日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Mechanism and function of GPR3 regulated by a negative allosteric modulator.

负变构调节剂调控 GPR3 的机制和功能

Chen Geng, Bláhová Jana, Staffen Nico, Hübner Harald, Nunhöfer Nadja, Qiu Chen, Gmeiner Peter, Weikert Dorothee, Du Yang, Xu Jun

Discovery of a functionally selective serotonin receptor (5-HT(1A)R) agonist for the treatment of pain.

发现一种功能选择性血清素受体(5-HT(1A)R)激动剂用于治疗疼痛

Ullrich Annika, Schneider Johannes, Braz João M, Neu Eduard, Staffen Nico, Stanek Markus, Bláhová Jana, Hove Tamsanqa, Albert Tamara, Allikalt Anni, Löber Stefan, Bhardwaj Karnika, Rodriguez-Rosado Sian, Fink Elissa, Rasmussen Tim, Hübner Harald, Inoue Asuka, Shoichet Brian K, Basbaum Allan I, Böttcher Bettina, Weikert Dorothee, Gmeiner Peter

Structural and functional characterization of the endogenous agonist for orphan receptor GPR3

孤儿受体GPR3内源性激动剂的结构和功能表征

Chen, Geng; Staffen, Nico; Wu, Zhangsong; Xu, Xinyu; Pan, Jinheng; Inoue, Asuka; Shi, Tingyi; Gmeiner, Peter; Du, Yang; Xu, Jun