日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural Determinants of Indole-2-carboxamides: Identification of Lead Acetamides with Pan Antimycobacterial Activity

吲哚-2-甲酰胺的结构决定因素:鉴定具有泛抗分枝杆菌活性的先导乙酰胺类化合物

Bhattarai, Pankaj; Hegde, Pooja; Li, Wei; Prathipati, Pavan Kumar; Stevens, Casey M; Yang, Lixinhao; Zhou, Hinman; Pandya, Amit; Cunningham, Katie; Grissom, Jenny; Roman Sotelo, Mariaelena; Sowards, Melanie; Calisto, Lilian; Destache, Christopher J; Rocha-Sanchez, Sonia; Gumbart, James C; Zgurskaya, Helen I; Jackson, Mary; North, E Jeffrey

Microbiological profile, preclinical pharmacokinetics and efficacy of CRS0393, a novel antimycobacterial agent targeting MmpL3.

CRS0393 是一种新型抗分枝杆菌药物,靶向 MmpL3,其微生物学特征、临床前药代动力学和疗效研究

Ochsner Urs A, De Groote Mary A, Jarvis Thale C, Liu Hang, Youmans Tessa, Hoang Teresa, Ribble Wendy, Day Joshua, Li Wei, Pearce Camron, Walz Amanda, Panthi Chandra M, Rimal Binayak, Stevens Casey M, Zgurskaya Helen I, Jackson Mary, Ordway Diane, Gonzalez-Juarrero Mercedes, Sun Xicheng, Lamichhane Gyanu, Mason Clifford

Transporters Involved in the Biogenesis and Functionalization of the Mycobacterial Cell Envelope

参与分枝杆菌细胞包膜生物合成和功能的转运蛋白

Jackson, Mary; Stevens, Casey M; Zhang, Lei; Zgurskaya, Helen I; Niederweis, Michael