日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Direct and selective pharmacological disruption of the YAP-TEAD interface by IAG933 inhibits Hippo-dependent and RAS-MAPK-altered cancers

IAG933通过直接和选择性地药理学手段破坏YAP-TEAD界面,从而抑制Hippo依赖性和RAS-MAPK改变的癌症。

Emilie A Chapeau ,Laurent Sansregret ,Giorgio G Galli ,Patrick Chène ,Markus Wartmann ,Thanos P Mourikis ,Patricia Jaaks ,Sabrina Baltschukat ,Ines A M Barbosa ,Daniel Bauer ,Saskia M Brachmann ,Clara Delaunay ,Claire Estadieu ,Jason E Faris ,Pascal Furet ,Stefanie Harlfinger ,Andreas Hueber ,Eloísa Jiménez Núñez ,David P Kodack ,Emeline Mandon ,Typhaine Martin ,Yannick Mesrouze ,Vincent Romanet ,Clemens Scheufler ,Holger Sellner ,Christelle Stamm ,Dario Sterker ,Luca Tordella ,Francesco Hofmann ,Nicolas Soldermann ,Tobias Schmelzle

Still an Unsolved Question: The Place of Cranial Magnetic Resonance Imaging in Acute Acquired Concomitant Esotropia

仍未解决的问题:颅脑磁共振成像在急性获得性伴随性内斜视中的地位

Mittendorf, Luisa; Bernhard, Matthias K; Sterker, Ina; Kiess, Wieland; Gburek-Augustat, Janina; Merkenschlager, Andreas

Transient Inhibition of the JAK/STAT Pathway Prevents B-ALL Development in Genetically Predisposed Mice

瞬时抑制JAK/STAT通路可预防遗传易感小鼠发生B细胞急性淋巴细胞白血病(B-ALL)

Ana Casado-García # ,Marta Isidro-Hernández # ,Ninad Oak # ,Andrea Mayado ,Christine Mann-Ran ,Javier Raboso-Gallego ,Silvia Alemán-Arteaga ,Alexandra Buhles ,Dario Sterker ,Elena G Sánchez ,Jorge Martínez-Cano ,Oscar Blanco ,Alberto Orfao ,Diego Alonso-López ,Javier De Las Rivas ,Susana Riesco ,Pablo Prieto-Matos ,África González-Murillo ,Francisco Javier García Criado ,María Begoña García Cenador ,Thomas Radimerski ,Manuel Ramírez-Orellana ,César Cobaleda ,Jun J Yang ,Carolina Vicente-Dueñas # ,Andreas Weiss # ,Kim E Nichols # ,Isidro Sánchez-García #

Consideration of specific key points improves outcome of decompression treatment in patients with endocrine orbitopathy: pre-/post-OP comparison and biomechanical simulation

考虑特定关键点可改善内分泌性眼眶病患者减压治疗的效果:术前/术后比较和生物力学模拟

Krause, Matthias; Neuhaus, Michael-Tobias; Sterker, Ina; Bartella, Alexander K; Schönfeld, Annika; Lethaus, Bernd; Zimmerer, Rüdiger; Gladilin, Evgeny

A Microphysiological Cell-Culturing System for Pharmacokinetic Drug Exposure and High-Resolution Imaging of Arrays of 3D Microtissues

用于药代动力学药物暴露和 3D 微组织阵列高分辨率成像的微生理细胞培养系统

Christian Lohasz, Jacqueline Loretan, Dario Sterker, Ekkehard Görlach, Kasper Renggli, Paul Argast, Olivier Frey, Marion Wiesmann, Markus Wartmann, Martin Rausch, Andreas Hierlemann

Eyes wide shut: necessity and effect of adjunctive procedures after decompression surgery in patients with endocrine orbitopathy

睁大眼睛:内分泌性眼眶病患者减压手术后辅助治疗的必要性和效果

Krause, Matthias; Kamal, Mohammad; Halama, Dirk; Hierl, Thomas; Sterker, Ina; Zimmerer, Rüdiger; Lethaus, Bernd; Bartella, Alexander K

Neuro-Ophthalmic Literature Review

神经眼科文献综述

Rauscher, Franziska G; Lange, Heike; Yahiaoui-Doktor, Maryam; Tegetmeyer, Helmut; Sterker, Ina; Hinz, Andreas; Wahl, Siegfried; Wiedemann, Peter; Ohlendorf, Arne; Blendowske, Ralf; Bellows, David; Chan, Noel; Chen, John; Cheng, Hui-Chen; Jindahra, Panitha; Kaiyrzhanov, Rauan; MacIntosh, Peter; Vaphiades, Michael; Weber, Konrad P; Wong, Sui

Dose and Schedule Determine Distinct Molecular Mechanisms Underlying the Efficacy of the p53-MDM2 Inhibitor HDM201

剂量和给药方案决定了 p53-MDM2 抑制剂 HDM201 疗效背后的不同分子机制

Sébastien Jeay #, Stéphane Ferretti #, Philipp Holzer #, Jeanette Fuchs, Emilie A Chapeau, Markus Wartmann, Dario Sterker, Vincent Romanet, Masato Murakami, Grainne Kerr, Eric Y Durand, Swann Gaulis, Marta Cortes-Cros, Stephan Ruetz, Therese-Marie Stachyra, Joerg Kallen, Pascal Furet, Jens Würthner,

JAK1/2 and Pan-deacetylase inhibitor combination therapy yields improved efficacy in preclinical mouse models of JAK2V617F-driven disease

JAK1/2 与泛脱乙酰酶抑制剂联合治疗在 JAK2V617F 驱动疾病的临床前小鼠模型中疗效提高

Emeline Evrot, Nicolas Ebel, Vincent Romanet, Claudia Roelli, Rita Andraos, Zhiyan Qian, Arno Dölemeyer, Ernesta Dammassa, Dario Sterker, Robert Cozens, Francesco Hofmann, Masato Murakami, Fabienne Baffert, Thomas Radimerski

K-RAS mutant pancreatic tumors show higher sensitivity to MEK than to PI3K inhibition in vivo

K-RAS 突变型胰腺肿瘤对 MEK 的敏感性高于对 PI3K 抑制的敏感性

Irmgard Hofmann, Andreas Weiss, Gaelle Elain, Maria Schwaederle, Dario Sterker, Vincent Romanet, Tobias Schmelzle, Albert Lai, Saskia M Brachmann, Mohamed Bentires-Alj, Thomas M Roberts, William R Sellers, Francesco Hofmann, Sauveur-Michel Maira