日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

In vivo screen of Plasmodium targets for mosquito-based malaria control

利用蚊媒控制疟疾的疟原虫靶标体内筛选

Probst, Alexandra S; Paton, Douglas G; Appetecchia, Federico; Bopp, Selina; Adams, Kelsey L; Rinvee, Tasneem A; Pou, Sovitj; Winter, Rolf; Du, Esrah W; Yahiya, Sabrina; Vidoudez, Charles; Singh, Naresh; Rodrigues, Janneth; Castañeda-Casado, Pablo; Tammaro, Chiara; Chen, Daisy; Godinez-Macias, Karla P; Jaramillo, Jasmine L; Poce, Giovanna; Rubal, Michael J; Nilsen, Aaron; Winzeler, Elizabeth A; Baum, Jake; Burrows, Jeremy N; Riscoe, Michael K; Wirth, Dyann F; Catteruccia, Flaminia

Structure, assembly and inhibition of the Toxoplasma gondii respiratory chain supercomplex

弓形虫呼吸链超复合物的结构、组装和抑制

Andrew E MacLean ,Shikha Shikha ,Mariana Ferreira Silva ,Max J Gramelspacher ,Aaron Nilsen ,Katherine M Liebman ,Sovitj Pou ,Rolf W Winter ,Amit Meir ,Michael K Riscoe ,J Stone Doggett ,Lilach Sheiner ,Alexander Mühleip

Long-acting intramuscular injections of ELQ-331, an antimalarial agent

长效肌注抗疟药ELQ-331

Karunakaran, Dipu; Mutyam, Shravan K; Fu, Melody; Chen, Jiaming; Pham, Kim Hue Nicky; Pou, Sovitj; Winter, Rolf W; Nilsen, Aaron; Dodean, Rozalia A; Smilkstein, Martin J; Riscoe, Michael K; Shankar, Gita

A fluorescence-based assay for measuring polyamine biosynthesis aminopropyl transferase-mediated catalysis

一种基于荧光的测定多胺生物合成氨丙基转移酶介导催化的方法

Pallavi Singh ,Jae-Yeon Choi ,Weiwei Wang ,Tukiet T Lam ,Philip Lechner ,Christopher D Vanderwal ,Sovitj Pou ,Aaron Nilsen ,Choukri Ben Mamoun

Effectiveness of Two New Endochin-like Quinolones, ELQ-596 and ELQ-650, in Experimental Mouse Models of Human Babesiosis

两种新型内切辛类喹诺酮类药物ELQ-596和ELQ-650在人类巴贝虫病实验小鼠模型中的疗效

Vydyam, Pratap; Chand, Meenal; Pou, Sovitj; Winter, Rolf W; Liebman, Katherine M; Nilsen, Aaron; Doggett, J Stone; Riscoe, Michael K; Ben Mamoun, Choukri

3-Position Biaryl Endochin-like Quinolones with Enhanced Antimalarial Performance

具有增强抗疟性能的3位联芳基内切辛类喹诺酮

Pou, Sovitj; Winter, Rolf W; Dodean, Rozalia A; Liebman, Katherine; Li, Yuexin; Mather, Michael W; Nepal, Binod; Nilsen, Aaron; Handford, Mason J; Riscoe, Teresa M; Laxson, Sydney; Kirtley, Payton J; Aleshnick, Maya; Zakharov, Lev N; Kelly, Jane X; Smilkstein, Martin J; Wilder, Brandon K; Kortagere, Sandhya; Vaidya, Akhil B; Alday, P Holland; Doggett, J Stone; Riscoe, Michael K

Synthesis of Deuterated Endochin-Like Quinolones

氘代内切辛类喹诺酮的合成

Pou, Sovitj; Winter, Rolf W; Liebman, Katherine M; Dodean, Rosie A; Nilsen, Aaron; DeBarber, Andrea; Doggett, J Stone; Riscoe, Michael K

Effective Therapy Targeting Cytochrome bc(1) Prevents Babesia Erythrocytic Development and Protects from Lethal Infection.

针对细胞色素bc(1)的有效疗法可预防巴贝虫红细胞发育并防止致命感染

Chiu Joy E, Renard Isaline, Pal Anasuya C, Singh Pallavi, Vydyam Pratap, Thekkiniath Jose, Kumar Madelyn, Gihaz Shalev, Pou Sovitj, Winter Rolf W, Dodean Rozalia, Frueh Lisa, Nilsen Aaron C, Riscoe Michael K, Doggett J Stone, Mamoun Choukri Ben

A New Scalable Synthesis of ELQ-300, ELQ-316, and other Antiparasitic Quinolones

ELQ-300、ELQ-316 和其他抗寄生虫喹诺酮类药物的新型可扩展合成方法

Sovitj Pou, Rozalia A Dodean, Lisa Frueh, Katherine M Liebman, Rory T Gallagher, Haihong Jin, Robert T Jacobs, Aaron Nilsen, David R Stuart, J Stone Doggett, Michael K Riscoe, Rolf W Winter

Novel Endochin-Like Quinolones Exhibit Potent In Vitro Activity against Plasmodium knowlesi but Do Not Synergize with Proguanil

新型内皮素样喹诺酮类药物对诺氏疟原虫具有强效体外活性,但与氯胍无协同作用

Donelly A van Schalkwyk, Michael K Riscoe, Sovitj Pou, Rolf W Winter, Aaron Nilsen, Maëlle Duffey, Robert W Moon, Colin J Sutherland