日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A coronavirus assembly inhibitor that targets the viral membrane protein.

一种针对病毒膜蛋白的冠状病毒组装抑制剂

Laporte Manon, Jochmans Dirk, Bardiot Dorothée, Desmarets Lowiese, Debski-Antoniak Oliver J, Mizzon Giulia, Abdelnabi Rana, Leyssen Pieter, Chiu Winston, Zhang Zhikuan, Nomura Norimichi, Boland Sandro, Ohto Umeharu, Stahl Yannick, Wuyts Jurgen, De Jonghe Steven, Stevaert Annelies, van Hemert Martijn J, Bontes Brenda W, Wanningen Patrick, Groenewold G J Mirjam, Zegar Aneta, Owczarek Katarzyna, Joshi Sanjata, Koukni Mohamed, Arzel Philippe, Klaassen Hugo, Vanherck Jean-Christophe, Vandecaetsbeek Ilse, Cremers Niels, Donckers Kim, Francken Thibault, Van Buyten Tina, Rymenants Jasper, Schepers Joost, Pyrc Krzysztof, Hilgenfeld Rolf, Dubuisson Jean, Bosch Berend-Jan, Van Kuppeveld Frank, Eydoux Cecilia, Decroly Etienne, Canard Bruno, Naesens Lieve, Weynand Birgit, Snijder Eric J, Belouzard Sandrine, Shimizu Toshiyuki, Bartenschlager Ralf, Hurdiss Daniel L, Marchand Arnaud, Chaltin Patrick, Neyts Johan

Trypstatin as a Novel TMPRSS2 Inhibitor with Broad-Spectrum Efficacy against Corona and Influenza Viruses.

胰蛋白酶抑制剂作为一种新型TMPRSS2抑制剂,对冠状病毒和流感病毒具有广谱疗效

Lawrenz Jan, Wettstein Lukas, Rodríguez Alfonso Armando, Nchioua Rayhane, von Maltitz Pascal, Albers Dan Pascal Jean, Zech Fabian, Vandeput Julie, Naesens Lieve, Fois Giorgio, Neubauer Veronika, Preising Nico, Schmierer Emilia, Almeida-Hernandez Yasser, Petersen Moritz, Ständker Ludger, Wiese Sebastian, Braubach Peter, Frick Manfred, Barth Eberhard, Sauter Daniel, Kirchhoff Frank, Sanchez-Garcia Elsa, Stevaert Annelies, Münch Jan

N-[(Thiophen-3-yl)methyl]benzamides as Fusion Inhibitors of Influenza Virus Targeting H1 and H5 Hemagglutinins

N-[(噻吩-3-基)甲基]苯甲酰胺类化合物作为流感病毒H1和H5血凝素融合抑制剂

Silke Rimaux,Aitor Valdivia,Juan Martín-López,Valeria Francesconi,Celia Escriche,Cato Mestdagh,Ria Van Berwaer,Lieselotte Schurmans,Kaat Verleye,Samuel Noppen,Óscar Lozano,Annelies Stevaert,F Javier Luque,Lieve Naesens,Santiago Vázquez

A guanidine-based coronavirus replication inhibitor which targets the nsp15 endoribonuclease and selects for interferon-susceptible mutant viruses

一种基于胍的冠状病毒复制抑制剂,靶向nsp15核糖核酸内切酶,并筛选出对干扰素敏感的突变病毒。

Van Loy, Benjamin; Pujol, Eugènia; Kamata, Kenichi; Lee, Xiao Yin; Bakirtzoglou, Nikolai; Van Berwaer, Ria; Vandeput, Julie; Mestdagh, Cato; Persoons, Leentje; De Wijngaert, Brent; Goovaerts, Quinten; Noppen, Sam; Jacquemyn, Maarten; Ahmadzadeh, Kourosh; Bernaerts, Eline; Martín-López, Juan; Escriche, Celia; Vanmechelen, Bert; Krasniqi, Besir; Singh, Abhimanyu K; Daelemans, Dirk; Maes, Piet; Matthys, Patrick; Dehaen, Wim; Rozenski, Jef; Das, Kalyan; Voet, Arnout; Vázquez, Santiago; Naesens, Lieve; Stevaert, Annelies

Profiling Bacteria in the Lungs of Patients with Severe Influenza Versus COVID-19 with or without Aspergillosis

对重症流感患者与伴或不伴曲霉病的 COVID-19 患者肺部细菌进行分析

Feys, Simon; Cardinali-Benigni, Martina; Lauwers, Hanne Moon; Jacobs, Cato; Stevaert, Annelies; Gonçalves, Samuel M; Cunha, Cristina; Debaveye, Yves; Hermans, Greet; Heylen, Jannes; Humblet-Baron, Stephanie; Lagrou, Katrien; Maessen, Lenn; Meersseman, Philippe; Peetermans, Marijke; Redondo-Rios, Alvaro; Seldeslachts, Laura; Starick, Marick R; Thevissen, Karin; Vande Velde, Greetje; Vandenbriele, Christophe; Vanderbeke, Lore; Wilmer, Alexander; Naesens, Lieve; van de Veerdonk, Frank L; Van Weyenbergh, Johan; Gabaldón, Toni; Wauters, Joost; Carvalho, Agostinho

Cellular electrical impedance to profile SARS-CoV-2 fusion inhibitors and to assess the fusogenic potential of spike mutants

利用细胞电阻抗分析SARS-CoV-2融合抑制剂并评估刺突蛋白突变体的融合潜力

Emiel Vanhulle ,Jordi Doijen ,Joren Stroobants ,Becky Provinciael ,Sam Noppen ,Dominique Schols ,Annelies Stevaert ,Kurt Vermeire

PRO-2000 exhibits SARS-CoV-2 antiviral activity by interfering with spike-heparin binding

PRO-2000 通过干扰尖峰肝素结合表现出 SARS-CoV-2 抗病毒活性

Evelien Vanderlinden, Arnaud Boonen, Sam Noppen, Geert Schoofs, Maya Imbrechts, Nick Geukens, Robert Snoeck, Annelies Stevaert, Lieve Naesens, Graciela Andrei, Dominique Schols

Novel Polymyxin-Inspired Peptidomimetics Targeting the SARS-CoV-2 Spike:hACE2 Interface

受多粘菌素启发的新型肽模拟物,针对 SARS-CoV-2 Spike:hACE2 界面

Kelly Bugatti, Andrea Sartori, Lucia Battistini, Crescenzo Coppa, Emiel Vanhulle, Sam Noppen, Becky Provinciael, Lieve Naesens, Annelies Stevaert, Alessandro Contini, Kurt Vermeire, Franca Zanardi

Functional Analysis of Human and Feline Coronavirus Cross-Reactive Antibodies Directed Against the SARS-CoV-2 Fusion Peptide

针对 SARS-CoV-2 融合肽的人与猫冠状病毒交叉反应抗体的功能分析

Nathalie Vanderheijden, Annelies Stevaert, Jiexiong Xie, Xiaolei Ren, Cyril Barbezange, Sam Noppen, Isabelle Desombere, Bruno Verhasselt, Peter Geldhof, Nick Vereecke, Veerle Stroobants, Dayoung Oh, Merijn Vanhee, Lieve M J Naesens, Hans J Nauwynck

Impact of SARS-CoV-2 Spike Mutations on Its Activation by TMPRSS2 and the Alternative TMPRSS13 Protease

SARS-CoV-2 刺突突变对 TMPRSS2 和替代 TMPRSS13 蛋白酶激活的影响

Annelies Stevaert, Ria Van Berwaer, Cato Mestdagh, Julie Vandeput, Els Vanstreels, Valerie Raeymaekers, Manon Laporte, Lieve Naesens