日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Discovery of Bridged Benzoazepine Amides as Selective Allosteric Modulators of RIPK1

桥联苯并氮杂卓酰胺作为RIPK1选择性变构调节剂的发现

Chen, Joanna L; Methot, Joey L; Mitcheltree, Matthew J; Musacchio, Andrew; Corcoran, Emily B; Feng, Guo; Lammens, Alfred; Maskos, Klaus; Palte, Rachel L; Rickard, Meredith M; Otte, Karin M; Mansueto, My S; Venkat, Sriraman; Sondey, Christopher; Thomsen, Maren; Lesburg, Charles A; Fradera, Xavier; Fell, Matthew J; DiMauro, Erin F; Siliphaivanh, Phieng

Mechanistic insights on novel small molecule allosteric activators of cGMP-dependent protein kinase PKG1α

cGMP 依赖性蛋白激酶 PKG1α 的新型小分子变构激活剂的机制见解

Paul Tawa, Lei Zhang, Essam Metwally, Yan Hou, Mark A McCoy, W Michael Seganish, Rumin Zhang, Emily Frank, Payal Sheth, Jennifer Hanisak, Christopher Sondey, David Bauman, Aileen Soriano

Establishing and Validating Cellular Functional Target Engagement Assay for Selective IRAK4 Inhibitor Discovery

建立并验证细胞功能靶标参与分析以发现选择性 IRAK4 抑制剂

Yiping Chen, Dongyu Sun, Ruojing Yang, Jongwon Lim, Christopher Sondey, Jeremy Presland, Larissa Rakhilina, George Addona, Ilona Kariv, Hongmin Chen

Allosteric Modulation of Protein Arginine Methyltransferase 5 (PRMT5)

蛋白质精氨酸甲基转移酶 5 (PRMT5) 的变构调节

Palte, Rachel L; Schneider, Sebastian E; Altman, Michael D; Hayes, Robert P; Kawamura, Shuhei; Lacey, Brian M; Mansueto, My Sam; Reutershan, Michael; Siliphaivanh, Phieng; Sondey, Christopher; Xu, Haiyan; Xu, Zangwei; Ye, Yingchun; Machacek, Michelle R

Genome-Scale CRISPR Screens Identify Human Pluripotency-Specific Genes

基因组规模的 CRISPR 筛选可识别人类多能性特异性基因

Robert J Ihry, Max R Salick, Daniel J Ho, Marie Sondey, Sravya Kommineni, Steven Paula, Joe Raymond, Beata Henry, Elizabeth Frias, Qiong Wang, Kathleen A Worringer, Chaoyang Ye, Carsten Russ, John S Reece-Hoyes, Robert C Altshuler, Ranjit Randhawa, Zinger Yang, Gregory McAllister, Gregory R Hoffman,

The SENS algorithm-a new nutrient profiling system for food labelling in Europe

SENS算法——欧洲食品标签用新型营养成分分析系统

Darmon, Nicole; Sondey, Juliette; Azaïs-Braesco, Véronique; Maillot, Matthieu

The simplified nutrient profiling system (SENS) adequately ranks foods in relation to the overall nutritional quality of diets: a validation study

简化的营养成分分析系统(SENS)能够根据膳食的整体营养质量对食物进行充分排序:一项验证性研究

Maillot, Matthieu; Sondey, Juliette; Braesco, Véronique; Darmon, Nicole

Chronic Verubecestat Treatment Suppresses Amyloid Accumulation in Advanced Aged Tg2576-AβPPswe Mice Without Inducing Microhemorrhage

长期服用维鲁贝司他可抑制老年Tg2576-AβPPswe小鼠体内淀粉样蛋白的积累,且不诱发微出血

Villarreal, Stephanie; Zhao, Fuqiang; Hyde, Lynn A; Holder, Daniel; Forest, Thomas; Sondey, Marie; Chen, Xia; Sur, Cyrille; Parker, Eric M; Kennedy, Matthew E

Potent and Selective Amidopyrazole Inhibitors of IRAK4 That Are Efficacious in a Rodent Model of Inflammation

强效且选择性的IRAK4氨基吡唑抑制剂在啮齿动物炎症模型中有效

McElroy, William T; Tan, Zheng; Ho, Ginny; Paliwal, Sunil; Li, Guoqing; Seganish, W Michael; Tulshian, Deen; Tata, James; Fischmann, Thierry O; Sondey, Christopher; Bian, Hong; Bober, Loretta; Jackson, James; Garlisi, Charles G; Devito, Kristine; Fossetta, James; Lundell, Daniel; Niu, Xiaoda

Interaction of a neurotropic strain of Borrelia turicatae with the cerebral microcirculation system.

嗜神经性伯氏疏螺旋体菌株与脑微循环系统的相互作用

Sethi Nilay, Sondey Marie, Bai Yunhong, Kim Kwang S, Cadavid Diego