日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural and Functional Analyses of Trypanosoma brucei Nucleoside Diphosphate Kinase

布氏锥虫核苷二磷酸激酶的结构和功能分析

Makori, Patricia; Boeckman, Michael P; David, Heidi S; Payne, Finley; Gatling, Markenya; Greer, Colby; Hayes, Dylan; Jefferson, Alexandra; Maxwell, Micaela; Smith, Christian; Watson, Jamilah; Williams, London; Barkley, Jazmin; Pepper, Caitlyn; Zininga, Tawanda; Subramanian, Sandhya; Abramov, Ariel; Gardberg, Anna S; Edwards, Thomas E; Staker, Bart L; Stewart, Lance J; Myler, Peter J; Asojo, Oluwatoyin A; Jeje, Olamide; Fanucchi, Sylvia; Achilonu, Ikechukwu; Smith, Craig L; Chakafana, Graham

Crystal structure of carbon-nitrogen hydrolase from Helicobacter pylori G27

幽门螺杆菌G27碳氮水解酶的晶体结构

Srivastava, Aruesha; Ayanlade, Jesuferanmi P; Suleiman, Lema; Udell, Hannah; Abendroth, Jan; Lorimer, Donald J; Edwards, Thomas E; Staker, Bart L; Zigweid, Rachael; Subramanian, Sandhya; Myler, Peter J; Chakafana, Graham; Asojo, Oluwatoyin A

Discovery and mechanism of a highly selective, antifungal acetyl-CoA synthetase inhibitor

发现并阐明了一种高选择性抗真菌乙酰辅酶A合成酶抑制剂的作用机制

Jezewski, Andrew J; Alden, Katy M; Propp, Jonah; Daraji, Drashti G; Lail, Charles L 3rd; Heene, Michael E; Fuller, Andrew J; Ferreira, Jeffery C; Liu, Lijun; Battaile, Kevin P; Williams, Noelle S; Staker, Bart L; Lovell, Scott; Hagen, Timothy J; Krysan, Damian J

Architecture of Pseudomonas aeruginosa glutamyl-tRNA synthetase defines a subfamily of dimeric class Ib aminoacyl-tRNA synthetases

铜绿假单胞菌谷氨酰-tRNA合成酶的结构定义了二聚体Ib类氨酰-tRNA合成酶的一个亚家族。

Fenwick, Michael K; Mayclin, Stephen J; Seibold, Steve; DeRocher, Amy E; Subramanian, Sandhya; Phan, Isabelle Q; Dranow, David M; Lorimer, Donald D; Abramov, Ariel B; Choi, Ryan; Hewitt, Stephen Nakazawa; Edwards, Thomas E; Bullard, James M; Battaile, Kevin P; Wower, Iwona K; Soe, Aimee C; Tsutakawa, Susan E; Lovell, Scott; Myler, Peter J; Wower, Jacek; Staker, Bart L

Bumped Kinase Inhibitors Inhibit both Toxoplasma gondii MAPKL1 and CDPK1

激酶抑制剂可同时抑制弓形虫 MAPKL1 和 CDPK1。

Montgomery, Jemma A; Alday, P Holland; Choi, Ryan; Khim, Monique; Staker, Bart L; Hulverson, Matthew A; Ojo, Kayode K; Fan, Erkang; Van Voorhis, Wesley C; Doggett, J Stone

Versatile Imidazole Scaffold with Potent Activity against Multiple Apicomplexan Parasites.

多功能咪唑骨架,对多种顶复门寄生虫具有强效活性

Khim Monique, Montgomery Jemma, Laureano De Souza Mariana, Delvillar Melvin, Weible Lyssa J, Prabakaran Mayuri, Hulverson Matthew A, Eck Tyler, Bheemanabonia Rammohan Y, Alday P Holland, Rotella David P, Doggett J Stone, Staker Bart L, Ojo Kayode K, Bhanot Purnima

Crystal structures of Mycobacterium tuberculosis and Mycobacterium thermoresistibile glycyl-tRNA synthetases in various liganded states

结核分枝杆菌和耐热分枝杆菌甘氨酰-tRNA合成酶在不同配体结合状态下的晶体结构

Fenwick, Michael K; DeRocher, Amy E; Craig, Justin K; Harmon, Elizabeth K; Seibold, Steve; Liu, Lijun; Battaile, Kevin P; Barrett, Lynn K; Van Voorhis, Wesley C; Phan, Isabelle Q; Staker, Bart L; Subramanian, Sandhya; Lovell, Scott; Myler, Peter J

Structure guided modification of 2-chloro-5-(ethyl-phenyl-sulfamoyl)-N-[2-(2-oxo-pyrrolidin-1-yl)-phenyl]-benzamide to afford selective inhibitors of Cryptosporidium parvum N-myristoyltransferase

以2-氯-5-(乙基苯基磺酰基)-N-[2-(2-氧代吡咯烷-1-基)苯基]-苯甲酰胺为模板,构建选择性小隐孢子虫N-肉豆蔻酰转移酶抑制剂

Sigalapalli, Dilep K; Groustra, Sophia; Fenwick, Michael K; Zigweid, Rachael; Hulverson, Matthew A; Owsley, Eric; Khim, Monique; Shibata, Sayaka; Van Voorhis, Wesley C; Staker, Bart L; Fan, Erkang

The crystal structures of apo and tryptophan-bound tryptophanyl-tRNA synthetase from Neisseria gonorrhoeae

淋病奈瑟菌的脱辅基和色氨酸结合的色氨酰-tRNA合成酶的晶体结构

Baral, Jessika; Song, David; Edwards, Thomas E; Dranow, David M; Lorimer, Donald D; Staker, Bart L; Myler, Peter; Smith, Craig L

Analysis of Burkholderia pseudomallei IspF in complex with sulfapyridine, sulfamonomethoxine, ethoxzolamide and acetazolamide

分析类鼻疽伯克霍尔德菌 IspF 与磺胺吡啶、磺胺甲氧嘧啶、乙氧唑胺和乙酰唑胺的复合物

Grote, Dakota; Stewart, Christopher G; Daraji, Drashti G; Enayati, Parisa; Braverman, Kristina N; Romanaggi, CeAnn; Bolejack, Madison J; Yano, Jason K; Abendroth, Jan; Dranow, David M; Pierce, Phillip G; Lorimer, Donald D; Horanyi, Peter S; Staker, Bart L; Edwards, Thomas E; Myler, Peter J; Horn, James R; Hagen, Timothy J