日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction to "Next-Generation MDMA Analogue SDMA: Pharmacological and Metabolic Insights"

对“下一代 MDMA 类似物 SDMA:药理学和代谢学见解”的更正

Kastner, Nina; Nadal-Gratacós, Núria; Hemmer, Selina; Alves da Silva, Leticia; McKee, John L; Hell, Tamara; Cicalese, Giulia; Holy, Marion; Kooti, Fatemeh; Jäntsch, Kathrin; Baron, Ricarda; Shacham, Naomi; Cuccurazzu, Bruna; Halberstadt, Adam L; McCorvy, John D; Stockner, Thomas; Meyer, Markus R; López-Arnau, Raúl; Grill, Matthias; Sitte, Harald H

Revealing the location and dynamics of a concealed binding site in the dopamine transporter.

揭示多巴胺转运蛋白中隐藏结合位点的位置和动态

Zhu Rong, Sandtner Walter, Stockner Thomas, Heilinger Alexander, Holy Marion, Kudlacek Oliver, Wildling Linda, Saha Kusumika, Fröhlich Anna Sophie, Bindl Michael, Tziortzouda Paraskevi, Haider Anna, Gobl Julia, Suh Saanfor Hubert, Khan Jawad Akbar, Bicher Julia, Kastner Nina, Ebner Andreas, Gruber Hermann J, Freissmuth Michael, Newman Amy Hauck, Sitte Harald H, Hinterdorfer Peter

Health risks of cocaine adulteration: local anesthetics as modulators of monoamine and organic cation transporters

可卡因掺杂的健康风险:局部麻醉剂作为单胺和有机阳离子转运体的调节剂

Kudlacek, Oliver; Senning, Niklas; Karden, Alexandra; Ludwig, Iina; Bicher, Julia; Kooti, Fatemeh; Holy, Marion; Stockner, Thomas; Luf, Anton; Sitte, Harald H

Next-Generation MDMA Analogue SDMA: Pharmacological and Metabolic Insights

下一代MDMA类似物SDMA:药理学和代谢学见解

Kastner, Nina; Nadal-Gratacós, Núria; Hemmer, Selina; Alves da Silva, Leticia; McKee, John L; Hell, Tamara; Cicalese, Giulia; Holy, Marion; Kooti, Fatemeh; Jäntsch, Kathrin; Baron, Ricarda; Shacham, Naomi; Cuccurazzu, Bruna; Halberstadt, Adam L; McCorvy, John D; Stockner, Thomas; Meyer, Markus R; López-Arnau, Raúl; Grill, Matthias; Sitte, Harald H

Substrate-specific effects point to the important role of Y361 as part of the YER motif in closing the binding pocket of OCT1

底物特异性效应表明,Y361作为YER基序的一部分,在OCT1结合口袋的闭合中发挥着重要作用。

Römer, Sarah; Lazzarin, Erika; Neumann, Anna; Lindemann, Erik; Meyer-Tönnies, Marleen J; Stockner, Thomas; Tzvetkov, Mladen V

Prolintane analogs as hybrid monoamine transporter ligands: Structural determinants and species differences

脯氨酰胺类似物作为杂合单胺转运体配体:结构决定因素和物种差异

Kastner, Nina; Islam, Mohammad N; Dybek, Michael; Roth, Evelyn; Heisinger, Simon; Holy, Marion; Jäntsch, Kathrin; Walther, Donna; Stockner, Thomas; Baumann, Michael H; Brandt, Simon D; Wallach, Jason; Sitte, Harald H; Kudlacek, Oliver

PIP(2) modulates TRPC3 activity via TRP helix and S4-S5 linker.

PIP(2) 通过 TRP 螺旋和 S4-S5 连接子调节 TRPC3 活性

Clarke Amy, Skerjanz Julia, Gsell Mathias A F, Wiedner Patrick, Erkan-Candag Hazel, Groschner Klaus, Stockner Thomas, Tiapko Oleksandra

Unveiling the crucial role of betaine: modulation of GABA homeostasis via SLC6A1 transporter (GAT1)

揭示甜菜碱的关键作用:通过 SLC6A1 转运蛋白 (GAT1) 调节 GABA 稳态

Bhatt, Manan; Lazzarin, Erika; Alberto-Silva, Ana Sofia; Domingo, Guido; Zerlotti, Rocco; Gradisch, Ralph; Bazzone, Andre; Sitte, Harald H; Stockner, Thomas; Bossi, Elena

De novo variants in GABRA4 are associated with a neurological phenotype including developmental delay, behavioral abnormalities and epilepsy

GABRA4基因的新生变异与神经系统表型相关,包括发育迟缓、行为异常和癫痫。

Sajan, Samin A; Gradisch, Ralph; Vogel, Florian D; Coffey, Alison J; Salyakina, Daria; Soler, Diana; Jayakar, Parul; Jayakar, Anuj; Bianconi, Simona E; Cooper, Annina H; Liu, Shuxi; William, Nancy; Benkel-Herrenbrück, Ira; Maiwald, Robert; Heller, Corina; Biskup, Saskia; Leiz, Steffen; Westphal, Dominik S; Wagner, Matias; Clarke, Amy; Stockner, Thomas; Ernst, Margot; Kesari, Akanchha; Krenn, Martin

Bioisosteric analogs of MDMA: Improving the pharmacological profile?

MDMA的生物等排体类似物:能否改善其药理特性?

Alberto-Silva Ana Sofia, Hemmer Selina, Bock Hailey A, da Silva Leticia Alves, Scott Kenneth R, Kastner Nina, Bhatt Manan, Niello Marco, Jäntsch Kathrin, Kudlacek Oliver, Bossi Elena, Stockner Thomas, Meyer Markus R, McCorvy John D, Brandt Simon D, Kavanagh Pierce, Sitte Harald H