日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fluorescently engineered KRAS-mutant organoids as versatile tools for in vitro and in vivo cancer modeling

荧光标记的KRAS突变类器官作为体外和体内癌症建模的多功能工具

Savadipour, Alireza; Tummala, Krishna S; Muise, Eric S; Buchanan, Mark; Vidimar, Vania; Veling, Mike; Liu, Jun; Kopinja, Johnny; Schneider, Charlie; Chan, Brian Pak Ho; Carr, Richard; Norton, Scott; Gaspar, John M; Piesvaux, Jennifer; Leccese, Erica; Park, Eunsil; Moy, Lily Y; Long, Brian J; Solban, Nicolas

Utilization of Metabolite Identification and Structural Data to Guide Design of Low-Dose IDO1 Inhibitors

利用代谢物鉴定和结构数据指导低剂量IDO1抑制剂的设计

Hopkins, Brett; Zhang, Hongjun; Bharathan, Indu; Li, Derun; Pu, Qinglin; Zhou, Hua; Martinot, Theodore A; Fradera, Xavier; Lammens, Alfred; Lesburg, Charles A; Cohen, Ryan D; Ballard, Jeanine; Knemeyer, Ian; Otte, Karin; Vincent, Stella; Miller, J Richard; Solban, Nicolas; Cheng, Mangeng; Geda, Prasanthi; Smotrov, Nadya; Song, Xuelei; Bennett, David Jonathan; Han, Yongxin

Discovery of Potent and Orally Available Bicyclo[1.1.1]pentane-Derived Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitors

发现高效且口服有效的双环[1.1.1]戊烷衍生的吲哚胺-2,3-双加氧酶1 (IDO1) 抑制剂

Pu, Qinglin; Zhang, Hongjun; Guo, Liangqin; Cheng, Mangeng; Doty, Amy C; Ferguson, Heidi; Fradera, Xavier; Lesburg, Charles A; McGowan, Meredeth A; Miller, J Richard; Geda, Prasanthi; Song, Xuelei; Otte, Karin; Sciammetta, Nunzio; Solban, Nicolas; Yu, Wensheng; Sloman, David L; Zhou, Hua; Lammens, Alfred; Neumann, Lars; Bennett, David Jonathan; Pasternak, Alexander; Han, Yongxin

Discovery of Amino-cyclobutarene-derived Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitors for Cancer Immunotherapy

发现氨基环丁烯衍生的吲哚胺-2,3-双加氧酶1 (IDO1) 抑制剂用于癌症免疫治疗

Zhang, Hongjun; Liu, Kun; Pu, Qinglin; Achab, Abdelghani; Ardolino, Michael J; Cheng, Mangeng; Deng, Yongqi; Doty, Amy C; Ferguson, Heidi; Fradera, Xavier; Knemeyer, Ian; Kurukulasuriya, Ravi; Lam, Yu-Hong; Lesburg, Charles A; Martinot, Theodore A; McGowan, Meredeth A; Miller, J Richard; Otte, Karin; Biju, Purakattle J; Sciammetta, Nunzio; Solban, Nicolas; Yu, Wensheng; Zhou, Hua; Wang, Xiao; Bennett, David Jonathan; Han, Yongxin

COMMD5/HCaRG Hooks Endosomes on Cytoskeleton and Coordinates EGFR Trafficking

COMMD5/HCaRG 将内体钩在细胞骨架上并协调 EGFR 运输

Carole G Campion, Kossay Zaoui, Thomas Verissimo, Suzanne Cossette, Hiroyuki Matsuda, Nicolas Solban, Pavel Hamet, Johanne Tremblay

Cortical-Bone Fragility--Insights from sFRP4 Deficiency in Pyle's Disease

皮质骨脆性——来自派尔氏病中sFRP4缺乏症的启示

Kiper, Pelin O Simsek; Saito, Hiroaki; Gori, Francesca; Unger, Sheila; Hesse, Eric; Yamana, Kei; Kiviranta, Riku; Solban, Nicolas; Liu, Jeff; Brommage, Robert; Boduroglu, Koray; Bonafé, Luisa; Campos-Xavier, Belinda; Dikoglu, Esra; Eastell, Richard; Gossiel, Fatma; Harshman, Keith; Nishimura, Gen; Girisha, Katta M; Stevenson, Brian J; Takita, Hiroyuki; Rivolta, Carlo; Superti-Furga, Andrea; Baron, Roland

Inhibition of ALK1 signaling with dalantercept combined with VEGFR TKI leads to tumor stasis in renal cell carcinoma

达兰特西普联合VEGFR TKI抑制ALK1信号通路可导致肾细胞癌肿瘤停滞。

Wang, Xiaoen; Solban, Nicolas; Khanna, Prateek; Callea, Marcella; Song, Jiaxi; Alsop, David C; Pearsall, R Scott; Atkins, Michael B; Mier, James W; Signoretti, Sabina; Alimzhanov, Marat; Kumar, Ravi; Bhasin, Manoj K; Bhatt, Rupal S

A soluble bone morphogenetic protein type IA receptor increases bone mass and bone strength

可溶性骨形态发生蛋白 IA 型受体可增加骨量和骨强度

Marc Baud'huin, Nicolas Solban, Milton Cornwall-Brady, Dianne Sako, Yoshimi Kawamoto, Katia Liharska, Darren Lath, Mary L Bouxsein, Kathryn W Underwood, Jeffrey Ucran, Ravindra Kumar, Eileen Pobre, Asya Grinberg, Jasbir Seehra, Ernesto Canalis, R Scott Pearsall, Peter I Croucher

Soluble endoglin specifically binds bone morphogenetic proteins 9 and 10 via its orphan domain, inhibits blood vessel formation, and suppresses tumor growth

可溶性内皮糖蛋白通过其孤儿结构域特异性结合骨形态发生蛋白 9 和 10,抑制血管形成并抑制肿瘤生长

Roselyne Castonguay, Eric D Werner, Robert G Matthews, Eleonora Presman, Aaron W Mulivor, Nicolas Solban, Dianne Sako, R Scott Pearsall, Kathryn W Underwood, Jasbir Seehra, Ravindra Kumar, Asya V Grinberg

ALK1-Fc inhibits multiple mediators of angiogenesis and suppresses tumor growth

ALK1-Fc 抑制多种血管生成介质并抑制肿瘤生长

Dianne Mitchell, Eileen G Pobre, Aaron W Mulivor, Asya V Grinberg, Roselyne Castonguay, Travis E Monnell, Nicolas Solban, Jeffrey A Ucran, R Scott Pearsall, Kathryn W Underwood, Jasbir Seehra, Ravindra Kumar