日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction to "Sebetralstat (KVD900): A Potent and Selective Small Molecule Plasma Kallikrein Inhibitor Featuring a Novel P1 Group as a Potential Oral On-Demand Treatment for Hereditary Angioedema"

对“Sebetralstat (KVD900):一种具有新型 P1 基团的强效选择性小分子血浆激肽释放酶抑制剂,有望成为遗传性血管性水肿的按需口服治疗药物”一文的更正

Davie, Rebecca L; Edwards, Hannah J; Evans, D Michael; Hodgson, Simon T; Stocks, Michael J; Smith, Alun J; Rushbrooke, Louise J; Pethen, Stephen J; Roe, Michael B; Clark, David E; McEwan, Paul A; Hampton, Sally L

Drug-like Antagonists of P2Y Receptor Subtypes: An Update

P2Y受体亚型的类药物拮抗剂:最新进展

Puthanveedu, Mahesh; Knight, Rebecca; Stocks, Michael J

Design, Synthesis, and Evaluation of Selective Ubiquitin-Specific Protease 11 (USP11) Inhibitors

选择性泛素特异性蛋白酶11 (USP11) 抑制剂的设计、合成和评价

Hassan, Mostafa A; Dekker, Lodewijk V; Stocks, Michael J; Dreveny, Ingrid

The Characterization of a Gonococcal HicAB Toxin-Antitoxin System Capable of Causing Bacteriostatic Growth Arrest

淋球菌 HicAB 毒素-抗毒素系统能够引起抑菌生长停滞的特性分析

Bagabas, Salwa S; Trujillo-Mendoza, Jorge; Stocks, Michael J; Turner, David P J; Oldfield, Neil J

Discovery of Highly Potent BET Inhibitors based on a Tractable Tricyclic Scaffold

基于易于合成的三环骨架发现高效BET抑制剂

Zaidi, Jaffer M; Comeo, Eleonora; Baxter, Andrew; Preston, Alex G S; Chan, Weng C; Stocks, Michael J

Design, Synthesis, and Evaluation of a New Chemotype Fluorescent Ligand for the P2Y(2) Receptor

P2Y(2)受体新型化学型荧光配体的设计、合成与评价

Knight, Rebecca; Kilpatrick, Laura E; Hill, Stephen J; Stocks, Michael J

Discovery of α-Amidobenzylboronates as Highly Potent Covalent Inhibitors of Plasma Kallikrein

发现α-氨基苄基硼酸酯是血浆激肽释放酶的高效共价抑制剂

Allison, Matthew; Davie, Rebecca L; Mogg, Adrian J; Hampton, Sally L; Emsley, Jonas; Stocks, Michael J

Small Molecule Fluorescent Ligands for the Atypical Chemokine Receptor 3 (ACKR3)

非典型趋化因子受体 3 (ACKR3) 的小分子荧光配体

Dekkers, Sebastian; Comez, Dehan; Karsai, Noemi; Arimont-Segura, Marta; Canals, Meritxell; Caspar, Birgit; de Graaf, Chris; Kilpatrick, Laura E; Leurs, Rob; Kellam, Barrie; Hill, Stephen J; Briddon, Stephen J; Stocks, Michael J

Theoretical Study on the Biosynthesis of the Mandapamates: Mechanistic Insights Using Density Functional Theory

曼达帕酯生物合成的理论研究:基于密度泛函理论的机制解析

Wang, Di; Pattenden, Gerald; Fow, Kam Loon; Stocks, Michael J; Hirst, Jonathan D; Tang, Bencan

Assessing Lymphatic Uptake of Lipids Using Magnetic Resonance Imaging: A Feasibility Study in Healthy Human Volunteers with Potential Application for Tracking Lymph Node Delivery of Drugs and Formulation Excipients

利用磁共振成像评估脂质的淋巴吸收:一项在健康人体志愿者中进行的可行性研究,具有追踪药物和制剂辅料淋巴结递送的潜在应用价值

Jewell, Adelaide; Williams, Hannah; Hoad, Caroline L; Gellert, Paul R; Ashford, Marianne B; Butler, James; Stolnik, Snow; Scurr, David; Stocks, Michael J; Marciani, Luca; Gowland, Penny A; Gershkovich, Pavel