Torin 2 Derivative, NCATS-SM3710, Has Potent Multistage Antimalarial Activity through Inhibition of P. falciparum Phosphatidylinositol 4-Kinase (Pf PI4KIIIβ)
Torin 2 衍生物 NCATS-SM3710 通过抑制恶性疟原虫磷脂酰肌醇 4-激酶 (Pf PI4KIIIβ) 发挥强效的多阶段抗疟活性
期刊:ACS Pharmacology and Translational Science
影响因子:3.7
doi:10.1021/acsptsci.0c00078
Krishnan, Karthik; Ziniel, Peter; Li, Hao; Huang, Xiuli; Hupalo, Daniel; Gombakomba, Nita; Guerrero, Sandra Mendoza; Dotrang, Thoai; Lu, Xiao; Caridha, Diana; Sternberg, Anna R; Hughes, Emma; Sun, Wei; Bargieri, Daniel Y; Roepe, Paul D; Sciotti, Richard J; Wilkerson, Matthew D; Dalgard, Clifton L; Tawa, Gregory J; Wang, Amy Q; Xu, Xin; Zheng, Wei; Sanderson, Philip E; Huang, Wenwei; Williamson, Kim C