日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Small molecule-constrained paratope mimetic bicyclic peptides as potent inhibitors of group 1 and 2 influenza A virus hemagglutinins

小分子约束的互补位模拟双环肽作为1组和2组甲型流感病毒血凝素的强效抑制剂

Kadam, Rameshwar U; Juraszek, Jarek; Brandenburg, Boerries; Garg, Divita; Zhu, Xueyong; Jongeneelen, Mandy; Tang, Chan; Schepens, Wim B G; Buyck, Christophe; Stoops, Bart; Vermond, Jan; Vogels, Ronald; Friesen, Robert H E; van Dongen, Maria J P; Wilson, Ian A

Menaquinone depletion resensitises bedaquiline-resistant tuberculosis

甲萘醌耗竭可使耐贝达喹啉结核病重新敏感

Wetzel, Jennefer; Dallow, John; Davis, Ellie; Pearson, William H; Daems, Stijn; Govaerts, Matthias; Hereijgers, Joyce; Sprangers, Joke; Truebody, Barry; Maes, Valerie; van Hasselt, Vera; Leemans, Annelies; Pujari, Venugopal; Vos, Ann; Viturro, Carlos M Martínez; Gómez, José Enrique; Peeters, Mirte; Gerber, Michelle; Chhabra, Nandini; Wouters, Annelies; Everaerts, Melissa; Painter, Hannah; Fathima, Raisha; Willcocks, Sam J; Davies, Cadi; Raeymaekers, Valerie; Clark, Taane G; Draghia-Akli, Ruxandra; Fletcher, Helen; Van Loock, Marnix; Hibberd, Martin L; Mostowy, Serge; Crick, Dean C; Pym, Alexander S; Samby, Kirandeep; Jackson, Paul; Trabanco, Andrés A; Larrouy-Maumus, Gerald; Steyn, Adrie J C; Stoops, Bart; Dhar, Neeraj; Aguilar-Pérez, Clara; Lamprecht, Dirk A; Wall, Richard J; Koul, Anil

Targeting de novo purine biosynthesis for tuberculosis treatment

靶向嘌呤从头合成治疗结核病

Lamprecht, Dirk A; Wall, Richard J; Leemans, Annelies; Truebody, Barry; Sprangers, Joke; Fiogbe, Patricia; Davies, Cadi; Wetzel, Jennefer; Daems, Stijn; Pearson, William; Pillay, Vanessa; Saylock, Samantha; Ricketts, M Daniel; Davis, Ellie; Huff, Adam; Grell, Tsehai; Lin, Shiming; Gerber, Michelle; Vos, Ann; Dallow, John; Willcocks, Sam J; Roubert, Christine; Sans, Stéphanie; Desorme, Amandine; Chappat, Nicolas; Ray, Aurélie; Pereira Moraes, Mariana; Washington, Tracy; D'Erasmo, Hope; Sancheti, Pavankumar; Everaerts, Melissa; Monshouwer, Mario; Esquivias, Jorge; Larrouy-Maumus, Gerald; Draghia Akli, Ruxandra; Fletcher, Helen; Pym, Alexander S; Aldridge, Bree B; Sarathy, Jansy P; Clancy, Kathleen W; Stoops, Bart; Dhar, Neeraj; Steyn, Adrie J C; Jackson, Paul; Aguilar-Pérez, Clara; Koul, Anil

The role of cytochrome bc(1) inhibitors in future tuberculosis treatment regimens

细胞色素bc(1)抑制剂在未来结核病治疗方案中的作用

Aguilar-Pérez, Clara; Lenaerts, Anne J; Villellas, Cristina; Guillemont, Jerome; Dallow, John; Painter, Hannah; Ammerman, Nicole C; Hassan, Anis; Golovkine, Guillaume; Brock, Laure; Sordello, Sylvie; Chauffour, Aurélie; Aubry, Alexandra; Mai, Thi Cuc; Wong, Sarah; Clark, Taane G; Nam, Kiyean; Kim, Jeongjun; Choi, Jinho; Crabbe, Marjolein; Esquivias, Jorge; Lounis, Nacer; Stoops, Bart; Amssoms, Katie; Bartolome-Nebreda, Jose M; Gruppo, Veronica; Robertson, Gregory T; Veziris, Nicolas; Upton, Anna M; Nuermberger, Eric L; Cox, Vivian; Ballell, Lluis; Baeten, Benny; Koul, Anil; Pym, Alexander S; Wall, Richard J; Lamprecht, Dirk A

Discovery of a non-nucleoside inhibitor that binds to a novel site in the palm domain of the respiratory syncytial virus RNA-dependent RNA polymerase.

发现一种非核苷类抑制剂,可与呼吸道合胞病毒 RNA 依赖性 RNA 聚合酶掌状结构域中的新位点结合

Kalin Jay H, Yin Yanting, Tran Minh T, Piassek Madison, Fung Amy, Grosse Sandrine, Jacoby Edgar, Bhaumik Anusarka, Adhikary Suraj, Miller Robyn, Lemmens Cynthia, Lutter Ferdinand H, Pieters Serge, Cooymans Ludwig, Rombouts Geert, Oehlrich Daniel, Tomaso Sonia, Lozada Kate, Garcia Miguel Osorio, Anson Brandon, De Bruyn Suzanne, Smith-Monroy Constance, Neefs Jean-Marc, Conceição-Neto Nádia, Stoops Bart, van Vlijmen Herman, Patrick Aaron, Yu Xiaodi, Wong Victoria, Krosky Daniel, Abeywickrema Pravien, Mason Stephen, Jin Zhinan, Jonckers Tim H M, Sharma Sujata

V(H)H antibody loop guides design of a synthetic macrocyclic peptide that potently blocks influenza virus membrane fusion

V(H)H抗体环指导合成大环肽的设计,该大环肽能有效阻断流感病毒膜融合。

Kadam, Rameshwar U; Juraszek, Jarek; Brandenburg, Boerries; Garg, Divita; Zhu, Xueyong; Jongeneelen, Mandy; Schepens, Wim B G; Stoops, Bart; Vermond, Jan; Goutier, Wouter; Tang, Chan; Blokland, Sven; Vogels, Ronald; Friesen, Robert H E; van Dongen, Maria J P; Wilson, Ian A

Potent peptidic fusion inhibitors of influenza virus

流感病毒的强效肽融合抑制剂

Kadam, Rameshwar U; Juraszek, Jarek; Brandenburg, Boerries; Buyck, Christophe; Schepens, Wim B G; Kesteleyn, Bart; Stoops, Bart; Vreeken, Rob J; Vermond, Jan; Goutier, Wouter; Tang, Chan; Vogels, Ronald; Friesen, Robert H E; Goudsmit, Jaap; van Dongen, Maria J P; Wilson, Ian A