Antiviral Activity, Safety, and Exposure-Response Relationships of GSK3532795, a Second-Generation Human Immunodeficiency Virus Type 1 Maturation Inhibitor, Administered as Monotherapy or in Combination With Atazanavir With or Without Ritonavir in a Phase 2a Randomized, Dose-Ranging, Controlled Trial (AI468002)
在 2a 期随机、剂量范围、对照试验 (AI468002) 中,评估了第二代人类免疫缺陷病毒 1 型成熟抑制剂 GSK3532795 作为单药治疗或与阿扎那韦联合治疗(含或不含利托那韦)的抗病毒活性、安全性和暴露-反应关系。
期刊:Clinical Infectious Diseases
影响因子:7.3
doi:10.1093/cid/cix239
Hwang, Carey; Schürmann, Dirk; Sobotha, Christian; Boffito, Marta; Sevinsky, Heather; Ray, Neelanjana; Ravindran, Palanikumar; Xiao, Hong; Keicher, Christian; Hüser, Andreas; Krystal, Mark; Dicker, Ira B; Grasela, Dennis; Lataillade, Max