日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Chemoprevention of Preclinical Breast and Lung Cancer with the Bromodomain Inhibitor I-BET 762

利用溴结构域抑制剂 I-BET 762 对临床前乳腺癌和肺癌进行化学预防

Zhang, Di; Leal, Ana S; Carapellucci, Sarah; Zydeck, Kayla; Sporn, Michael B; Liby, Karen T

The triterpenoid CDDO-imidazolide reduces immune cell infiltration and cytokine secretion in the KrasG12D;Pdx1-Cre (KC) mouse model of pancreatic cancer

三萜类化合物CDDO-咪唑化物可减少KrasG12D;Pdx1-Cre (KC)小鼠胰腺癌模型中的免疫细胞浸润和细胞因子分泌。

Leal, Ana S; Sporn, Michael B; Pioli, Patricia A; Liby, Karen T

The Nrf2 triterpenoid activator, CDDO-imidazolide, protects kidneys from ischemia-reperfusion injury in mice

Nrf2三萜类激活剂CDDO-咪唑化物可保护小鼠肾脏免受缺血再灌注损伤。

Liu, Manchang; Reddy, Narsa M; Higbee, Elizabeth M; Potteti, Haranatha R; Noel, Sanjeev; Racusen, Lorraine; Kensler, Thomas W; Sporn, Michael B; Reddy, Sekhar P; Rabb, Hamid

Targeting Nrf2-mediated gene transcription by extremely potent synthetic triterpenoids attenuate dopaminergic neurotoxicity in the MPTP mouse model of Parkinson's disease

利用高效合成三萜类化合物靶向Nrf2介导的基因转录,可减轻MPTP诱导的帕金森病小鼠模型中的多巴胺能神经毒性。

Kaidery, Navneet Ammal; Banerjee, Rebecca; Yang, Lichuan; Smirnova, Natalya A; Hushpulian, Dmitry M; Liby, Karen T; Williams, Charlotte R; Yamamoto, Masayuki; Kensler, Thomas W; Ratan, Rajiv R; Sporn, Michael B; Beal, M Flint; Gazaryan, Irina G; Thomas, Bobby

NADPH oxidase and Nrf2 regulate gastric aspiration-induced inflammation and acute lung injury.

NADPH 氧化酶和 Nrf2 调节胃吸入引起的炎症和急性肺损伤

Davidson Bruce A, Vethanayagam R Robert, Grimm Melissa J, Mullan Barbara A, Raghavendran Krishnan, Blackwell Timothy S, Freeman Michael L, Ayyasamy Vanniarajan, Singh Keshav K, Sporn Michael B, Itagaki Kiyoshi, Hauser Carl J, Knight Paul R, Segal Brahm H

NRF2 and cancer: the good, the bad and the importance of context

NRF2与癌症:利弊及背景的重要性

Sporn, Michael B; Liby, Karen T

Synthetic oleanane triterpenoids: multifunctional drugs with a broad range of applications for prevention and treatment of chronic disease

合成齐墩果烷三萜类化合物:多功能药物,在慢性疾病的预防和治疗中具有广泛的应用前景

Liby, Karen T; Sporn, Michael B

Triterpenoid modulation of IL-17 and Nrf-2 expression ameliorates neuroinflammation and promotes remyelination in autoimmune encephalomyelitis

三萜类化合物对IL-17和Nrf-2表达的调节可减轻自身免疫性脑脊髓炎的神经炎症并促进髓鞘再生。

Pareek, Tej K; Belkadi, Abdelmadjid; Kesavapany, Sashi; Zaremba, Anita; Loh, Sook L; Bai, Lianhua; Cohen, Mark L; Meyer, Colin; Liby, Karen T; Miller, Robert H; Sporn, Michael B; Letterio, John J

CDDO-imidazolide induces DNA damage, G2/M arrest and apoptosis in BRCA1-mutated breast cancer cells

CDDO-咪唑利德可诱导BRCA1突变乳腺癌细胞的DNA损伤、G2/M期阻滞和细胞凋亡。

Kim, Eun-Hee; Deng, Chu-Xia; Sporn, Michael B; Liby, Karen T

NADPH oxidase limits innate immune responses in the lungs in mice

NADPH氧化酶限制小鼠肺部的先天免疫反应。

Segal, Brahm H; Han, Wei; Bushey, Jennifer J; Joo, Myungsoo; Bhatti, Zahida; Feminella, Joy; Dennis, Carly G; Vethanayagam, R Robert; Yull, Fiona E; Capitano, Maegan; Wallace, Paul K; Minderman, Hans; Christman, John W; Sporn, Michael B; Chan, Jefferson; Vinh, Donald C; Holland, Steven M; Romani, Luigina R; Gaffen, Sarah L; Freeman, Michael L; Blackwell, Timothy S