Ugi-Tetrazole-Derived α‑Aminomethyl Scaffolds Reveal Unexpected Binding Modes in SARS-CoV‑2 3CLpro
Ugi-四唑衍生的α-氨甲基骨架揭示了SARS-CoV-2 3CLpro中意想不到的结合模式
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00773
van der Straat, Robin; Oerlemans, Rick; Cong, Yingying; Boxma, Jeffrey; Bulai, Radu G; Río-Bergé, Clàudia; Koekemoer, Lizbé; Zarganes Tzitzikas, Tryfon; Guan, Zhirui; Marples, Peter George; Reggiori, Fulvio; Groves, Matthew; Dömling, Alexander