日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Novel G Protein-Biased Agonist at the δ Opioid Receptor with Analgesic Efficacy in Models of Chronic Pain

一种新型的δ阿片受体G蛋白偏向性激动剂,在慢性疼痛模型中具有镇痛功效

Conibear, Alexandra E; Asghar, Junaid; Hill, Rob; Henderson, Graeme; Borbely, Eva; Tekus, Valeria; Helyes, Zsuzsanna; Palandri, Josephine; Bailey, Chris; Starke, Ingemar; von Mentzer, Bengt; Kendall, David; Kelly, Eamonn

Discovery of a Series of Indole-2 Carboxamides as Selective Secreted Phospholipase A(2) Type X (sPLA(2)-X) Inhibitors.

发现一系列吲哚-2 甲酰胺类化合物作为选择性分泌型磷脂酶 A(2) X 型 (sPLA(2)-X) 抑制剂

Knerr Laurent, Giordanetto Fabrizio, Nordberg Peter, Pettersen Daniel, Selmi Nidhal, Beisel Hans-Georg, de la Motte Hannah, Olsson Thomas, Perkins Tim D J, Herslöf Margareta, Månsson à sa, Dahlström Mikael, Starke Ingemar, Broddefalk Johan, Saarinen Gabrielle, Klingegård Fredrik, Hurt-Camejo Eva, Rosengren Birgitta, Brengdahl Johan, Jansen Frank, Rohman Mattias, Sandmark Jenny, Hallberg Kenth, à kerud Tomas, Roth Robert G, Ahlqvist Marie