日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cyclization-blocked proguanil as a strategy to improve the antimalarial activity of atovaquone

环化阻断氯胍作为提高阿托伐醌抗疟活性的策略

Tina S Skinner-Adams #, Gillian M Fisher, Andrew G Riches, Oliver E Hutt, Karen E Jarvis, Tony Wilson, Mark von Itzstein, Pradeep Chopra, Yevgeniya Antonova-Koch, Stephan Meister, Elizabeth A Winzeler, Mary Clarke, David A Fidock, Jeremy N Burrows, John H Ryan #, Katherine T Andrews #

One-pot, multi-component synthesis and structure-activity relationships of peptoid-based histone deacetylase (HDAC) inhibitors targeting malaria parasites

针对疟原虫的基于肽的组蛋白去乙酰化酶 (HDAC) 抑制剂的一锅法多组分合成及构效关系

Daniela Diedrich, Katharina Stenzel, Eva Hesping, Yevgeniya Antonova-Koch, Tamirat Gebru, Sandra Duffy, Gillian Fisher, Andrea Schöler, Stephan Meister, Thomas Kurz, Vicky M Avery, Elizabeth A Winzeler, Jana Held, Katherine T Andrews, Finn K Hansen

Plasmodium falciparum Cyclic Amine Resistance Locus (PfCARL), a Resistance Mechanism for Two Distinct Compound Classes

恶性疟原虫环胺抗性位点 (PfCARL),两种不同化合物类别的抗性机制

Pamela A Magistrado, Victoria C Corey, Amanda K Lukens, Greg LaMonte, Erika Sasaki, Stephan Meister, Melanie Wree, Elizabeth Winzeler, Dyann F Wirth

Discovery of HDAC inhibitors with potent activity against multiple malaria parasite life cycle stages

发现对疟原虫生命周期多个阶段具有强效活性的 HDAC 抑制剂

Finn K Hansen, Subathdrage D M Sumanadasa, Katharina Stenzel, Sandra Duffy, Stephan Meister, Linda Marek, Rebekka Schmetter, Krystina Kuna, Alexandra Hamacher, Benjamin Mordmüller, Matthias U Kassack, Elizabeth A Winzeler, Vicky M Avery, Katherine T Andrews, Thomas Kurz

TMPRSS2-ERG -specific transcriptional modulation is associated with prostate cancer biomarkers and TGF-β signaling

TMPRSS2-ERG特异性转录调控与前列腺癌生物标志物和TGF-β信号通路相关

Brase, Jan C; Johannes, Marc; Mannsperger, Heiko; Fälth, Maria; Metzger, Jennifer; Kacprzyk, Lukasz A; Andrasiuk, Tatjana; Gade, Stephan; Meister, Michael; Sirma, Hüseyin; Sauter, Guido; Simon, Ronald; Schlomm, Thorsten; Beissbarth, Tim; Korf, Ulrike; Kuner, Ruprecht; Sültmann, Holger