日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Glutathione transport: a new role for PfCRT in chloroquine resistance

谷胱甘肽转运:PfCRT在氯喹耐药性中的新作用

Patzewitz, Eva-Maria; Salcedo-Sora, J Enrique; Wong, Eleanor H; Sethia, Sonal; Stocks, Paul A; Maughan, Spencer C; Murray, James A H; Krishna, Sanjeev; Bray, Patrick G; Ward, Stephen A; Müller, Sylke

Generation of quinolone antimalarials targeting the Plasmodium falciparum mitochondrial respiratory chain for the treatment and prophylaxis of malaria.

开发针对恶性疟原虫线粒体呼吸链的喹诺酮类抗疟药,用于治疗和预防疟疾

Biagini Giancarlo A, Fisher Nicholas, Shone Alison E, Mubaraki Murad A, Srivastava Abhishek, Hill Alisdair, Antoine Thomas, Warman Ashley J, Davies Jill, Pidathala Chandrakala, Amewu Richard K, Leung Suet C, Sharma Raman, Gibbons Peter, Hong David W, Pacorel Bénédicte, Lawrenson Alexandre S, Charoensutthivarakul Sitthivut, Taylor Lee, Berger Olivier, Mbekeani Alison, Stocks Paul A, Nixon Gemma L, Chadwick James, Hemingway Janet, Delves Michael J, Sinden Robert E, Zeeman Anne-Marie, Kocken Clemens H M, Berry Neil G, O'Neill Paul M, Ward Stephen A

Identification, design and biological evaluation of heterocyclic quinolones targeting Plasmodium falciparum type II NADH:quinone oxidoreductase (PfNDH2)

针对恶性疟原虫 II 型 NADH:醌氧化还原酶 (PfNDH2) 的杂环喹诺酮的鉴定、设计和生物学评价

Leung, Suet C; Gibbons, Peter; Amewu, Richard; Nixon, Gemma L; Pidathala, Chandrakala; Hong, W David; Pacorel, Bénédicte; Berry, Neil G; Sharma, Raman; Stocks, Paul A; Srivastava, Abhishek; Shone, Alison E; Charoensutthivarakul, Sitthivut; Taylor, Lee; Berger, Olivier; Mbekeani, Alison; Hill, Alasdair; Fisher, Nicholas E; Warman, Ashley J; Biagini, Giancarlo A; Ward, Stephen A; O'Neill, Paul M

Identification of novel antimalarial chemotypes via chemoinformatic compound selection methods for a high-throughput screening program against the novel malarial target, PfNDH2: increasing hit rate via virtual screening methods.

通过化学信息学化合物选择方法鉴定新型抗疟疾化学类型,用于针对新型疟疾靶点 PfNDH2 的高通量筛选程序:通过虚拟筛选方法提高命中率

Sharma Raman, Lawrenson Alexandre S, Fisher Nicholas E, Warman Ashley J, Shone Alison E, Hill Alasdair, Mbekeani Alison, Pidathala Chandrakala, Amewu Richard K, Leung Suet, Gibbons Peter, Hong David W, Stocks Paul, Nixon Gemma L, Chadwick James, Shearer Joanne, Gowers Ian, Cronk David, Parel Serge P, O'Neill Paul M, Ward Stephen A, Biagini Giancarlo A, Berry Neil G

HDQ, a potent inhibitor of Plasmodium falciparum proliferation, binds to the quinone reduction site of the cytochrome bc1 complex.

HDQ 是一种强效的恶性疟原虫增殖抑制剂,它与细胞色素 bc1 复合物的醌还原位点结合

Vallières Cindy, Fisher Nicholas, Antoine Thomas, Al-Helal Mohammed, Stocks Paul, Berry Neil G, Lawrenson Alexandre S, Ward Stephen A, O'Neill Paul M, Biagini Giancarlo A, Meunier Brigitte

The molecular basis of folate salvage in Plasmodium falciparum: characterization of two folate transporters.

恶性疟原虫叶酸补救的分子基础:两种叶酸转运蛋白的特征

Salcedo-Sora J Enrique, Ochong Edwin, Beveridge Susan, Johnson David, Nzila Alexis, Biagini Giancarlo A, Stocks Paul A, O'Neill Paul M, Krishna Sanjeev, Bray Patrick G, Ward Stephen A

Modeling the trade-off between effective case management and imported malaria cases in different settings of P. falciparum malaria transmission intensity

在不同恶性疟原虫疟疾传播强度环境下,建立有效病例管理与输入性疟疾病例之间权衡模型

Billingsley, Peter F; Storm, Janet; Müller, Sylke; Batwala, Vincent; Magnussen, Pascal; Nuwaha, Fred; Dahlbäck, Madeleine; Jørgensen, Lars M; Christoffersen, Stig; Nielsen, Morten A; Theander, Thor G; Arnot, David E; Larsen, Sine; Salanti, Ali; Sibley, Carol Hopkins; Liu, Weimin; Li, Yingying; Learn, Gerald H; Rudicell, Rebecca S; Robertson, Joel D; Keele, Brandon F; Ndjango, Jean-Bosco N; Sanz, Crickette M; Morgan, David B; Locatelli, Sabrina; Gonder, Mary K; Kranzusch, Philip J; Walsh, Peter D; Delaporte, Eric; Mpoudi-Ngole, Eitel; Georgiev, Alexander V; Muller, Martin N; Shaw, George M; Peeters, Martine; Sharp, Paul M; Rayner, Julian C; Hahn, Beatrice H; Deplaine, Guillaume; Safeukui, Innocent; Jeddi, Fakhri; Lacoste, François; Brousse, Valentine; Perrot, Sylvie; Biligui, Sylvestre; Guillotte, Micheline; Guitton, Corinne; Dokmak, Safi; Aussilhou, Béatrice; Sauvanet, Alain; Couvelard, Anne; Paye, François; Thellier, Marc; Mazier, Dominique; Milon, Geneviève; Mohandas, Narla; Puijalon, Odile Mercereau; David, Peter H; Buffet, Pierre A; Di Pasquale, Aurelio; Maire, Nicolas; Smith, Thomas; Jean-Bernard, Duchemin; Cyrille, Czeher; Rabiou, Labbo; Lamine, Ibrahim M; Stefan, Hoyer; Isabelle, Jeanne; Maude, Richard James; Sayeed, Abdullah Abu; Beare, Nicholas AV; Charunwatthana, Prakaykaew; Faiz, Abul M; Hossain, Amir; Yunus, Emran Bin; Hoque, Gofranul M; Hasan, Mahtab Uddin; White, Nicholas J; Day, Nicholas PJ; Dondorp, Arjen M; Mota, Maria M; Staines, Henry; Assogba, Benoît S; Djogbenou, Luc S; Dabiré, Roch K; Diabaté, Abdoulaye; Baldet, Thierry; Fatih, Farrah A; Siner, Angela; Ahmed, Atique; Woon, Lu Chan; Craig, Alister; Staines, Henry M; Singh, Balbir; Krishna, Sanjeev; Cox-Singh, Janet; Felger, Ingrid; Schoepflin, Sonja; Kiniboro, Benson; Zimmerman, Peter A; Mueller, Ivo; Gholizadeh, Saber; Karimi, Ameneh; Bayat, Nooshin; Djadid, Navid Dinparast; Zakeri, Sedigheh; Rodrigues, Louise A; Henriques, Gisela; Borges, Sofia T; Hunt, Paul; Sanchez, Cecília P; Martinelli, Axel; Cravo, Pedro; Martins, Joao; Zwi, Anthony; Kelly, Paul; Niemand, J; Birkholtz, L; Louw, AI; Kirk, K; Riglar, David; Richard, Dave; Boyle, Michelle; Wilson, Danny; Angrisano, Fiona; Turnbull, Lynne; Whitchurch, Cynthia; Cowman, Alan; Beeson, James; Ralph, Stuart; Baum, Jake; Kapulu, Melissa C; Biswas, Sumi; Blagborough, Andrew; Gilbert, Sarah C; Sinden, Robert E; Hill, Adrian VS; Jones, Matthew L; Collins, Mark O; Choudhary, Jyoti; Rayner, Julian C; Kaiser, Marco; Bray, Dorothy H; Zommers, Zinta; Couacy-Hymann, Emmanuel; Gillespie, Thomas R; Ellerbrok, Heinz; Leendertz, Fabian H; Gouagna, Louis C; Bancone, Germana; Yao, Frank; Costantini, Carlo; Ouedraogo, Jean-Bosco; Modiano, David; Hulden, Lena; Tanabe, Kazuyuki; Mita, Toshihiro; Balloux, Francois; Saeed, Sadia; Tremp, Annie Z; Dessens, Johannes T; Skorokhod, Oleksii A; Caione, Luisa; Migliardi, Giorgia; Barrera, Valentina; Piacibello, Wanda; Schwarzer, Evelin; Arese, Paolo; Smallegange, Renate C; Schmied, Wolfgang H; van Roey, Karel J; Verhulst, Niels O; Spitzen, Jeroen; Mukabana, Wolfgang R; Takken, Willem; Marin-Menendez, Alejandro; Bell, Angus; Biagini, Giancarlo A; Hill, Alasdair; Mbekeani, Alison; Shone, Alison; Nixon, Gemma; Stocks, Paul; Gibbons, Peter; Amewu, Richard; Hong, David W; Barton, Victoria; Pidathala, Chandra; Chadwick, James; Le Pensee, Louise; Warman, Ashley; Sharma, Raman; Fisher, Nick; Berry, Neil G; O'Neill, Paul M; Ward, Steve A; Brooke, Basil D; Kaiser, Maria L; Koekemoer, Lizette L; Coetzee, Maureen; Hunt, Richard H; Burgess, Steven J; Xu-Kelly, Jane; Liebmann, Katherine; Gunsaru, Bornface; Morrill, Westin; Peyton, David H; Chitnis, Nakul; Hardy, Diggory; Gnaegi, Guillaume; Boutsika, Konstantina; Maire, Nicolas; Steketee, Richard; Schapira, Allan; Smith, Tom; Tang, Jianxia; Inoue, Megumi; Sunahara, Toshihiko; Kanda, Moe; Kaneko, Osamu; Culleton, Richard; van Brummlen, Tharina; Becker, John VW; Mancama, Dalu T; Hoppe, Heinrich; Crosnier, Cecile; Wanaguru, Madushi; McDade, Brian; Rayner, Julian; Wright, Gavin J; de Oliveira, Alaíde Braga; Dolabela, Maria Fâni; Póvoa, Marinete Marins; Santos, Cid Aimbiré M; de Pilla Varotti, Fernando; Afolabi, Bamgboye M; Dunkwu, Antonia; Oparah, A C; Filipe, Ermelindo M; Antunes, Lina; Tomás, Esmael F; Viegas, Edna; Bernardo, João; Silva, Fortunato R; Tripathi, Abhai; Rienhoff, Hugh; Sullivan, David; Udagama-Randeniya, Preethi; Dias, Sajani; Premaratne, Prasad; Wickramarachchi, Thilan; Waitumbi, John; Nyakoe, Nancy; Muringo, Linda; Mahat, Ismail; Otiende, Moses; Susanna, Dewi; Eryando, Tris; Temidayo, Soniran O; Olufunmilayo, Idowu; Babatunde, Idowu A; Olusegun, Ajana; Tomás, Esmael; Filipe, E; Viegas, E; Sá, A; Silva, F; Antunes, L; Lafuente, E; Tonwong, Natda; Sattabongkot, Jetsumon; Sirichaisinthop, Jeeraphat; Udomsangpetch, Rachanee; Spjeldnæs, Astrid; Blomberg, Bjørn; Ginsburg, Hagai; Inoue, Megumi; Tang, Jianxia; Kaneko, Osamu; Yui, Katsuyuki; Culleton, Richard; Aubouy, Agnès; Kheliouen, Nabila; Tuikue-Ndam, Nicaise; Viwami, Firmine; Lalya, Francis; Eboumbou Moukoko, Else C; Rogier, Christophe; Deloron, Philippe; Omoregie, Ehimwenma S; Pal, Anirban; Darokar, Mahendra P; Chanda, Debabrata; Sisodia, Brijesh; Mogendi, Shem Oroo; Osman, Mamoun MM; Nour, Bakri YM; Sedig, Mohamed F; de Bes, Laura; Babikir, Adil M; Mohamedani, Ahmed A; Mens, Petra F; Ouédraogo, Alphonse; Coulibaly, Sheick O; Diarra, Amidou; Traoré, Abdoulaye; Sirima, Sodiomon B; Magnussen, Pascal; Ball, Elizabeth; Gonçalves, Carlos Penha; Pooe, Ofentse J; Shonhai, Addmore; Mharakurwa, Sungano; Roobsoong, Wanlapa; Roytrakul, Sittiruk; Kiatfuengfoo, Rachada; Nuchpramool, Wilairat; Cui, Liwang; Udomsangpetch, Rachanee; Schneider, Petra; Bell, Andy S; Read, Andrew F; Reece, Sarah E; Singh, Gavendra; Prakash, Soam; Siri, José G; Brown, Zachary; Spielauer, Martin; Rajasekariah, G-Halli R; Dogcio, Diane; Lee, Rogan; Hudson, Bernard J; Mazure, Hubert G; Smithyman, Anthony M; Rankin, Kathleen E; Tavares, Joana; Struck, Nicole S; Menard, Robert; Heussler, Volker T; Amino, Rogerio; Riglar, David; Richard, Dave; Boyle, Michelle; Wilson, Danny; Angrisano, Fiona; Turnbull, Lynne; Whitchurch, Cynthia; Cowman, Alan; Beeson, James; Ralph, Stuart; Baum, Jake; Rodrigues, Louise A; Henriques, Gisela; Cravo, Pedro; Prato, Mauro; Ulliers, Daniela; Gallo, Valentina; Schwarzer, Evelin; Akide-Ndunge, Oscar B; Mandili, Giorgia; Khadjavi, Amina; Saviozzi, Silvia; Calogero, Raffaele A; Arese, Paolo; Giribaldi, Giuliana; Bansal, Devendra; Herbert, Fabien; Deshpande, Prakash; Bécavin, Christophe; Guiyedi, Vincent; de Maria, Ilaria; Cazenave, Pierre-André; Mishra, Gyan Chandra; Ferlini, Cristiano; Fesel, Constantin; Benecke, Arndt; Pied, Sylviane; Hamid, Muzamil Mahdi Abdel; Remarque, Edmond J; Faber, Bart W; van Duivenvoorde, Leonie M; Kocken, Clemens HM; Thomas, Alan W; Houzé, Sandrine; Hubert, Véronique; Cohen, Pressler D; Rivetz, Baruch; Le Bras, Jacques; Jones, Matthew L; Collins, Mark O; Choudhary, Jyoti S; Rayner, Julian C; Koekemoer, Lizette L; Spillings, Belinda S; Christian, Riann; Wood, Oliver S; Kaiser, Maria; Norton, Ryan; Choi, Kwang S; Brooke, Basil D; Hunt, Richard H; Coetzee, Maureen; Gitau, Grace; Shonhai, Addmore; Dean Goldring, J P; Hurdayal, Ramona; Choveaux, David; Liehl, Peter; Prudêncio, Miguel; Carret, Céline; Mota, Maria M; Akter, Jasmin; Ahmed, Sabeena; Prue, Chai; Khan, Wasif; Sack, David; Haque, Rashidul; Sullivan, David; Kabanywany, Abdunoor Mulokozi; Mulure, Nathan; Migoha, Christopher; Malila, Aggrey; Lengeler, Christian; Schlienger, Raymond; Genton, Blaise; Niemand, J; Birkholtz, L; Louw, A I; Kirk, K; Ogonda, Lilian A; Orago, Alloys SS; Otieno, Michael F; Adhiambo, Christine; Otieno, Walter; Stoute, José A; Sutherland, Colin J; Oguike, Mary C; Smith, Valerie; Betson, Martha; Bousema, Teun; Chiodini, Peter L; Wells, Timothy NC; Takken, Willem; Cox-Singh, Janet; Crabb, Brendan; Bullen, Hayley; Charnaud, Sarah; Haase, Silvia; Boddey, Justin; Cowman, Alan; de Koning-Ward, Tania; Gilson, Paul; Tanner, Marcel; Alonso, Pedro L; van den Berg, Henk; Takken, Willem; Van den Steen, Philippe E; Geurts, Nathalie; Deroost, Katrien; Van Aelst, Ilse; Verhenne, Sebastien; Heremans, Hubertine; Van Damme, Jo; Opdenakker, Ghislain; Ward, Steve A; Fisher, Nicholas; Hill, Alasdair; Mbekeani, Alison; Shone, Alison; Nixon, Gemma; Stocks, Paul; Gibbons, Peter; Amewu, Richard; Hong, David W; Barton, Victoria; Pidathala, Chandra; Chadwick, James; Le Pensee, Louise; Warman, Ashley; Sharma, Raman; Berry, Neil G; O'Neill, Paul M; Biagini, Giancarlo A; Oyeyemi, Adebusola O; Alawode, Abdul-Gafar; Sogunro, Remi; Panichakul, Tasanee; Payuhakrit, Witchuda; Wongborisuth, Chokdee; Hongeng, Suradej; Udomsangpetch, Rachanee; Parikh, Ravi; Amole, Isaac; Tarpley, Margaret; Gbadero, Daniel; Davidson, Mario; Vermund, Sten H; Patzewitz, Eva-Maria; Müller, Sylke; Noor, Ramadhani A; Thiesen, Michael; Mordmuller, Benjamin; Milligan, Paul; Atuguba, Frank; Sirima, Sodiomon; Issifou, Saadou; Bojang, Kalifa; Kironde, Fred; Tiono, Alfred; Okech, Brenda; Chilengi, Roma; Ngoa, Ateba; Mukasa, Kaddu; Jepsen, Soren; Ochola, Lucy B; Siddondo, Bethsheba R; Ocholla, Harold; Nyka, Siana; Kimani, Eva N; Williams, Thomas N; Makale, Johnstone O; Liljander, Anne; Urban, Britta C; Bull, Pete; Szestak, Tadge; Marsh, Kevin; Craig, Alister G; Malisa, Allen; Pearce, Richard; Abdullah, Salim; Mshinda, Hassan; Kachur, Patrick; Bloland, Peter; Roper, Cally; Mbugi, Erasto V; Meijerink, Marjolein; Veenemans, Jacobien; Jeurink, Prescilla V; McCall, Matthew; Olomi, Raimos M; Shao, John F; Chilongola, Jaffu O; Verhoef, Hans; Savelkoul, Huub FJ; Mirghani, Samia E; Nour, Bakri YM; Bushra, Sayed M; Hassan, Ibrahim El; Snow, Robert W; Noor, Abdisalan M; Mnyone, Ladslaus L; Lyimo, Issa N; Lwetoijera, Dickson W; Mpingwa, Monica W; Nchimbi, Nuru; Hancock, Penny; Russell, Tanya L; Kirby, Matthew J; Takken, Willem; Koenraadt, Constantianus JM; Odhiambo, Collins O; Otieno, Walter; Adhiambo, Christine; Odera, Michael M; Stoute, José A; Ferrer, Jordi; Prats, Clara; López, Daniel; Valls, Joaquim; Gargallo, Domingo; Wijayalath, Wathsala; Cheesman, Sandie; Rajakaruna, Jagath; Weerasinghe, Sudath; Kapilananda, Gamini; Gamage, Kamal; Perera, Kamal; Handunnetti, Shiroma; Carter, Richard; Pathirana, Sisira; Wanjala, Christine L; Githeko, Andrew K; Waitumbi, John N; Gomes-Santos, Carina SS; Braks, J Anneke M; Prudêncio, Miguel; Carret, Céline K; Gomes, Ana Rita; Pain, Arnab; Feltwell, Theresa; Khan, Shahid M; Waters, Andrew P; Janse, Chris J; Mair, Gunnar R; Mota, Maria M; Kyabayinze, Daniel J; Asiimwe, Caroline; Nakanjako, Damalie; Nabakooza, Jane; Counihan, Helen; Tibenderana, James K; Donegan, G; Forrester, C A; Ward, S A; Boyom, Fabrice F; Madiesse, Eugénie K; Bankeu, Jean J; Tsouh, Valere P; Lenta, Bruno N; Mbacham, Wilfred F; Tsamo, Etienne; Zollo, Paul HA; Gut, Jiri; Rosenthal, Philip J; Yoon, Ho Sup; Alag, Reema; Kang, Congbao; Ye, Hong; Kotaka, Masayo; Qureshi, Insaf A; Bharatham, Nagakumar; Shin, Joon; Bozdech, Zbynek; Preiser, Peter; Lescar, Julien; Wanaguru, Madushi; Wright-Crosnier, Cecile; Bustamante, Leyla; McDade, Brian; Rayner, Julian; Wright, Gavin J; Crowell, Valerie; Hardy, Diggory; Chitnis, Nakul; Maire, Nicolas; Smith, Thomas

PfCRT and the trans-vacuolar proton electrochemical gradient: regulating the access of chloroquine to ferriprotoporphyrin IX.

PfCRT 和跨液泡质子电化学梯度:调节氯喹与铁原卟啉 IX 的接触

Bray Patrick G, Mungthin Mathirut, Hastings Ian M, Biagini Giancarlo A, Saidu Dauda K, Lakshmanan Viswanathan, Johnson David J, Hughes Ruth H, Stocks Paul A, O'Neill Paul M, Fidock David A, Warhurst David C, Ward Stephen A