日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Favorable Preclinical Pharmacological Profile of a Novel Antimalarial Pyrrolizidinylmethyl Derivative of 4-amino-7-chloroquinoline with Potent In Vitro and In Vivo Activities

一种新型抗疟吡咯里西啶甲基衍生物(4-氨基-7-氯喹啉)具有良好的临床前药理学特性,并表现出强大的体外和体内活性。

Basilico, Nicoletta; Parapini, Silvia; D'Alessandro, Sarah; Misiano, Paola; Romeo, Sergio; Dondio, Giulio; Yardley, Vanessa; Vivas, Livia; Nasser, Shereen; Rénia, Laurent; Russell, Bruce M; Suwanarusk, Rossarin; Nosten, François; Sparatore, Anna; Taramelli, Donatella

3,3-Disubstituted 3,4-Dihydro-1,2,4-benzotriazines: Chemistry, Biological Activity, and Affinity to Sigma Receptors

3,3-二取代的3,4-二氢-1,2,4-苯并三嗪:化学性质、生物活性及对σ受体的亲和力

Sparatore, Fabio; Sparatore, Anna

Further Quinolizidine Derivatives as Antiarrhythmic Agents- 3

喹诺里西啶衍生物作为抗心律失常药物的进一步研究-3

Tasso, Bruno; Mattioli, Laura Beatrice; Tonelli, Michele; Boido, Vito; Chiarini, Alberto; Sparatore, Fabio; Budriesi, Roberta

MZe786, a hydrogen sulfide-releasing aspirin prevents preeclampsia in heme oxygenase-1 haplodeficient pregnancy under high soluble flt-1 environment

MZe786,一种释放硫化氢的阿司匹林,可在高可溶性Flt-1环境下预防血红素加氧酶-1单倍体缺陷妊娠中的先兆子痫。

Rezai, Homira; Ahmad, Shakil; Alzahrani, Faisal A; Sanchez-Aranguren, Lissette; Dias, Irundika Hk; Agrawal, Swati; Sparatore, Anna; Wang, Keqing; Ahmed, Asif

Hydrogen sulfide releasing molecule MZe786 inhibits soluble Flt-1 and prevents preeclampsia in a refined RUPP mouse model

硫化氢释放分子MZe786抑制可溶性Flt-1,并在改良的RUPP小鼠模型中预防先兆子痫。

Saif, Jaimy; Ahmad, Shakil; Rezai, Homira; Litvinova, Karina; Sparatore, Anna; Alzahrani, Faisal A; Wang, Keqing; Ahmed, Asif

Design, Synthesis and In Vitro Investigation of Novel Basic Celastrol Carboxamides as Bio-Inspired Leishmanicidal Agents Endowed with Inhibitory Activity against Leishmania Hsp90

新型碱性雷公藤红素酰胺作为具有利什曼原虫 Hsp90 抑制活性的仿生利什曼杀虫剂的设计、合成及体外研究

Ivan Bassanini, Silvia Parapini, Erica E Ferrandi, Elena Gabriele, Nicoletta Basilico, Donatella Taramelli, Anna Sparatore

Superior Properties of N-Acetylcysteine Ethyl Ester over N-Acetyl Cysteine to Prevent Retinal Pigment Epithelial Cells Oxidative Damage

N-乙酰半胱氨酸乙酯在预防视网膜色素上皮细胞氧化损伤方面优于 N-乙酰半胱氨酸

Gian Marco Tosi, Daniela Giustarini, Lorenzo Franci, Alberto Minetti, Francesco Imperatore, Elena Caldi, Paolo Fiorenzani, Anna Maria Aloisi, Anna Sparatore, Ranieri Rossi, Mario Chiariello, Maurizio Orlandini, Federico Galvagni

Benzimidazole derivatives endowed with potent antileishmanial activity

具有强效抗利什曼原虫活性的苯并咪唑衍生物

Tonelli, Michele; Gabriele, Elena; Piazza, Francesca; Basilico, Nicoletta; Parapini, Silvia; Tasso, Bruno; Loddo, Roberta; Sparatore, Fabio; Sparatore, Anna

New sulfurated derivatives of cinnamic acids and rosmaricine as inhibitors of STAT3 and NF-κB transcription factors

肉桂酸和迷迭香碱的新型硫化衍生物作为 STAT3 和 NF-κB 转录因子的抑制剂

Elena Gabriele, Dario Brambilla, Chiara Ricci, Luca Regazzoni, Kyoko Taguchi, Nicola Ferri, Akira Asai, Anna Sparatore

In Vivo and In Vitro Activities and ADME-Tox Profile of a Quinolizidine-Modified 4-Aminoquinoline: A Potent Anti-P. falciparum and Anti-P. vivax Blood-Stage Antimalarial

喹诺里西啶修饰的 4-氨基喹啉的体内和体外活性以及 ADME-Tox 特性:一种有效的抗恶性疟原虫和抗间日疟原虫血液阶段抗疟药

Nicoletta Basilico, Silvia Parapini, Anna Sparatore, Sergio Romeo, Paola Misiano, Livia Vivas, Vanessa Yardley, Simon L Croft, Annette Habluetzel, Leonardo Lucantoni, Laurent Renia, Bruce Russell, Rossarin Suwanarusk, Francois Nosten, Giulio Dondio, Chiara Bigogno, Daniela Jabes, Donatella Taramelli