日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Nanocrystallization Effectively Improves the Oral Efficacy of an Antileishmanial Chalcone

纳米晶化有效提高了抗利什曼原虫查尔酮的口服疗效。

Borsodi, Maria Paula Gonçalves; Pacienza-Lima, Wallace; Menezes, Jaqueline Correia Villaça; Escrivani-Oliveira, Douglas; Arruda-Costa, Natalia; Silva, Alcides José Monteiro da; Cabral, Lucio Mendes; Steel, Patrick G; Sousa-Batista, Ariane de Jesus; Rossi-Bergmann, Bartira

Activity-based chemoproteomic profiling reveals the active kinome of Leishmania

基于活性的化学蛋白质组学分析揭示了利什曼原虫的活性激酶组

Porta, Exequiel O J; Kalesh, Karunakaran; Steel, Patrick G

Simple accessible clemastine fumarate analogues as effective antileishmanials

简单易得的富马酸克立马汀类似物作为有效的抗利什曼原虫药物

Charlton, Rebecca L; Escrivani, Douglas O; Brown, Christopher; Thota, Niranjan; Agostino, Victor S; Porta, Exequiel O J; Avkiran, Timur; Merritt, Andrew T; Denny, Paul W; Rossi-Bergmann, Bartira; Steel, Patrick G

Profiling Serine Hydrolases in the Leishmania Host-Pathogen Interactome Using Cell-Permeable Activity-Based Fluorophosphonate Probes

利用细胞渗透性活性氟膦酸酯探针分析利什曼原虫宿主-病原体相互作用组中的丝氨酸水解酶

Isern, Jaime A; Porta, Exequiel O J; Kalesh, Karunakaran; Koutsogiannis, Zisis; Cazzola, Davide; Pohl, Ehmke; Denny, Paul W; Steel, Patrick G

Applications of Transition Metal-Catalyzed ortho-Fluorine-Directed C-H Functionalization of (Poly)fluoroarenes in Organic Synthesis

过渡金属催化邻位氟导向的(多)氟代芳烃CH官能化在有机合成中的应用

Budiman, Yudha P; Perutz, Robin N; Steel, Patrick G; Radius, Udo; Marder, Todd B

Navigating drug repurposing for Chagas disease: advances, challenges, and opportunities

探索药物再利用在恰加斯病治疗中的应用:进展、挑战与机遇

Porta, Exequiel O J; Kalesh, Karunakaran; Steel, Patrick G

Synthesis and vectorial functionalisation of pyrazolo[3,4-c]pyridines

吡唑并[3,4-c]吡啶的合成及矢量功能化

Bedwell, Elizabeth V; da Silva Emery, Flavio; Clososki, Giuliano C; Steel, Patrick G

Assessing Dose-Exposure-Response Relationships of Miltefosine in Adults and Children using Physiologically-Based Pharmacokinetic Modeling Approach

采用基于生理的药代动力学模型方法评估米替福新在成人和儿童中的剂量-暴露-反应关系

Madu, Shadrack J; Wang, Ke; Chirumamilla, Siri Kalyan; Turner, David B; Steel, Patrick G; Li, Mingzhong

Inhibition of HSP90 distinctively modulates the global phosphoproteome of Leishmania mexicana developmental stages.

抑制 HSP90 可显著调节墨西哥利什曼原虫发育阶段的整体磷酸化蛋白质组

Porta Exequiel O, Gao Liqian, Denny Paul W, Steel Patrick G, Kalesh Karunakaran

Activity-based protein profiling: A graphical review

基于活性的蛋白质谱分析:图解综述

Porta, Exequiel O J; Steel, Patrick G