Discovery of VU6028418: A Highly Selective and Orally Bioavailable M4 Muscarinic Acetylcholine Receptor Antagonist
发现 VU6028418:一种高选择性且口服生物可利用的 M4 毒蕈碱乙酰胆碱受体拮抗剂
期刊:ACS Medicinal Chemistry Letters
影响因子:3.5
doi:10.1021/acsmedchemlett.1c00363
Matthew Spock, Trever R Carter, Katrina A Bollinger, Changho Han, Logan A Baker, Alice L Rodriguez, Li Peng, Jonathan W Dickerson, Aidong Qi, Jerri M Rook, Jordan C O'Neill, Katherine J Watson, Sichen Chang, Thomas M Bridges, Julie L Engers, Darren W Engers, Colleen M Niswender, P Jeffrey Conn, Crai