Discovery and Preclinical Evaluation of BMS-955829, a Potent Positive Allosteric Modulator of mGluR5
发现和临床前评估 BMS-955829,一种强效的 mGluR5 正向变构调节剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5b00450
Yang, Fukang; Snyder, Lawrence B; Balakrishnan, Anand; Brown, Jeffrey M; Sivarao, Digavalli V; Easton, Amy; Fernandes, Alda; Gulianello, Michael; Hanumegowda, Umesh M; Huang, Hong; Huang, Yanling; Jones, Kelli M; Li, Yu-Wen; Matchett, Michele; Mattson, Gail; Miller, Regina; Santone, Kenneth S; Senapati, Arun; Shields, Eric E; Simutis, Frank J; Westphal, Ryan; Whiterock, Valerie J; Bronson, Joanne J; Macor, John E; Degnan, Andrew P