日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Butyrolactol A enhances caspofungin efficacy via flippase inhibition in drug-resistant fungi.

丁内酯 A 通过抑制抗药真菌中的翻转酶来增强卡泊芬净的疗效。

Chen Xuefei, Duan H Diessel, Hoy Michael J, Koteva Kalinka, Spitzer Michaela, Guitor Allison K, Puumala Emily, Fiebig Aline A, Hu Guanggan, Yiu Bonnie, Chou Sommer, Bian Zhuyun, Choi Yeseul, Guo Amelia Bing Ya, Wang Wenliang, Sun Sheng, Robbins Nicole, Averette Anna Floyd, Cook Michael A, Truant Ray, MacNeil Lesley T, Brown Eric D, Kronstad James W, Coombes Brian K, Cowen Leah E, Heitman Joseph, Li Huilin, Wright Gerard D

Butyrolactol A potentiates caspofungin efficacy against resistant fungi via phospholipid flippase inhibition

丁内酯A通过抑制磷脂翻转酶增强卡泊芬净对耐药真菌的疗效

Chen, Xuefei; Diessel Duan, H; Hoy, Michael J; Koteva, Kalinka; Spitzer, Michaela; Guitor, Allison K; Puumala, Emily; Fiebig, Aline A; Hu, Guanggan; Yiu, Bonnie; Chou, Sommer; Bian, Zhuyun; Choi, Yeseul; Guo, Amelia Bing Ya; Wang, Wenliang; Sun, Sheng; Robbins, Nicole; Averette, Anna Floyd; Cook, Michael A; Truant, Ray; MacNeil, Lesley T; Brown, Eric D; Kronstad, James W; Coombes, Brian K; Cowen, Leah E; Heitman, Joseph; Li, Huilin; Wright, Gerard D

Open Targets Platform: supporting systematic drug-target identification and prioritisation

开放靶点平台:支持系统性的药物靶点识别和优先级排序

Ochoa, David; Hercules, Andrew; Carmona, Miguel; Suveges, Daniel; Gonzalez-Uriarte, Asier; Malangone, Cinzia; Miranda, Alfredo; Fumis, Luca; Carvalho-Silva, Denise; Spitzer, Michaela; Baker, Jarrod; Ferrer, Javier; Raies, Arwa; Razuvayevskaya, Olesya; Faulconbridge, Adam; Petsalaki, Eirini; Mutowo, Prudence; Machlitt-Northen, Sandra; Peat, Gareth; McAuley, Elaine; Ong, Chuang Kee; Mountjoy, Edward; Ghoussaini, Maya; Pierleoni, Andrea; Papa, Eliseo; Pignatelli, Miguel; Koscielny, Gautier; Karim, Mohd; Schwartzentruber, Jeremy; Hulcoop, David G; Dunham, Ian; McDonagh, Ellen M

ALDH2 Mediates 5-Nitrofuran Activity in Multiple Species

ALDH2介导多种物种中的5-硝基呋喃活性

Zhou, Linna; Ishizaki, Hironori; Spitzer, Michaela; Taylor, Kerrie L; Temperley, Nicholas D; Johnson, Stephen L; Brear, Paul; Gautier, Philippe; Zeng, Zhiqiang; Mitchell, Amy; Narayan, Vikram; McNeil, Ewan M; Melton, David W; Smith, Terry K; Tyers, Mike; Westwood, Nicholas J; Patton, E Elizabeth

Applications of machine learning in drug discovery and development

机器学习在药物发现和开发中的应用

Vamathevan, Jessica; Clark, Dominic; Czodrowski, Paul; Dunham, Ian; Ferran, Edgardo; Lee, George; Li, Bin; Madabhushi, Anant; Shah, Parantu; Spitzer, Michaela; Zhao, Shanrong

Zebrafish MITF-Low Melanoma Subtype Models Reveal Transcriptional Subclusters and MITF-Independent Residual Disease

斑马鱼MITF低表达黑色素瘤亚型模型揭示转录亚簇和MITF非依赖性残留疾病

Travnickova, Jana; Wojciechowska, Sonia; Khamseh, Ava; Gautier, Philippe; Brown, Daniel V; Lefevre, Thomas; Brombin, Alessandro; Ewing, Ailith; Capper, Amy; Spitzer, Michaela; Dilshat, Ramile; Semple, Colin A; Mathers, Marie E; Lister, James A; Steingrimsson, Eiríkur; Voet, Thierry; Ponting, Chris P; Patton, E Elizabeth

Open Targets Platform: new developments and updates two years on

开放目标平台:两年来的新进展和更新

Carvalho-Silva, Denise; Pierleoni, Andrea; Pignatelli, Miguel; Ong, ChuangKee; Fumis, Luca; Karamanis, Nikiforos; Carmona, Miguel; Faulconbridge, Adam; Hercules, Andrew; McAuley, Elaine; Miranda, Alfredo; Peat, Gareth; Spitzer, Michaela; Barrett, Jeffrey; Hulcoop, David G; Papa, Eliseo; Koscielny, Gautier; Dunham, Ian

Combinatorial strategies for combating invasive fungal infections

对抗侵袭性真菌感染的组合策略

Spitzer, Michaela; Robbins, Nicole; Wright, Gerard D

Systematic chemical-genetic and chemical-chemical interaction datasets for prediction of compound synergism.

用于预测化合物协同作用的系统化学遗传和化学化学相互作用数据集

Wildenhain Jan, Spitzer Michaela, Dolma Sonam, Jarvik Nick, White Rachel, Roy Marcia, Griffiths Emma, Bellows David S, Wright Gerard D, Tyers Mike

An Antifungal Combination Matrix Identifies a Rich Pool of Adjuvant Molecules that Enhance Drug Activity against Diverse Fungal Pathogens

抗真菌组合基质鉴定出丰富的佐剂分子库,这些分子可增强药物对多种真菌病原体的活性。

Robbins, Nicole; Spitzer, Michaela; Yu, Tennison; Cerone, Robert P; Averette, Anna K; Bahn, Yong-Sun; Heitman, Joseph; Sheppard, Donald C; Tyers, Mike; Wright, Gerard D