Discovery of MD-265: A Potent MDM2 Degrader That Achieves Complete Tumor Regression and Improves Long-Term Survival of Mice with Leukemia
MD-265 的发现:一种强效的 MDM2 降解剂,可实现肿瘤完全消退并提高白血病小鼠的长期生存率
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c01818
Aguilar, Angelo; Yang, Jiuling; Li, Yangbing; McEachern, Donna; Huang, Liyue; Razzouk, Stevenchoukry; Wang, Shaomeng