Alkylsulfanyl-1,2,4-triazoles, a new class of allosteric valosine containing protein inhibitors. Synthesis and structure-activity relationships
烷基硫烷基-1,2,4-三唑,一类新型变构缬氨酸蛋白抑制剂。合成和结构-活性关系
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm3013213
Paolo Polucci, Paola Magnaghi, Mauro Angiolini, Daniela Asa, Nilla Avanzi, Alessandra Badari, Jay Bertrand, Elena Casale, Silvia Cauteruccio, Alessandra Cirla, Liviana Cozzi, Arturo Galvani, Peter K Jackson, Yichin Liu, Steven Magnuson, Beatrice Malgesini, Stefano Nuvoloni, Christian Orrenius, Feder