Noncompetitive antagonism and inverse agonism as mechanism of action of nonpeptidergic antagonists at primate and rodent CXCR3 chemokine receptors
非竞争性拮抗和逆向激动是非肽能拮抗剂对灵长类和啮齿类 CXCR3 趋化因子受体的作用机制
期刊:Journal of Pharmacology and Experimental Therapeutics
影响因子:3.1
doi:10.1124/jpet.107.134783
Dennis Verzijl, Stefania Storelli, Danny J Scholten, Leontien Bosch, Todd A Reinhart, Daniel N Streblow, Cornelis P Tensen, Carlos P Fitzsimons, Guido J R Zaman, James E Pease, Iwan J P de Esch, Martine J Smit, Rob Leurs