日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Clinical Outcomes of Intravenous Thrombolysis in Acute Ischemic Stroke: A Prospective Observational Study From Mumbai

急性缺血性卒中静脉溶栓的临床结果:一项来自孟买的前瞻性观察研究

Solapure, Vivek; Gore, Sandeep; Shah, Keyur; Shah, Pradip

Erratum for Brunschwig et al., "UCT943, a Next-Generation Plasmodium falciparum PI4K Inhibitor Preclinical Candidate for the Treatment of Malaria"

Brunschwig 等人的论文“UCT943,一种用于治疗疟疾的下一代恶性疟原虫 PI4K 抑制剂临床前候选药物”的勘误

Brunschwig, Christel; Lawrence, Nina; Taylor, Dale; Abay, Efrem; Njoroge, Mathew; Basarab, Gregory S; Le Manach, Claire; Paquet, Tanya; Gonzàlez Cabrera, Diego; Nchinda, Aloysius T; de Kock, Carmen; Wiesner, Lubbe; Denti, Paolo; Waterson, David; Blasco, Benjamin; Leroy, Didier; Witty, Michael J; Donini, Cristina; Duffy, James; Wittlin, Sergio; White, Karen L; Charman, Susan A; Jiménez-Díaz, Maria Belén; Angulo-Barturen, Iñigo; Herreros, Esperanza; Gamo, Francisco Javier; Rochford, Rosemary; Mancama, Dalu; Coetzer, Theresa L; van der Watt, Mariëtte E; Reader, Janette; Birkholtz, Lyn-Marie; Marsh, Kennan C; Solapure, Suresh M; Burke, John E; McPhail, Jacob A; Vanaerschot, Manu; Fidock, David A; Fish, Paul V; Siegl, Peter; Smith, Dennis A; Wirjanata, Grennady; Noviyanti, Rintis; Price, Ric N; Marfurt, Jutta; Silue, Kigbafori D; Street, Leslie J; Chibale, Kelly

UCT943, a Next-Generation Plasmodium falciparum PI4K Inhibitor Preclinical Candidate for the Treatment of Malaria

UCT943,一种用于治疗疟疾的下一代恶性疟原虫PI4K抑制剂临床前候选药物

Brunschwig, Christel; Lawrence, Nina; Taylor, Dale; Abay, Efrem; Njoroge, Mathew; Basarab, Gregory S; Le Manach, Claire; Paquet, Tanya; Cabrera, Diego Gonzàlez; Nchinda, Aloysius T; de Kock, Carmen; Wiesner, Lubbe; Denti, Paolo; Waterson, David; Blasco, Benjamin; Leroy, Didier; Witty, Michael J; Donini, Cristina; Duffy, James; Wittlin, Sergio; White, Karen L; Charman, Susan A; Jiménez-Díaz, Maria Belén; Angulo-Barturen, Iñigo; Herreros, Esperanza; Gamo, Francisco Javier; Rochford, Rosemary; Mancama, Dalu; Coetzer, Theresa L; van der Watt, Mariëtte E; Reader, Janette; Birkholtz, Lyn-Marie; Marsh, Kennan C; Solapure, Suresh M; Burke, John E; McPhail, Jacob A; Vanaerschot, Manu; Fidock, David A; Fish, Paul V; Siegl, Peter; Smith, Dennis A; Wirjanata, Grennady; Noviyanti, Rintis; Price, Ric N; Marfurt, Jutta; Silue, Kigbafori D; Street, Leslie J; Chibale, Kelly

Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate

三氨基嘧啶是一种速效且长效的抗疟疾候选药物。

Hameed P, Shahul; Solapure, Suresh; Patil, Vikas; Henrich, Philipp P; Magistrado, Pamela A; Bharath, Sowmya; Murugan, Kannan; Viswanath, Pavithra; Puttur, Jayashree; Srivastava, Abhishek; Bellale, Eknath; Panduga, Vijender; Shanbag, Gajanan; Awasthy, Disha; Landge, Sudhir; Morayya, Sapna; Koushik, Krishna; Saralaya, Ramanatha; Raichurkar, Anandkumar; Rautela, Nikhil; Roy Choudhury, Nilanjana; Ambady, Anisha; Nandishaiah, Radha; Reddy, Jitendar; Prabhakar, K R; Menasinakai, Sreenivasaiah; Rudrapatna, Suresh; Chatterji, Monalisa; Jiménez-Díaz, María Belén; Martínez, María Santos; Sanz, Laura María; Coburn-Flynn, Olivia; Fidock, David A; Lukens, Amanda K; Wirth, Dyann F; Bandodkar, Balachandra; Mukherjee, Kakoli; McLaughlin, Robert E; Waterson, David; Rosenbrier-Ribeiro, Lyn; Hickling, Kevin; Balasubramanian, V; Warner, Peter; Hosagrahara, Vinayak; Dudley, Adam; Iyer, Pravin S; Narayanan, Shridhar; Kavanagh, Stefan; Sambandamurthy, Vasan K

In silico-based high-throughput screen for discovery of novel combinations for tuberculosis treatment

利用计算机模拟高通量筛选发现治疗结核病的新组合

Singh, Ragini; Ramachandran, Vasanthi; Shandil, Radha; Sharma, Sreevalli; Khandelwal, Swati; Karmarkar, Malancha; Kumar, Naveen; Solapure, Suresh; Saralaya, Ramanatha; Nanduri, Robert; Panduga, Vijender; Reddy, Jitendar; Prabhakar, K R; Rajagopalan, Swaminathan; Rao, Narasimha; Narayanan, Shridhar; Anandkumar, Anand; Balasubramanian, V; Datta, Santanu

Bactericidal activity and mechanism of action of AZD5847, a novel oxazolidinone for treatment of tuberculosis

AZD5847(一种用于治疗结核病的新型噁唑烷酮类药物)的杀菌活性和作用机制

Balasubramanian, V; Solapure, S; Iyer, H; Ghosh, A; Sharma, S; Kaur, P; Deepthi, R; Subbulakshmi, V; Ramya, V; Ramachandran, V; Balganesh, M; Wright, L; Melnick, D; Butler, S L; Sambandamurthy, V K

MK-5172, a Selective Inhibitor of Hepatitis C Virus NS3/4a Protease with Broad Activity across Genotypes and Resistant Variants

MK-5172,一种选择性抑制丙型肝炎病毒NS3/4a蛋白酶的药物,对多种基因型和耐药变异株均具有广泛活性。

Draper, Michael P; Weir, S; Macone, A; Donatelli, J; Trieber, C A; Tanaka, S K; Levy, Stuart B; P, Shahul Hameed; Solapure, Suresh; Mukherjee, Kakoli; Nandi, Vrinda; Waterson, David; Shandil, Radha; Balganesh, Meenakshi; Sambandamurthy, Vasan K; Raichurkar, Anand Kumar; Deshpande, Abhijeet; Ghosh, Anirban; Awasthy, Disha; Shanbhag, Gajanan; Sheikh, Gulebahar; McMiken, Helen; Puttur, Jayashree; Reddy, Jitendar; Werngren, Jim; Read, Jon; Kumar, Mahesh; R, Manjunatha; Chinnapattu, Murugan; Madhavapeddi, Prashanti; Manjrekar, Praveena; Basu, Reetobrata; Gaonkar, Sheshagiri; Sharma, Sreevalli; Hoffner, Sven; Humnabadkar, Vaishali; Subbulakshmi, Venkita; Panduga, Vijender; Summa, Vincenzo; Ludmerer, Steven W; McCauley, John A; Fandozzi, Christine; Burlein, Christine; Claudio, Giuliano; Coleman, Paul J; DiMuzio, Jillian M; Ferrara, Marco; Filippo, Marcello Di; Gates, Adam T; Graham, Donald J; Harper, Steven; Hazuda, Daria J; Huang, Qian; McHale, Carolyn; Monteagudo, Edith; Pucci, Vincenzo; Rowley, Michael; Rudd, Michael T; Soriano, Aileen; Stahlhut, Mark W; Vacca, Joseph P; Olsen, David B; Liverton, Nigel J; Carroll, Steven S

1,4-azaindole, a potential drug candidate for treatment of tuberculosis

1,4-氮杂吲哚,一种潜在的结核病治疗候选药物

Chatterji, Monalisa; Shandil, Radha; Manjunatha, M R; Solapure, Suresh; Ramachandran, Vasanthi; Kumar, Naveen; Saralaya, Ramanatha; Panduga, Vijender; Reddy, Jitendar; Prabhakar, K R; Sharma, Sreevalli; Sadler, Claire; Cooper, Christopher B; Mdluli, Khisi; Iyer, Pravin S; Narayanan, Shridhar; Shirude, Pravin S

Pharmacokinetic and pharmacodynamic evaluation of AZD5847 in a mouse model of tuberculosis

AZD5847 在小鼠结核病模型中的药代动力学和药效学评估

V Balasubramanian, Suresh Solapure, Radha Shandil, Sheshagiri Gaonkar, K N Mahesh, Jitender Reddy, Abhijeet Deshpande, Sowmya Bharath, Naveen Kumar, Lindsay Wright, David Melnick, Scott L Butler

Optimization of pyrrolamides as mycobacterial GyrB ATPase inhibitors: structure-activity relationship and in vivo efficacy in a mouse model of tuberculosis

吡咯酰胺作为分枝杆菌 GyrB ATPase 抑制剂的优化:结构-活性关系和小鼠结核病模型中的体内功效

Shahul Hameed P, Suresh Solapure, Kakoli Mukherjee, Vrinda Nandi, David Waterson, Radha Shandil, Meenakshi Balganesh, Vasan K Sambandamurthy, Anand Kumar Raichurkar, Abhijeet Deshpande, Anirban Ghosh, Disha Awasthy, Gajanan Shanbhag, Gulebahar Sheikh, Helen McMiken, Jayashree Puttur, Jitendar Reddy,