日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Favorable impact of PD1/PD-L1 antagonists on bone remodeling: an exploratory prospective clinical study and ex vivo validation

PD1/PD-L1 拮抗剂对骨重建的有利影响:一项探索性前瞻性临床研究和体外验证

Tamara Gassner, Christina Chittilappilly, Theo Pirich, Benjamin Neuditschko, Klaus Hackner, Judith Lind, Osman Aksoy, Uwe Graichen, Sascha Klee, Franz Herzog, Christoph Wiesner, Peter Errhalt, Martin Pecherstorfer, Klaus Podar, Sonia Vallet

JunB is a key regulator of multiple myeloma bone marrow angiogenesis

JunB 是多发性骨髓瘤骨髓血管生成的关键调节剂

Fengjuan Fan, Stefano Malvestiti, Sonia Vallet, Judith Lind, Jose Manuel Garcia-Manteiga, Eugenio Morelli, Qinyue Jiang, Anja Seckinger, Dirk Hose, Hartmut Goldschmidt, Andreas Stadlbauer, Chunyan Sun, Heng Mei, Martin Pecherstorfer, Latifa Bakiri, Erwin F Wagner, Giovanni Tonon, Martin Sattler, Yu

Rationally derived drug combinations with the novel Mcl-1 inhibitor EU-5346 in breast cancer

乳腺癌中新型 Mcl-1 抑制剂 EU-5346 的合理药物组合

Sonia Vallet, Fengjuan Fan, Stefano Malvestiti, Martin Pecherstorfer, Martin Sattler, Andreas Schneeweiss, Henning Schulze-Bergkamen, Joseph T Opferman, Michael H Cardone, Dirk Jäger, Klaus Podar

Mcl-1 confers protection of Her2-positive breast cancer cells to hypoxia: therapeutic implications

Mcl-1 保护 Her2 阳性乳腺癌细胞免于缺氧:治疗意义

Muhammad Hasan Bashari, Fengjuan Fan, Sonia Vallet, Martin Sattler, Melissa Arn, Claudia Luckner-Minden, Henning Schulze-Bergkamen, Inka Zörnig, Frederik Marme, Andreas Schneeweiss, Michael H Cardone, Joseph T Opferman, Dirk Jäger, Klaus Podar

Pre-Osteoblasts Stimulate Migration of Breast Cancer Cells via the HGF/MET Pathway

前成骨细胞通过 HGF/MET 通路刺激乳腺癌细胞迁移

Sonia Vallet, Muhammad Hasan Bashari, Feng-Juan Fan, Stefano Malvestiti, Andreas Schneeweiss, Patrick Wuchter, Dirk Jäger, Klaus Podar

Niche-Based Screening in Multiple Myeloma Identifies a Kinesin-5 Inhibitor with Improved Selectivity over Hematopoietic Progenitors

基于微环境的多发性骨髓瘤筛选鉴定出一种对造血祖细胞具有更高选择性的驱动蛋白-5抑制剂

Shrikanta Chattopadhyay ,Alison L Stewart ,Siddhartha Mukherjee ,Cherrie Huang ,Kimberly A Hartwell ,Peter G Miller ,Radhika Subramanian ,Leigh C Carmody ,Rushdia Z Yusuf ,David B Sykes ,Joshiawa Paulk ,Amedeo Vetere ,Sonia Vallet ,Loredana Santo ,Diana D Cirstea ,Teru Hideshima ,Vlado Dančík ,Max M Majireck ,Mahmud M Hussain ,Shambhavi Singh ,Ryan Quiroz ,Jonathan Iaconelli ,Rakesh Karmacharya ,Nicola J Tolliday ,Paul A Clemons ,Malcolm A S Moore ,Andrew M Stern ,Alykhan F Shamji ,Benjamin L Ebert ,Todd R Golub ,Noopur S Raje ,David T Scadden ,Stuart L Schreiber

Antimyeloma activity of a multitargeted kinase inhibitor, AT9283, via potent Aurora kinase and STAT3 inhibition either alone or in combination with lenalidomide

多靶点激酶抑制剂 AT9283 可通过强效抑制 Aurora 激酶和 STAT3 发挥抗骨髓瘤活性,单独使用或与来那度胺联合使用

Loredana Santo, Teru Hideshima, Diana Cirstea, Madhavi Bandi, Erik A Nelson, Gullu Gorgun, Scott Rodig, Sonia Vallet, Samantha Pozzi, Kishan Patel, Christine Unitt, Matt Squires, Yiguo Hu, Dharminder Chauhan, Anuj Mahindra, Nikhil C Munshi, Kenneth C Anderson, Noopur Raje

PI3K/p110{delta} is a novel therapeutic target in multiple myeloma

PI3K/p110{delta} 是多发性骨髓瘤的新治疗靶点

Hiroshi Ikeda, Teru Hideshima, Mariateresa Fulciniti, Giulia Perrone, Naoya Miura, Hiroshi Yasui, Yutaka Okawa, Tanyel Kiziltepe, Loredana Santo, Sonia Vallet, Diana Cristea, Elisabetta Calabrese, Gullu Gorgun, Noopur S Raje, Paul Richardson, Nikhil C Munshi, Brian J Lannutti, Kamal D Puri, Neill A

SNX-2112, a selective Hsp90 inhibitor, potently inhibits tumor cell growth, angiogenesis, and osteoclastogenesis in multiple myeloma and other hematologic tumors by abrogating signaling via Akt and ERK

SNX-2112 是一种选择性 Hsp90 抑制剂,可通过消除 Akt 和 ERK 信号传导,有效抑制多发性骨髓瘤和其他血液肿瘤中的肿瘤细胞生长、血管生成和破骨细胞生成

Yutaka Okawa, Teru Hideshima, Paul Steed, Sonia Vallet, Steven Hall, Ken Huang, John Rice, Amy Barabasz, Brianna Foley, Hiroshi Ikeda, Noopur Raje, Tanyel Kiziltepe, Hiroshi Yasui, Sotaro Enatsu, Kenneth C Anderson

Pharmacologic targeting of a stem/progenitor population in vivo is associated with enhanced bone regeneration in mice

体内干细胞/祖细胞群的药物靶向作用与小鼠骨再生增强相关

Siddhartha Mukherjee, Noopur Raje, Jesse A Schoonmaker, Julie C Liu, Teru Hideshima, Marc N Wein, Dallas C Jones, Sonia Vallet, Mary L Bouxsein, Samantha Pozzi, Shweta Chhetri, Y David Seo, Joshua P Aronson, Chirayu Patel, Mariateresa Fulciniti, Louise E Purton, Laurie H Glimcher, Jane B Lian, Gary