日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of a functionally selective serotonin receptor (5-HT(1A)R) agonist for the treatment of pain.

发现一种功能选择性血清素受体(5-HT(1A)R)激动剂用于治疗疼痛

Ullrich Annika, Schneider Johannes, Braz João M, Neu Eduard, Staffen Nico, Stanek Markus, Bláhová Jana, Hove Tamsanqa, Albert Tamara, Allikalt Anni, Löber Stefan, Bhardwaj Karnika, Rodriguez-Rosado Sian, Fink Elissa, Rasmussen Tim, Hübner Harald, Inoue Asuka, Shoichet Brian K, Basbaum Allan I, Böttcher Bettina, Weikert Dorothee, Gmeiner Peter

An allosteric modulator binds to a conformational hub in the β(2) adrenergic receptor.

变构调节剂与β(2)肾上腺素能受体的构象枢纽结合

Liu Xiangyu, Kaindl Jonas, Korczynska Magdalena, Stößel Anne, Dengler Daniela, Stanek Markus, Hübner Harald, Clark Mary J, Mahoney Jake, Matt Rachel Ann, Xu Xinyu, Hirata Kunio, Shoichet Brian K, Sunahara Roger K, Kobilka Brian K, Gmeiner Peter