日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The multi-CDK inhibitor dinaciclib reverses bromo- and extra-terminal domain (BET) inhibitor resistance in acute myeloid leukemia via inhibition of Wnt/β-catenin signaling

多 CDK 抑制剂 dinaciclib 通过抑制 Wnt/β-catenin 信号传导逆转急性髓系白血病中溴和额外末端结构域 (BET) 抑制剂的耐药性

Alexander R Marr, Madeline Halpin, Dominique L Corbin, Yerdanos Asemelash, Steven Sher, Britten K Gordon, Ethan C Whipp, Shaneice Mitchell, Bonnie K Harrington, Shelley Orwick, Samon Benrashid, Virginia M Goettl, Vedat Yildiz, Andrew D Mitchell, Olivia Cahn, Alice S Mims, Karilyn T M Larkin, Meixao

Dysregulation of PRMT5 in chronic lymphocytic leukemia promotes progression with high risk of Richter's transformation

慢性淋巴细胞白血病中 PRMT5 失调会促进病情进展,且存在 Richter 转化的高风险

Zachary A Hing #, Janek S Walker #, Ethan C Whipp #, Lindsey Brinton, Matthew Cannon, Pu Zhang, Steven Sher, Casey B Cempre, Fiona Brown, Porsha L Smith, Claudio Agostinelli, Stefano A Pileri, Jordan N Skinner, Katie Williams, Hannah Phillips, Jami Shaffer, Larry P Beaver, Alexander Pan, Kyle Shin, 

VIP152 is a selective CDK9 inhibitor with pre-clinical in vitro and in vivo efficacy in chronic lymphocytic leukemia

VIP152 是一种选择性 CDK9 抑制剂,在慢性淋巴细胞白血病中具有临床前体外和体内疗效

Steven Sher, Ethan Whipp, Janek Walker, Pu Zhang, Larry Beaver, Katie Williams, Shelley Orwick, Janani Ravikrishnan, Brandi Walker, Elizabeth Perry, Charles Gregory, Matthew Purcell, Alexander Pan, Pearlly Yan, Lapo Alinari, Amy J Johnson, Melanie M Frigault, Joy M Greer, Ahmed Hamdy, Raquel Izumi, 

Microenvironmental control of hematopoietic stem cell fate via CXCL8 and protein kinase C

通过 CXCL8 和蛋白激酶 C 微环境控制造血干细胞命运

Vera Binder, Wantong Li, Muhammad Faisal, Konur Oyman, Donn L Calkins, Jami Shaffer, Emily M Teets, Steven Sher, Andrew Magnotte, Alex Belardo, William Deruelle, T Charles Gregory, Shelley Orwick, Elliott J Hagedorn, Julie R Perlin, Serine Avagyan, Asher Lichtig, Francesca Barrett, Michelle Ammerman

DJ-1 Molecular Chaperone Activity Depresses Tau Aggregation Propensity through Interaction with Monomers

DJ-1 分子伴侣活性通过与单体相互作用抑制 Tau 聚集倾向

Daniela Jimenez-Harrison, Carol J Huseby, Claire N Hoffman, Steven Sher, Dalton Snyder, Brayden Seal, Chunhua Yuan, Hongjun Fu, Vicki Wysocki, Flaviano Giorgini, Jeff Kuret

Targeting OXPHOS de novo purine synthesis as the nexus of FLT3 inhibitor-mediated synergistic antileukemic actions

以 OXPHOS 从头嘌呤合成为目标,作为 FLT3 抑制剂介导的协同抗白血病作用的纽带

Pu Zhang, Lindsey T Brinton, Mehdi Gharghabi, Steven Sher, Katie Williams, Matthew Cannon, Janek S Walker, Daniel Canfield, Larry Beaver, Casey B Cempre, Hannah Phillips, Xuyong Chen, Pearlly Yan, Amy Lehman, Peggy Scherle, Min Wang, Kris Vaddi, Robert Baiocchi, Ruoning Wang, Deepa Sampath, Lapo Ali

Rare t(X;14)(q28;q32) translocation reveals link between MTCP1 and chronic lymphocytic leukemia

罕见的t(X;14)(q28;q32)易位揭示了MTCP1与慢性淋巴细胞白血病之间的联系

Janek S Walker # ,Zachary A Hing # ,Steven Sher ,James Cronin ,Katie Williams ,Bonnie Harrington ,Jordan N Skinner ,Casey B Cempre ,Charles T Gregory ,Alexander Pan ,Max Yano ,Larry P Beaver ,Brandi R Walker ,Jadwiga M Labanowska ,Nyla A Heerema ,Krzysztof Mrózek ,Jennifer A Woyach ,Amy S Ruppert ,Amy Lehman ,Hatice Gulcin Ozer ,Vincenzo Coppola ,Pearlly Yan ,John C Byrd ,James S Blachly ,Rosa Lapalombella

Genomic analysis of cellular hierarchy in acute myeloid leukemia using ultrasensitive LC-FACSeq

利用超灵敏LC-FACSeq技术对急性髓系白血病细胞层级进行基因组分析

Caner Saygin ,Eileen Hu ,Pu Zhang ,Steven Sher ,Arletta Lozanski ,Tzyy-Jye Doong ,Deedra Nicolet ,Shelley Orwick ,Jadwiga Labanowska ,Jordan N Skinner ,Casey Cempre ,Tierney Kauffman ,Virginia M Goettl ,Nyla A Heerema ,Lynne Abruzzo ,Cecelia Miller ,Rosa Lapalombella ,Gregory Behbehani ,Alice S Mims ,Karilyn Larkin ,Nicole Grieselhuber ,Alison Walker ,Bhavana Bhatnagar ,Clara D Bloomfield ,John C Byrd ,Gerard Lozanski # ,James S Blachly #

Targeting DNA Damage Repair Functions of Two Histone Deacetylases, HDAC8 and SIRT6, Sensitizes Acute Myeloid Leukemia to NAMPT Inhibition

靶向两种组蛋白去乙酰化酶 HDAC8 和 SIRT6 的 DNA 损伤修复功能,增强急性髓系白血病对 NAMPT 抑制的敏感性

Pu Zhang, Lindsey T Brinton, Katie Williams, Steven Sher, Shelley Orwick, Lai Tzung-Huei, Alice S Mims, Christopher C Coss, Samuel K Kulp, Youssef Youssef, Wing Keung Chan, Shaneice Mitchell, Allison Mustonen, Matthew Cannon, Hannah Phillips, Amy M Lehman, Tierney Kauffman, Larry Beaver, Daniel Canf

Cotargeting of XPO1 Enhances the Antileukemic Activity of Midostaurin and Gilteritinib in Acute Myeloid Leukemia

XPO1 的共靶向作用增强了米哚妥林和吉特替尼在急性髓系白血病中的抗白血病活性

Lindsey T Brinton, Steven Sher, Katie Williams, Daniel Canfield, Shelley Orwick, Ronni Wasmuth, Casey Cempre, Jordan Skinner, Amy Lehman, James S Blachly, John C Byrd, Rosa Lapalombella