日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Author Correction: Targeting the SHOC2-RAS interaction in RAS-mutant cancers

作者更正:靶向 RAS 突变癌症中的 SHOC2-RAS 相互作用

Hauseman, Zachary J; Stauffer, Frédéric; Beyer, Kim S; Mollé, Sandra; Cavicchioli, Elena; Marchand, Jean-Remy; Fodor, Michelle; Viscomi, Jessica; Dhembi, Anxhela; Katz, Stéphanie; Faggion, Beatrice; Lanter, Mylene; Kerr, Grainne; Schildknecht, Daniela; Handl, Cornelia; Maddalo, Danilo; Pissot Soldermann, Carole; Brady, Jacob; Shrestha, Om; Nguyen, Zachary; Leder, Lukas; Cremosnik, Gregor; Lopez Romero, Sandra; Hassiepen, Ulrich; Stams, Travis; Linder, Markus; Galli, Giorgio G; Guthy, Daniel A; King, Daniel A; Maira, Sauveur-Michel; Thoma, Claudio R; Ehmke, Veronika; Tordella, Luca

Targeting the SHOC2-RAS interaction in RAS-mutant cancers.

靶向 RAS 突变癌症中的 SHOC2-RAS 相互作用

Hauseman Zachary J, Stauffer Frédéric, Beyer Kim S, Mollé Sandra, Cavicchioli Elena, Marchand Jean-Remy, Fodor Michelle, Viscomi Jessica, Dhembi Anxhela, Katz Stéphanie, Faggion Beatrice, Lanter Mylene, Kerr Grainne, Schildknecht Daniela, Handl Cornelia, Maddalo Danilo, Pissot Soldermann Carole, Brady Jacob, Shrestha Om, Nguyen Zachary, Leder Lukas, Cremosnik Gregor, Lopez Romero Sandra, Hassiepen Ulrich, Stams Travis, Linder Markus, Galli Giorgio G, Guthy Daniel A, King Daniel A, Maira Sauveur-Michel, Thoma Claudio R, Ehmke Veronika, Tordella Luca

Author Correction: Direct and selective pharmacological disruption of the YAP-TEAD interface by IAG933 inhibits Hippo-dependent and RAS-MAPK-altered cancers

作者更正:IAG933 通过直接和选择性地药理学手段破坏 YAP-TEAD 界面,从而抑制 Hippo 依赖性和 RAS-MAPK 改变的癌症。

Chapeau, Emilie A; Sansregret, Laurent; Galli, Giorgio G; Chène, Patrick; Wartmann, Markus; Mourikis, Thanos P; Jaaks, Patricia; Baltschukat, Sabrina; Barbosa, Ines A M; Bauer, Daniel; Brachmann, Saskia M; Delaunay, Clara; Estadieu, Claire; Faris, Jason E; Furet, Pascal; Harlfinger, Stefanie; Hueber, Andreas; Jiménez Núñez, Eloísa; Kodack, David P; Mandon, Emeline; Martin, Typhaine; Mesrouze, Yannick; Romanet, Vincent; Scheufler, Clemens; Sellner, Holger; Stamm, Christelle; Sterker, Dario; Tordella, Luca; Hofmann, Francesco; Soldermann, Nicolas; Schmelzle, Tobias

Direct and selective pharmacological disruption of the YAP-TEAD interface by IAG933 inhibits Hippo-dependent and RAS-MAPK-altered cancers

IAG933通过直接和选择性地药理学手段破坏YAP-TEAD界面,从而抑制Hippo依赖性和RAS-MAPK改变的癌症。

Emilie A Chapeau ,Laurent Sansregret ,Giorgio G Galli ,Patrick Chène ,Markus Wartmann ,Thanos P Mourikis ,Patricia Jaaks ,Sabrina Baltschukat ,Ines A M Barbosa ,Daniel Bauer ,Saskia M Brachmann ,Clara Delaunay ,Claire Estadieu ,Jason E Faris ,Pascal Furet ,Stefanie Harlfinger ,Andreas Hueber ,Eloísa Jiménez Núñez ,David P Kodack ,Emeline Mandon ,Typhaine Martin ,Yannick Mesrouze ,Vincent Romanet ,Clemens Scheufler ,Holger Sellner ,Christelle Stamm ,Dario Sterker ,Luca Tordella ,Francesco Hofmann ,Nicolas Soldermann ,Tobias Schmelzle

Discovery of New Binders for DCAF1, an Emerging Ligase Target in the Targeted Protein Degradation Field

在靶向蛋白降解领域,发现了一种新兴的连接酶靶点——DCAF1 的新型结合剂。

Vulpetti, Anna; Holzer, Philipp; Schmiedeberg, Niko; Imbach-Weese, Patricia; Pissot-Soldermann, Carole; Hollingworth, Gregory J; Radimerski, Thomas; Thoma, Claudio R; Stachyra, Therese-Marie; Wojtynek, Matthias; Maschlej, Magdalena; Chau, Suzanne; Schuffenhauer, Ansgar; Fernández, César; Schröder, Martin; Renatus, Martin

Effective "activated PI3Kδ syndrome"-targeted therapy with the PI3Kδ inhibitor leniolisib

使用PI3Kδ抑制剂leniolisib进行有效的“活化PI3Kδ综合征”靶向治疗

Rao, V Koneti; Webster, Sharon; Dalm, Virgil A S H; Šedivá, Anna; van Hagen, P Martin; Holland, Steven; Rosenzweig, Sergio D; Christ, Andreas D; Sloth, Birgitte; Cabanski, Maciej; Joshi, Aniket D; de Buck, Stefan; Doucet, Julie; Guerini, Danilo; Kalis, Christoph; Pylvaenaeinen, Ilona; Soldermann, Nicolas; Kashyap, Anuj; Uzel, Gulbu; Lenardo, Michael J; Patel, Dhavalkumar D; Lucas, Carrie L; Burkhart, Christoph

Modulation of activation-loop phosphorylation by JAK inhibitors is binding mode dependent

JAK 抑制剂对活化环磷酸化的调节依赖于结合模式

Rita Andraos #, Zhiyan Qian #, Débora Bonenfant, Joëlle Rubert, Eric Vangrevelinghe, Clemens Scheufler, Fanny Marque, Catherine H Régnier, Alain De Pover, Hugues Ryckelynck, Neha Bhagwat, Priya Koppikar, Aviva Goel, Lorenza Wyder, Gisele Tavares, Fabienne Baffert, Carole Pissot-Soldermann, Paul W Ma