日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Virtual screening of ultra-large chemical libraries identifies cell-permeable small-molecule inhibitors of a "non-druggable" target, STAT3 N-terminal domain

通过对超大型化合物库进行虚拟筛选,鉴定出可渗透细胞的小分子抑制剂,这些抑制剂针对的是一种“不可成药”靶点——STAT3 N端结构域。

Bonilla, Pedro Andrade; Hoop, Cody L; Stefanisko, Karen; Tarasov, Sergey G; Sinha, Sourav; Nicklaus, Marc C; Tarasova, Nadya I

Host Directed Therapy for Chronic Tuberculosis via Intrapulmonary Delivery of Aerosolized Peptide Inhibitors Targeting the IL-10-STAT3 Pathway

通过肺内输送针对 IL-10-STAT3 通路的气雾化肽抑制剂进行宿主定向治疗慢性结核病

Rashmi Upadhyay, Andrea Sanchez-Hidalgo, Carol J Wilusz, Anne J Lenaerts, Jennifer Arab, Joanna Yeh, Karen Stefanisko, Nadya I Tarasova, Mercedes Gonzalez-Juarrero

Mycobacterium tuberculosis copper-regulated protein SocB is an intrinsically disordered protein that folds upon interaction with a synthetic phospholipid bilayer

结核分枝杆菌铜调控蛋白SocB是一种固有无序蛋白,它在与合成磷脂双层相互作用时会发生折叠。

Nowicka, Urszula; Hoffman, Morgan; Randles, Leah; Shi, Xiaoshan; Khavrutskii, Lyuba; Stefanisko, Karen; Tarasova, Nadya I; Darwin, K Heran; Walters, Kylie J

GTP-Dependent K-Ras Dimerization

GTP依赖性K-Ras二聚化

Muratcioglu, Serena; Chavan, Tanmay S; Freed, Benjamin C; Jang, Hyunbum; Khavrutskii, Lyuba; Freed, R Natasha; Dyba, Marzena A; Stefanisko, Karen; Tarasov, Sergey G; Gursoy, Attila; Keskin, Ozlem; Tarasova, Nadya I; Gaponenko, Vadim; Nussinov, Ruth

Protein purification-free method of binding affinity determination by microscale thermophoresis

无需纯化的微尺度热泳动法测定蛋白质结合亲和力

Lyuba Khavrutskii, Joanna Yeh, Olga Timofeeva, Sergey G Tarasov, Samuel Pritt, Karen Stefanisko, Nadya Tarasova

Retrotransposon suicide: formation of Ty1 circles and autointegration via a central DNA flap

逆转录转座子自杀:Ty1 环的形成和通过中心 DNA 瓣的自我整合

David J Garfinkel, Karen M Stefanisko, Katherine M Nyswaner, Sharon P Moore, Jangsuk Oh, Stephen H Hughes

Ty1 copy number dynamics in Saccharomyces

酿酒酵母中Ty1拷贝数动态

Garfinkel, David J; Nyswaner, Katherine M; Stefanisko, Karen M; Chang, Caroline; Moore, Sharon P