snyder, James P; Wilson, Lawrence J; Liotta, Dennis C

The GluN2B-Glu413Gly NMDA receptor variant arising from a de novo GRIN2B mutation promotes ligand-unbinding and domain opening

由新生GRIN2B突变产生的GluN2B-Glu413Gly NMDA受体变体促进配体解离和结构域开放

Wells, Gordon; Yuan, Hongjie; McDaniel, Miranda J; Kusumoto, Hirofumi; Snyder, James P; Liotta, Dennis C; Traynelis, Stephen F

Visualizing cancer and response to therapy in vivo using Cy5.5-labeled factor VIIa and anti-tissue factor antibody.

利用 Cy5.5 标记的因子 VIIa 和抗组织因子抗体在体内可视化癌症和治疗反应

Zhu Shijun, Kisiel Walter, Lu Yang J, Petersen Lars C, Ndungu John M, Moore Terry W, Parker Ernest T, Sun Aiming, Sarkaria Jann N, Snyder James P, Liotta Dennis C, Brat Daniel J, El-Rayes Bassel F, Shoji Mamoru

The quest for a simple bioactive analog of paclitaxel as a potential anticancer agent

寻找一种简单的紫杉醇生物活性类似物作为潜在的抗癌药物

Kingston, David G I; Snyder, James P

Eliminating the heart from the curcumin molecule: monocarbonyl curcumin mimics (MACs)

从姜黄素分子中去除核心结构:单羰基姜黄素类似物(MACs)

Shetty, Dinesh; Kim, Yong Joon; Shim, Hyunsuk; Snyder, James P

Structural determinants and mechanism of action of a GluN2C-selective NMDA receptor positive allosteric modulator

GluN2C选择性NMDA受体正向变构调节剂的结构决定因素和作用机制

Khatri, Alpa; Burger, Pieter B; Swanger, Sharon A; Hansen, Kasper B; Zimmerman, Sommer; Karakas, Erkan; Liotta, Dennis C; Furukawa, Hiro; Snyder, James P; Traynelis, Stephen F

Anti-HIV small-molecule binding in the peptide subpocket of the CXCR4:CVX15 crystal structure

抗HIV小分子与CXCR4:CVX15晶体结构肽亚口袋的结合

Cox, Bryan D; Prosser, Anthony R; Katzman, Brooke M; Alcaraz, Ana A; Liotta, Dennis C; Wilson, Lawrence J; Snyder, James P

Autophagy and apoptosis in hepatocellular carcinoma induced by EF25-(GSH)2: a novel curcumin analog

EF25-(GSH)2(一种新型姜黄素类似物)诱导肝细胞癌的自噬和凋亡

Zhou, Tao; Ye, Lili; Bai, Yu; Sun, Aiming; Cox, Bryan; Liu, Dahai; Li, Yong; Liotta, Dennis; Snyder, James P; Fu, Haian; Huang, Bei

Mouse pharmacokinetics and metabolism of the curcumin analog, 4-piperidinone,3,5-bis[(2-fluorophenyl)methylene]-acetate(3E,5E) (EF-24; NSC 716993)

姜黄素类似物 4-哌啶酮,3,5-双[(2-氟苯基)亚甲基]乙酸酯(3E,5E) (EF-24; NSC 716993) 的小鼠药代动力学和代谢

Reid, Joel M; Buhrow, Sarah A; Gilbert, Judith A; Jia, Lee; Shoji, Mamoru; Snyder, James P; Ames, Matthew M

Discovery of tetrahydroisoquinoline-based CXCR4 antagonists

发现基于四氢异喹啉的CXCR4拮抗剂

Truax, Valarie M; Zhao, Huanyu; Katzman, Brooke M; Prosser, Anthony R; Alcaraz, Ana A; Saindane, Manohar T; Howard, Randy B; Culver, Deborah; Arrendale, Richard F; Gruddanti, Prahbakar R; Evers, Taylor J; Natchus, Michael G; Snyder, James P; Liotta, Dennis C; Wilson, Lawrence J