日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural Analysis of 23S rRNA Methylating Enzyme Cfr Reveals RNA-Binding Determinants for Methylation Regiospecificity and Antibiotic Resistance

23S rRNA甲基化酶Cfr的结构分析揭示了甲基化区域特异性和抗生素耐药性的RNA结合决定因素

Fruci, Michael; Rodríguez Hernández, Annia; Skarina, Tatiana; Verellen, Lou Ann; Tsai, Kaitlyn; Virta, Johanna M; Fujimori, Danica Galonić; Savchenko, Alexei; Stogios, Peter J

Structure-guided optimization of small molecules targeting Yck2 as a strategy to combat Candida albicans

以Yck2为靶点的小分子结构导向优化作为对抗白色念珠菌的策略

Puumala, Emily; Nandakumar, Meganathan; Yiu, Bonnie; Stogios, Peter J; Strickland, Benjamin G; Zarnowski, Robert; Wang, Xiaoyu; Williams, Noelle S; Savchenko, Alexei; Andes, David R; Robbins, Nicole; Whitesell, Luke; Willson, Timothy M; Cowen, Leah E

Structural and functional insights into extreme thermal stability and activity of two GH12 domains of a multidomain glycosidase from a hyperthermophilic euryarchaeon.

对嗜热古菌多结构域糖苷酶的两个 GH12 结构域的极端热稳定性和活性的结构和功能进行了深入研究

Zayulina Kseniya S, Frolov Evgenii N, Stracke Christina, Klyukina Alexandra A, Khusnutdinova Anna N, Stogios Peter, Skarina Tatiana, Yakunin Alexander F, Golyshin Peter N, Siebers Bettina, Shugaeva Tatiana E, Kublanov Ilya V

Structural and functional analyses of SARS-CoV-2 Nsp3 and its specific interactions with the 5' UTR of the viral genome

对SARS-CoV-2 Nsp3的结构和功能分析及其与病毒基因组5'非翻译区的特异性相互作用

Lemak, Sofia; Skarina, Tatiana; Patel, Deepak T; Stogios, Peter J; Savchenko, Alexei

Structural analysis of extracellular ATP-independent chaperones of streptococcal species and protein substrate interactions

链球菌胞外ATP非依赖性分子伴侣的结构分析及其与蛋白质底物的相互作用

Agbavor, Charles; Torres, Madeline; Inniss, Nicole L; Latimer, Sarah; Minasov, George; Shuvalova, Ludmilla; Wawrzak, Zdzislaw; Borek, Dominika; Otwinowski, Zbyszek; Stogios, Peter J; Savchenko, Alexei; Anderson, Wayne F; Satchell, Karla J F; Cahoon, Laty A

Structural genomics of bacterial drug targets: Application of a high-throughput pipeline to solve 58 protein structures from pathogenic and related bacteria

细菌药物靶点的结构基因组学:应用高通量流程解析致病菌及相关细菌的58个蛋白质结构

Inniss, Nicole L; Minasov, George; Chang, Changsoo; Tan, Kemin; Kim, Youngchang; Maltseva, Natalia; Stogios, Peter; Filippova, Ekaterina; Michalska, Karolina; Osipiuk, Jerzy; Jaroszewki, Lukasz; Godzik, Adam; Savchenko, Alexei; Joachimiak, Andrzej; Anderson, Wayne F; Satchell, Karla J F

Structure-guided optimization of small molecules targeting the yeast casein kinase, Yck2, as a therapeutic strategy to combat Candida albicans

以酵母酪蛋白激酶Yck2为靶点的小分子结构导向优化,作为对抗白色念珠菌的治疗策略

Cowen, Leah; Puumala, Emily; Nandakumar, Meganathan; Yiu, Bonnie; Stogios, Peter; Strickland, Benjamin; Zarnowski, Robert; Wang, Xiaoyu; Williams, Noelle; Savchenko, Alexei; Andes, David; Robbins, Nicole; Whitesell, Luke; Willson, Timothy

Structural analysis of 23S rRNA methylating enzyme Cfr reveals RNA binding determinants for methylation regiospecificity and antibiotic resistance

对 23S rRNA 甲基化酶 Cfr 的结构分析揭示了其甲基化区域特异性和抗生素耐药性的 RNA 结合决定因素。

Fruci, Michael; Rodríguez Hernández, Annia; Skarina, Tatiana; Verellen, Lou Ann; Tsai, Kaitlyn; Virta, Johanna M; Fujimori, Danica Galonić; Savchenko, Alexei; Stogios, Peter J

Structure-activity Relationship for Diarylpyrazoles as Inhibitors of the Fungal Kinase Yck2.

二芳基吡唑类化合物作为真菌激酶Yck2抑制剂的构效关系

Shirley David J, Yiu Bonnie, Mancera-Ortiz Ikeer, Stogios Peter J, Liu Zhongle, Robbins Nicole, Whitesell Luke, Cowen Leah E, Drewry David H, Willson Timothy M

Computation-guided transcription factor biosensor specificity engineering for adipic acid detection

利用计算引导的转录因子生物传感器特异性工程设计检测己二酸

Pham, Chester; Stogios, Peter J; Savchenko, Alexei; Mahadevan, Radhakrishnan