日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A small-molecule modulator of cardiac myosin acts on multiple stages of the myosin chemomechanical cycle

一种小分子调节剂可调控心肌肌球蛋白,作用于肌球蛋白化学机械循环的多个阶段。

Kawas, Raja F; Anderson, Robert L; Ingle, Sadie R Bartholomew; Song, Yonghong; Sran, Arvinder S; Rodriguez, Hector M

Preclinical characterization of Aurora kinase inhibitor R763/AS703569 identified through an image-based phenotypic screen.

通过基于图像的表型筛选鉴定的 Aurora 激酶抑制剂 R763/AS703569 的临床前表征

McLaughlin John, Markovtsov Vadim, Li Hui, Wong Steve, Gelman Marina, Zhu Yanhong, Franci Christian, Lang D Wayne, Pali Erlina, Lasaga Joe, Low Caroline, Zhao Feifei, Chang Betty, Gururaja Tarikere L, Xu Weiduan, Baluom Muhammad, Sweeny David, Carroll David, Sran Arvinder, Thota Sambaiah, Parmer Manjeet, Romane Angela, Clemens George, Grossbard Elliott, Qu Kunbin, Jenkins Yonchu, Kinoshita Taisei, Taylor Vanessa, Holland Sacha J, Argade Ankush, Singh Rajinder, Pine Polly, Payan Donald G, Hitoshi Yasumichi