日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Inhibitors of malaria parasite cyclic nucleotide phosphodiesterases block asexual blood-stage development and mosquito transmission.

疟原虫环核苷酸磷酸二酯酶抑制剂可阻断无性血液期发育和蚊子传播

Gomez-Gonzalez Paula-Josefina, Gupta Antima, Drought Laura G, Patel Avnish, Okombo John, van der Watt Mariëtte, Walker-Gray Ryan, Schindler Kyra A, Burkhard Anna Y, Yeo Tomas, Narwal Sunil K, Bloxham Talia S, Flueck Christian, Walker Eloise M, Rey Joshua A, Fairhurst Kate J, Reader Janette, Park Heekuk, Pollard Harry G, Stewart Lindsay B, Brandner-Garrod Luke, Kristan Mojca, Sterk Geert-Jan, van Nuland Youri M, Manko Emilia, van Schalkwyk Donelly A, Zheng Yang, Leurs Rob, Dechering Koen J, Aguiar Anna Caroline C, Guido Rafael V C, Pereira Dhelio B, Tumwebaze Patrick K, Nosbya Samuel L, Rosenthal Philip J, Cooper Roland A, Palmer Mike, Parkinson Tanya, Burrows Jeremy N, Uhlemann Anne-Catrin, Birkholtz Lyn-Marié, Small-Saunders Jennifer L, Duffy James, Fidock David A, Brown Alan, Gardner Mark, Baker David A

Adhesion of Crithidia fasciculata promotes a rapid change in developmental fate driven by cAMP signaling.

锥虫的粘附促进了由 cAMP 信号驱动的发育命运的快速改变

Denecke Shane, Malfara Madeline F, Hodges Kelly R, Holmes Nikki A, Williams Andre R, Gallagher-Teske Julia H, Pascarella Julia M, Daniels Abigail M, Sterk Geert Jan, Leurs Rob, Ruthel Gordon, Hoang Rachel, Povelones Megan L, Povelones Michael

Tetrahydrophthalazinone Inhibitor of Phosphodiesterase with In Vitro Activity against Intracellular Trypanosomatids

四氢酞嗪酮类磷酸二酯酶抑制剂,具有体外抗细胞内锥虫活性

de Araújo, Julianna Siciliano; Peres, Raiza Brandão; Bernardino da Silva, Patrícia; Batista, Marcos Meuser; Sterk, Geert Jan; Maes, Louis; Caljon, Guy; Leurs, Rob; de Koning, Harry P; Kalejaiye, Titilola D; Soeiro, Maria de Nazaré Correia

Structure Activity Relationship of N-Substituted Phenyldihydropyrazolones Against Trypanosoma cruzi Amastigotes

N-取代苯基二氢吡唑酮类化合物对克氏锥虫无鞭毛体的构效关系

Sijm, Maarten; Maes, Louis; de Esch, Iwan J P; Caljon, Guy; Sterk, Geert Jan; Leurs, Rob

Efficacy of Novel Pyrazolone Phosphodiesterase Inhibitors in Experimental Mouse Models of Trypanosoma cruzi

新型吡唑酮磷酸二酯酶抑制剂在克氏锥虫实验小鼠模型中的疗效

de Araújo, Julianna Siciliano; França da Silva, Cristiane; Batista, Denise da Gama Jaén; Nefertiti, Aline; Fiuza, Ludmila Ferreira de Almeida; Fonseca-Berzal, Cristina Rosa; Bernardino da Silva, Patrícia; Batista, Marcos Meuser; Sijm, Maarten; Kalejaiye, Titilola D; de Koning, Harry P; Maes, Louis; Sterk, Geert Jan; Leurs, Rob; Soeiro, Maria de Nazaré Correia

Structure-Activity Relationship of Phenylpyrazolones against Trypanosoma cruzi

苯基吡唑酮类化合物对克氏锥虫的构效关系

Sijm, Maarten; Sterk, Geert Jan; Caljon, Guy; Maes, Louis; de Esch, Iwan J P; Leurs, Rob

Identification of Phenylpyrazolone Dimers as a New Class of Anti-Trypanosoma cruzi Agents

苯基吡唑酮二聚体作为一类新型抗克氏锥虫药物的鉴定

Sijm, Maarten; Siciliano de Araújo, Julianna; Ramos Llorca, Alba; Orrling, Kristina; Stiny, Lydia; Matheeussen, An; Maes, Louis; de Esch, Iwan J P; de Nazaré Correia Soeiro, Maria; Sterk, Geert Jan; Leurs, Rob