X-ray Crystallography-Guided Design, Antitumor Efficacy, and QSAR Analysis of Metabolically Stable Cyclopenta-Pyrimidinyl Dihydroquinoxalinone as a Potent Tubulin Polymerization Inhibitor
代谢稳定的环戊二烯并嘧啶基二氢喹喔啉酮作为强效微管蛋白聚合抑制剂的 X 射线晶体学指导设计、抗肿瘤功效和 QSAR 分析
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.1c01202
Souvik Banerjee, Foyez Mahmud, Shanshan Deng, Lingling Ma, Mi-Kyung Yun, Sayo O Fakayode, Kinsie E Arnst, Lei Yang, Hao Chen, Zhongzhi Wu, Pradeep B Lukka, Keyur Parmar, Bernd Meibohm, Stephen W White, Yuxi Wang, Wei Li, Duane D Miller